The catecholamines, in particular norepinephrine and epinephrine, are targets of the G protein-coupled receptor class known as adrenergic receptors. These receptors are found on numerous cells, and when a catecholamine binds to one of these receptors, the sympathetic nervous system is typically stimulated. The fight-or-flight response is controlled by the sympathetic nervous system, which causes the eye pupils to dilate, the body to mobilize energy, and the blood supply to skeletal muscle to be diverted from non-essential organs.There are numerous subtypes of the two main groups of adrenergic receptors, and. The receptor subtypes 1 and 2 exist. There are three subtypes of receptors: 1, 2, and 3. They are all associated with Gs proteins, which are associated with adenylate cyclase. Thus, antagonist binding increases the level of the second messenger cAMP inside of the cell. The cAMP-dependent protein kinase (PKA), one of cAMP's downstream effectors, mediates some intracellular processes after hormone binding.
| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V1137 | Prazosin HCl | 19237-84-4 | Prazosin HCl (Furazosin, cp12299-1; cp-12299-1; Minipress, Peripress), the hydrochloride salt of prazosin, is a potent and competitive alpha-1 adrenoceptor antagonist with antihypertensive effects. |
|
V71247 | Prazosin-d8 (prazosin-d8) | 1006717-55-0 | Prazosin-d8 is the deuterated form of Prazosin. |
|
V71248 | Procaterol hydrochloride hemihydrate (OPC 2009 hydrochloride hemihydrate) | 81262-93-3 | Procaterol HCl hemihydrate is an orally bioactive β2 adrenoreceptor agonist (activator). |
|
V1152 | Propranolol HCl (AY64043, ICI45520, NCS91523) | 318-98-9 | Propranolol HCl (formerly ICI-45520, NCS-91523; AY-64043; Inderal among others), the hydrochloride salt of Propranolol, is a competitive and non-selective inhibitor of beta-adrenergic receptors with antihypertensive effects. |
|
V71244 | Propranolol-d7 (propranolol d7) | 98897-23-5 | Propranolol-d7 is the deuterated form of Propranolol. |
|
V71243 | Propranolol-d7 (ring-d7) | 344298-99-3 | Propranolol-d7 (ring-d7) is the deuterated form of Propranolol HCl. |
|
V71350 | Ractopamine | 97825-25-7 | Ractopamine is a potent β-adrenergic receptor (βAR) agonist/activator with a Kd of approximately 25 nM for porcine β1AR and β2AR. |
|
V71284 | Rauwolscine (α-Yohimbine; Corynanthidine; Isoyohimbine) | 131-03-3 | Rauwolscine is a selective α2-adrenoceptor antagonist that can inhibit tumor growth and cause apoptosis. |
|
V2433 | Reboxetine mesylate (FCE20124; PNU155950E) | 98769-84-7 | Reboxetine (also known as PNU 155950E; Trade name: Edronax)is a selective norepinephrine reuptake inhibitor with Ki of 8.2 nM and antidepressant activity. |
|
V8519 | Ritanserin | 87051-43-2 | Ritanserin (R55667; R-55667) is a novel, potent, andlong acting antagonist of serotonin-2 (5-HT2) receptor with an IC50 of 0.9 nM. |
|
V1118 | Ritodrine HCl (DU21220 HCl) | 23239-51-2 | Ritodrine HCl (DU21220; DU21220; ST51015115; ST-51015115; Pre-Par; Utopar), the hydrochloride salt of ritodrine, is a β-2 adrenergic receptor agonist used to treat premature labor. |
|
V71241 | Ro 363 hydrochloride | 250580-70-2 | Ro 363 HCl, a potent inotropic activator, is a potent and selective β1-adrenoceptor agonist. |
|
V71306 | Romifidine hydrochloride | 65896-14-2 | Romifidine HCl is an α2-adrenoceptor agonist. |
|
V1095 | Salbutamol Sulfate (AH-3365; Albuterol) | 51022-70-9 | Salbutamol Sulfate (AH-3365; AH3365; trade name Ventolin among others) is a potent, selective and short-acting β2-adrenergic receptor agonist with the potential to relax airway smooth muscles. |
|
V71268 | Salbutamol-d3 (Albutamol-d3; Albuterol-d3; AH-3365-d3) | 1219798-60-3 | Salbutamol-d3 is the deuterated form of Salbutamol. |
|
V71288 | Salbutamol-d9 acetate (Albuterol-d9 acetate; AH-3365-d9 acetate) | 1781417-68-2 | Salbutamol-d9 (acetate) is the deuterated form of Salbutamol. |
|
V1101 | Salmeterol Xinafoate (GR 33343X xinafoate) | 94749-08-3 | Salmeterol Xinafoate (GR-33343G,AHR-3929; AH-3923; Salmetedur, Serevent), theXinafoate salt of Salmeterol,is a potent and long-acting β2-adrenergic receptor agonist with anti-inflammatory effects. |
|
V71254 | Salmeterol-d3 | 497063-94-2 | Salmeterol-d3 is a deuterated form of Salmeterol. |
|
V81353 | Salmeterol-d3 xinafoate (GR 33343X-d3 (xinafoate)) | Salmeterol-d3 (xinafoate) is the deuterated form of Salmeterol xinafoate. | |
|
V1156 | Scopine | 498-45-3 | Scopine (6,7-Epoxytropine), ametabolite of scopolamine and anisodine (an α1-adrenergic receptor agonist), is a naturally occurring tropane alkaloid extracted from various plants such as Scopolia carniolica, Mandragora root, Senecio mikanoides (Delairea odorata), and Scopolia lurida. |
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