Structure | Cat No. | Product Name | CAS No. | Product Description |
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V83537 | (R)-MrgprX2 antagonist-3 | 2642174-20-5 | |
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V4494 | (S)-ZINC-3573 | 2095596-11-3 | (S)-ZINC-3573 is the inactive enantiomer of ZINC-3573. |
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V78342 | BAM(8-22) TFA | BAM(8-22) TFA, a proteolytic cleavage product of proenkephalin A, is a potent activator of Mas-related G protein-coupled receptors (Mrgprs), MrgprC11 and hMrgprX1, and induces in mice a Mrgpr-dependent manner. | |
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V2517 | MRGPRX1 agonist 1 | 2377379-39-8 | MRGPRX1 agonist 1 is a novel and highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1) (EC50 = 50 nM) with analgesic effects. |
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V75464 | MrgprX2 antagonist-1 | 2642162-06-7 | MrgprX2 antagonist-1 is an antagonist of MrgprX2. |
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V75469 | MrgprX2 antagonist-2 | 2642346-30-1 | MrgprX2 antagonist-2 is an antagonist of MrgprX2. |
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V75470 | MrgprX2 antagonist-3 | 2642174-19-2 | MrgprX2 antagonist-3 is an antagonist of MrgprX2. |
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V75468 | MrgprX2 antagonist-4 | 2641398-04-9 | MrgprX2 antagonist-4 is an antagonist of MrgprX2. |
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V75465 | MrgprX2 antagonist-5 | 2527815-74-1 | MrgprX2 antagonist-5 is an antagonist of MrgprX2. |
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V75467 | Mrgx2 antagonist-2 | 2767111-67-9 | Mrgx2 antagonist-2 is a Mrgx2 antagonist (refer to Example 123 in the patent) with pIC50 of 8.6. |
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V81036 | PAMP-12 (unmodified) (TFA) | PAMP-12 (unmodified) TFA is a potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM). | |
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V75466 | ZINC49534341 | 1274013-03-4 | ZINC49534341 is an MRGPRX2 antagonist (inhibitor) with Ki of 32 nM. |