The cell-surface serine protease known as fibroblast activation protein (FAP) affects different hormones and elements of the extracellular matrix. FAP is frequently used as a marker for pro-tumorigenic stroma and is highly upregulated in a variety of cancers.
Structure | Cat No. | Product Name | CAS No. | Product Description |
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V86175 | 3BP-3940 | 2803421-14-7 | |
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V86846 | [99mTc]Tc-6–1 | [99m Tc]Tc-6-1 is a 99mTc-labeled FAPI-46 derivative and a specific fibroblast activation protein (FAP) targeted radiotracer. | |
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V85878 | AlF-PD-FAPI | ||
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V93849 | DOTAGA.(SA.FAPi)2 analogue TFA | DOTAGA.(SA.FAPi)2 analog TFA is an analog of DOTAGA.(SA.FAPi)2 TFA, wherein the ligand and chelator moieties are the same as DOTAGA.(SA.FAPi)2 TFA. | |
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V94503 | DOTAGA.(SA.FAPi)2 TFA | DOTAGA.(SA.FAPi)2 TFA is a potent inhibitor of dimeric fibroblast activation protein (FAPi). | |
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V79388 | FAP-IN-1 | 2956858-96-9 | FAP-IN-1 is a fibroblast activation protein (FAP) inhibitor (antagonist) with IC50 of 3.3 nM. |
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V74897 | FAP-IN-2 | 2471983-20-5 | FAP-IN-2 is an analogue of 99mTc-labeled isonitrile-containing fibroblast activation protein (FAPI) inhibitor that can be used for tumor imaging. |
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V77022 | FAP-IN-2 TFA | FAP-IN-2 TFA is an analogue of 99mTc-labeled isonitrile-containing FAP inhibitor that can be used for tumor imaging. | |
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V86845 | FAP-IN-4 | FAP-IN-4 (Comp 10) is a fibroblast activation protein (FAP) inhibitor and a 18F-labeled PET tracer targeting FAP. | |
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V74893 | FAPI-2 | 2370952-98-8 | FAPI-2 is a fibroblast activation protein (FAP) inhibitor that has applications in cancer-related research. |
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V77023 | FAPI-2 TFA | FAPI-2 TFA is a fibroblast activation protein (FAP) inhibitor (antagonist) with potential use in cancer-related research. | |
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V74894 | FAPI-34 | 2374782-07-5 | FAPI-34 is a fibroblast activating protein (FAP) inhibitor (antagonist) with good pharmacokinetic and biochemical properties, disclosed in patent WO2019154886A1. |
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V51734 | FAPI-46 | 2374782-04-2 | FAPI-46 is a quinoline-based activator of fibroblast-activated protein (FAP). |
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V74898 | FAPI-74 | 2374782-76-8 | FAPI-74 is a PET (positron emission tomography) tracer for fibroblast activating protein. |
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V94533 | FAPI-mFS | 3023869-94-2 | FAPI-mFS is an irreversible fibroblast activation protein (FAP) inhibitor that enhances its uptake and retention time in cancer cells through its covalent binding properties to FAP. |
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V74895 | Fluorogen binding modulator-1 | 510716-65-1 | Fluorogen binding modulator-1 (PubChem SID 125240934) is a fluorescein-activated protein (FAP)-fluorogen binding modulator with a -log EC50 of 6.61 for AM2.2-β2AR and AM2.2-gpr32 respectively. |
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V100354 | FT-FAPI-12_9 | 2883407-81-4 | FT-FAPI-12_9 is a FAP conjugate that can be used to synthesize the FAP-targeted radiotracer FAPI-46. |
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V97374 | FT-FAPI-12_9 TFA | FT-FAPI-12_9 (TFA) is a FAP conjugate that can be used to synthesize the FAP-targeted radiotracer FAPI-46. | |
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V76701 | NH2-UAMC1110 TFA | 2990021-73-1 | NH2-UAMC1110 TFA is a UAMC1110 analogue that may be utilized in the synthesis/preparation of FAPI-QS. |
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V85436 | PNT6555 |