|
V0698
|
Aloxistatin (Loxistatin; E64d, NSC-694281)
|
88321-09-9 |
Aloxistatin (also known asE-64d,E-64c ethyl ester; EST, Loxistatin; NSC 694281) is a novel, potent, selective, irreversible,broad-spectrum and cell membrane-permeable cysteine protease inhibitor with anticoagulant activities. |
|
V4361
|
BALICATIB
|
354813-19-7 |
Balicatib (also known as AAE-581) is a novel, potent and selective inhibitor of cathepsin K with 10-100 fold higher potency in cell-based enzyme occupancy assays than against cathepsin B, L, and S. |
|
V0706
|
Calpeptin
|
117591-20-5 |
Calpeptin(sequence: Z-Leu-nLeu-H) is a novel, potent, cell-permeable calpain inhibitor with anti-fibrotic activity. |
|
V0699
|
Cathepsin Inhibitor 1
|
225120-65-0 |
Cathepsin Inhibitor 1 (CTS-IN-1) is a novel and potent inhibitor of Cathepsin (L, L2, S, K, B) with the potential to be used in the treatment of osteoarthritis. |
|
V33611
|
Cruzain-IN-1
|
1199523-24-4 |
Cruzain-IN-1 is a covalent reversible inhibitor of Trypanosoma cruzi cysteine protease (Cruzain) with IC50 of 10 nM. |
|
V0708
|
E-64
|
66701-25-5 |
E-64 (also known as Proteinase inhibitor E 64), a naturally occuring compound isolated from cultures of Aspergillus, is a novel, potent, irreversible and selective cysteine protease inhibitorwith potential antineoplastic andantiparasitic activity. |
|
V0703
|
Leupeptin Hemisulfate (NK381)
|
103476-89-7 |
Leupeptin Hemisulfate (NK-381; N-acetyl-L-leucyl-L-leucyl-L-argininal) is a naturally occurring, membrane-permeable, reversible and competitive inhibitor of the serine and cysteine proteases with potential antioxidant and anti-inflammatory activity. |
|
V0700
|
Loxistatin Acid (E-64C; NSC694279; EP475)
|
76684-89-4 |
Loxistatin Acid (formerly also known as E-64C; NSC-694279; EP-475), an analog of E-64, is a novel, potent, irreversible and membrane-permeable cysteine protease inhibitor with important biological activity. |
|
V28953
|
MDL-28170
|
88191-84-8 |
MDL-28170 (Calpain Inhibitor III) is a novel potent, selective and membrane-permeable cysteine protease inhibitor of calpain that rapidly penetrates the blood-brain barrier following systemic administration. |
|
V0705
|
MG-101 (ALLN)
|
110044-82-1 |
MG-101 (also known as MG101; Calpain Inhibitor I and ALLN) is a novel, cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins with potential antitumor activity. |
|
V3163
|
N-Ethylmaleimide (NEM)
|
128-53-0 |
N-Ethylmaleimide (also known as NEM) is an organic biochemical compound that is derived from maleic acid. |
|
V0696
|
Odanacatib (MK0822)
|
603139-19-1 |
Odanacatib (also known as MK-0822) is a potent, selective, and neutral inhibitor of cathepsin K (human/rabbit) with the potential to be used for thetreatment for osteoporosis and bone metastasis. |
|
V0704
|
PD 151746
|
179461-52-0 |
PD 151746 (PD-151746) is a novel, potent, selective, andcell-permeable calpain inhibitor with important biological activity. |
|
V0701
|
PMSF
|
329-98-6 |
PMSF (full name: Phenylmethanesulfonyl fluoride) is a potent and irreversible inhibitor of serine/cysteine protease (e.g. thrombin, trypsin and chymotrypsin) with potential analgesic effects. |
|
V0702
|
Z-FA-FMK
|
197855-65-5 |
Z-FA-FMK, a control peptidic fluoromethylketone (boc-Thr-CH2F), is a novel and irreversible cysteine protease inhibitor, and also inhibits effector caspases. |