| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V1168 | 5-hydroxymethyl tolterodine (PNU 200577) | 207679-81-0 | 5-hydroxymethyl tolterodine (Desfesoterodine, PNU 200577,PNU-200577, 5HMT, 5HM;5-HMT, 5-HM), the active metabolite of tolterodine which is a medicationused treat overactive bladder, is a novel and potent muscarinic receptor antagonist with a Kb of 0.84 nM. |
|
V15400 | Encenicline HCl salt (EVP6124; MT4666) | 550999-74-1 | Encenicline (EVP-6124; MT-4666) is a novel partial agonist of α7 nicotinic acetylcholine receptor. |
|
V1165 | LY2119620 | 886047-22-9 | LY2119620 (LY 2119620; LY-2119620) is a novel, potent, specific, high-affinity and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors, the so called positive allosteric modulator (PAM). |
|
V1191 | PNU-120596 (NSC-216666) | 501925-31-1 | PNU-120596 (PNU120596;NSC 216666;PNU 120596;NSC-216666)is a potent and selective PAM (positive allosteric modulator) of α7 nAChR (acetylcholine receptor) with an EC50 of 216 NM. |
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V1174 | Solifenacin succinate (YM905) | 242478-38-2 | Solifenacinsuccinate (formerly YM-905; YM905;Trade name: Vesikur; Vesicare), the succinate salt of solifenacin which is approved for treating overactive bladder, is a novel and potent muscarinic receptor antagonist withpKis of 7.6, 6.9 and 8.0 forM1,M2andM3receptors, respectively. |
|
V17279 | Butylscopolamine bromide | 149-64-4 | Butylscopolamine bromide is a potent antimuscarinic quaternary ammonium analogue acting as a competitive antagonist of mAChR (IC50: 55.3 ± 4.3 nM). |
|
V5514 | Scopolamine | 51-34-3 | Scopolamine (Hyoscine) isan approved medication used to treat motion sickness and postoperative nausea and vomiting. |
|
V0034 | Scopolamine HBr (Hyoscine) | 114-49-8 | Scopolamine HBr, also known as Hyoscine, is the hydrobromide salt of scopolamine which is a competitive and non-selective antagonist of muscarinic acetylcholine receptor with an IC50 of 55.3 nM. |
|
V1195 | Diphemanil Methylsulfate | 62-97-5 | Diphemanil methylsulfate (NSC 41725; NSC-41725; Prantal; Talpran; Diphemanil mesylate) is a quaternary ammonium anticholinergic agent used for a variety of conditions such as pylorospasm,peptic ulcer, gastric hyperacidity, hypermotility in gastritis, and hyperhidrosis. |
|
V1201 | Hexamethonium Bromide | 55-97-0 | Hexamethonium Bromide (Vegolysen; Esametina; Simpatoblock),a peripherally-acting and nondepolarizing neuromuscular blocker,is a selective antagonist of neuronal-type nicotinic AChR in ganglia that wasused to treat chronic hypertension. |
|
V13604 | Galanthamine | 357-70-0 | Galanthamine is a potent and long-acting AChE inhibitor with IC50 of 0.35 μM, it exhibits 50-fold selectivity against butyryl-cholinesterase. |
|
V1185 | Gallamine Triethiodide | 65-29-2 | Gallamine Triethiodide (Flaxedil; Tricuran; Gallamoni jodidum; Gallaminii iodidum),a non-depolarising muscle relaxant, is a potent and cardioselective cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM. |
|
V17514 | Carbachol | 51-83-2 | Carbachol is a cholinomimetic drug that binds and activates the acetylcholine receptor. |
|
V1196 | Homatropine Bromide (Homatropine hydrobromide) | 51-56-9 | Homatropine Bromide (Equipin, Isopto Homatropine), the hydrobromide salt of Homatropine, is a potent muscarinic AChR (acetylcholine receptor) antagonist used before eye examinations (i.e. refraction), before and after certain eye surgeries, and for treating certain eye conditions (e.g., uveitis). |
|
V1172 | Pyridostigmine Bromide | 101-26-8 | Pyridostigmine Bromide (Mestinon; Regonol; Kalimin) is a parasympathomimetic and a reversible cholinesterase inhibitor used in the treatment of myasthenia gravis and to reverse the actions of muscle relaxants. |
|
V1160 | Tiotropium Bromide hydrate (BA-679 BR) | 139404-48-1 | Tiotropium Bromide hydrate (PUR-0200; BA-679BR; BA679BR;PUR0200; Spiriva), the monohydrate form of tiotropium bromide, is an anticholinergic and bronchodilator and a muscarinic receptor antagonist used as a long-acting bronchodilator for the management of chronic obstructive pulmonary disease (COPD). |
|
V1186 | Oxybutynin | 5633-20-5 | Oxybutynin (Ditropan, Lyrinel XL, Lenditro,Oxybutynin, Uripan) is a potent and competitive antagonist of the M1, M2, and M3 subtypes of the muscarinic acetylcholine receptor, used to relieve urinary and bladder difficulties. |
|
V1192 | Otilonium Bromide (Octylonium bromide; SP63) | 26095-59-0 | Otilonium bromide (SP-63;Octylonium bromide; SP63; trade name Spasmomen among others) is a potent anti-muscarinic agent and a CCB (calcium channel blocker) used to relieve spasmodic pain of the gut, in particular in irritable bowel syndrome. |
|
V1163 | Fesoterodine Fumarate | 286930-03-8 | Fesoterodine Fumarate (SPM907; Toviaz, SPM-907), the fumarate salt of Fesoterodine which is a prodrug of 5-hydroxymethyl tolterodine, is a muscarinic AChR receptor antagonist that has been approved for treating overactive bladder syndrome. |
|
V11209 | Corydaline | 518-69-4 | Corydaline is a bioactive and naturally occurringisoquinoline alkaloid extracted fromCorydalis yanhusuo. |
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