| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V83537 | (R)-MrgprX2 antagonist-3 | 2642174-20-5 | |
|
V110928 | (Rac)-EP-2825 | 958571-34-1 | (Rac)-EP-2825 (compound 8-6) is an MRGPRD agonist with an IC50 value between 100 and 500 nM. |
|
V4494 | (S)-ZINC-3573 | 2095596-11-3 | (S)-ZINC-3573 is the inactive enantiomer of ZINC-3573. |
|
V107087 | 1-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid | 50264-63-6 | 1-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid (Compound 31) is a metabolite of AB-FUBINACA. |
|
V106996 | 4-Aminobenzimidamide Hydrochloride | 7761-72-0 | 4-Aminobenzamide hydrochloride (compound 4a) is a MRGPRX1 agonist. |
|
V78342 | BAM(8-22) TFA | BAM(8-22) TFA, a proteolytic cleavage product of proenkephalin A, is a potent activator of Mas-related G protein-coupled receptors (Mrgprs), MrgprC11 and hMrgprX1, and induces in mice a Mrgpr-dependent manner. | |
|
V109146 | BCFTP | 2781215-95-8 | BCFTP is a potent, orally effective, and selective positive allosteric modulator of human Mas-associated G protein-coupled receptor X1 (MrgprX1). |
|
V108978 | Catestatin (mouse) | 1461673-77-7 | Catestatin, a mouse-derived antimicrobial peptide, is an antimicrobial peptide. |
|
V111788 | JHU-58 | 1632140-61-4 | JHU-58 is a peptide mimic agonist that targets the MRGPRC11 receptor in mice and the MRGPRC receptor in rats. |
|
V111146 | LY3325656 | 1998714-25-2 | LY3325656 is a selective GPR142 receptor agonist. |
|
V2517 | MRGPRX1 agonist 1 | 2377379-39-8 | MRGPRX1 agonist 1 is a novel and highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1) (EC50 = 50 nM) with analgesic effects. |
|
V75464 | MrgprX2 antagonist-1 | 2642162-06-7 | MrgprX2 antagonist-1 is an antagonist of MrgprX2. |
|
V75469 | MrgprX2 antagonist-2 | 2642346-30-1 | MrgprX2 antagonist-2 is an antagonist of MrgprX2. |
|
V75470 | MrgprX2 antagonist-3 | 2642174-19-2 | MrgprX2 antagonist-3 is an antagonist of MrgprX2. |
|
V75468 | MrgprX2 antagonist-4 | 2641398-04-9 | MrgprX2 antagonist-4 is an antagonist of MrgprX2. |
|
V75465 | MrgprX2 antagonist-5 | 2527815-74-1 | MrgprX2 antagonist-5 is an antagonist of MrgprX2. |
|
V116619 | MrgprX2 antagonist-9 | 3095296-92-4 | MrgprX2 antagonist-9 (compound 10) is a potent MrgprX2 antagonist with an IC50 value of 0.1-100 nM. |
|
V86662 | MRGPRX2 modulator-1 | 2781839-42-5 | MRGPRX2 modulator-1 (example 17) is a mas-related g protein receptor x2 (MRGPRX2) modulator. |
|
V118821 | MRGPRX4 modulator-3 | MRGPRX4 modulator-3 (compound 1C) is a modulator of the negative allosteric MAS-associated G protein-coupled receptor X4 (MRGPRX4). | |
|
V75467 | Mrgx2 antagonist-2 | 2767111-67-9 | Mrgx2 antagonist-2 is a Mrgx2 antagonist (refer to Example 123 in the patent) with pIC50 of 8.6. |