GPR

GPR

GPR related products

Structure Cat No. Product Name CAS No. Product Description
V75415 (S)-CVN424 1799968-74-3 (S)-CVN424 is a potent modulator of G protein-coupled receptor 6 (GPR6).
V70305 2-Oleoylglycerol (2-octadecenoic acid monoglyceride; 2-glyceryl monooleate) 3443-84-3 2-Oleoylglycerol is a naturally occurring lipid in the diet.
V77329 2-PCCA hydrochloride 2-PCCA HCl is a racemate and a GPR88 receptor agonist.
V70558 [Ala17]-MCH 359784-84-2 [Ala17]-MCH is an analog of MCH and is a ligand for MCHR1 (Ki=0.16 nM) with greater selectivity for MCHR2 (Ki=34 nM).
V70561 Ac-hMCH(6-16)-NH2 1053601-50-5 Ac-hMCH(6-16)-NH2 is a non-selective peptide agonist of MCH in human brain, with IC50s of 0.16 nM and 2.7 nM for MCH-1R and MCH-2R, respectively.
V70556 AMG-076 1001438-96-5 AMG-076 is an orally bioactive, selective MCHR1 antagonist.
V11653 AS1269574 330981-72-1 AS1269574 is a potent, orally bioactive GPR119 agonist with EC50 of 2.5 μM in HEK293 cells expressing human GPR119.
V1806 AZD1981 802904-66-1 AZD1981 is a novel potent and selective CRTh2 (Chemoattractant receptor-homologous molecule expressed on TH2 cells; DP2-Prostaglandin D2 receptor 2, ) receptor antagonist with IC50 of 4 nM,it displayed>1000-fold selectivity over more than 340 other enzymes and receptors, including DP1.
V75408 BigLEN(mouse) 501036-69-7 BigLEN(mouse) is a potent and specific agonist of orphan G protein-coupled receptor 171 (GPR171) with a Kd of approximately 0.5 nM.
V75407 BigLEN(rat) 369377-66-2 BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM.
V78421 BigLEN(rat) TFA BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM.
V75409 CID 2745687 264233-05-8 CID 2745687 is a specific, reversible and competitive GPR35 antagonist (inhibitor) with Ki of 12.8 nM.
V75410 CID1231538 354126-20-8 CID1231538, a benzothiazole analog, is a potent GPR35 antagonist.
V3995 CID1375606 313493-80-0 CID 1375606 is the first selective surrogate agonist of orphan G protein-coupled receptor (GPCR) GPR27 identified fromscreening a diversity-oriented synthesis library.
V75416 CVN424 2254706-21-1 CVN424 is an orally bioactive and selective GPR6 inverse agonist/activator with a Ki of 9.4 nM and EC50 of 38 nM.
V70557 Ethyl linolenate 1191-41-9 Ethyl linolenate is a fatty acid ethyl ester (FAEE).
V70559 Ethyl linolenate-d5 (ethyl linolenate d5) 203633-16-3 Ethyl linolenate-d5 is the deuterated form of Ethyl linolenate.
V1803 Fasiglifam (TAK875) 1000413-72-8 Fasiglifam(formerly known as TAK-875; TAK875) is a novel, long-acting, selective and orally bioavailable GPR40 agonist with anti-diabetic activity.
V75404 GPCR agonist-2 291528-35-3 GPCR agonist-2 (Compound 5j) is a GPCR GPR109b (HM74) agonist/activator with pEC50 of 6.51.
V75405 GPR109 receptor agonist-2 957129-38-3 GPR109 receptor agonist (activator)-2 (Compound 5) is a selective GPR109a agonist with pEC50 of 5.53.
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