Structure | Cat No. | Product Name | CAS No. | Product Description |
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V75415 | (S)-CVN424 | 1799968-74-3 | (S)-CVN424 is a potent modulator of G protein-coupled receptor 6 (GPR6). |
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V70305 | 2-Oleoylglycerol (2-octadecenoic acid monoglyceride; 2-glyceryl monooleate) | 3443-84-3 | 2-Oleoylglycerol is a naturally occurring lipid in the diet. |
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V77329 | 2-PCCA hydrochloride | 2-PCCA HCl is a racemate and a GPR88 receptor agonist. | |
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V70558 | [Ala17]-MCH | 359784-84-2 | [Ala17]-MCH is an analog of MCH and is a ligand for MCHR1 (Ki=0.16 nM) with greater selectivity for MCHR2 (Ki=34 nM). |
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V70561 | Ac-hMCH(6-16)-NH2 | 1053601-50-5 | Ac-hMCH(6-16)-NH2 is a non-selective peptide agonist of MCH in human brain, with IC50s of 0.16 nM and 2.7 nM for MCH-1R and MCH-2R, respectively. |
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V70556 | AMG-076 | 1001438-96-5 | AMG-076 is an orally bioactive, selective MCHR1 antagonist. |
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V11653 | AS1269574 | 330981-72-1 | AS1269574 is a potent, orally bioactive GPR119 agonist with EC50 of 2.5 μM in HEK293 cells expressing human GPR119. |
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V1806 | AZD1981 | 802904-66-1 | AZD1981 is a novel potent and selective CRTh2 (Chemoattractant receptor-homologous molecule expressed on TH2 cells; DP2-Prostaglandin D2 receptor 2, ) receptor antagonist with IC50 of 4 nM,it displayed>1000-fold selectivity over more than 340 other enzymes and receptors, including DP1. |
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V75408 | BigLEN(mouse) | 501036-69-7 | BigLEN(mouse) is a potent and specific agonist of orphan G protein-coupled receptor 171 (GPR171) with a Kd of approximately 0.5 nM. |
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V75407 | BigLEN(rat) | 369377-66-2 | BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM. |
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V78421 | BigLEN(rat) TFA | BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM. | |
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V75409 | CID 2745687 | 264233-05-8 | CID 2745687 is a specific, reversible and competitive GPR35 antagonist (inhibitor) with Ki of 12.8 nM. |
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V75410 | CID1231538 | 354126-20-8 | CID1231538, a benzothiazole analog, is a potent GPR35 antagonist. |
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V3995 | CID1375606 | 313493-80-0 | CID 1375606 is the first selective surrogate agonist of orphan G protein-coupled receptor (GPCR) GPR27 identified fromscreening a diversity-oriented synthesis library. |
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V75416 | CVN424 | 2254706-21-1 | CVN424 is an orally bioactive and selective GPR6 inverse agonist/activator with a Ki of 9.4 nM and EC50 of 38 nM. |
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V70557 | Ethyl linolenate | 1191-41-9 | Ethyl linolenate is a fatty acid ethyl ester (FAEE). |
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V70559 | Ethyl linolenate-d5 (ethyl linolenate d5) | 203633-16-3 | Ethyl linolenate-d5 is the deuterated form of Ethyl linolenate. |
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V1803 | Fasiglifam (TAK875) | 1000413-72-8 | Fasiglifam(formerly known as TAK-875; TAK875) is a novel, long-acting, selective and orally bioavailable GPR40 agonist with anti-diabetic activity. |
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V75404 | GPCR agonist-2 | 291528-35-3 | GPCR agonist-2 (Compound 5j) is a GPCR GPR109b (HM74) agonist/activator with pEC50 of 6.51. |
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V75405 | GPR109 receptor agonist-2 | 957129-38-3 | GPR109 receptor agonist (activator)-2 (Compound 5) is a selective GPR109a agonist with pEC50 of 5.53. |