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Vasopressin Receptor

Vasopressin Receptor

Neurohypophysial hormone arginine vasopressin (AVP) regulates body fluid homeostasis, causes vasoconstriction, and releases adrenocorticotropic hormone, among other things. Three subtypes of vasopressin receptors—designated V1a, V1b (or V3), and V2—mediate these physiological effects. They are all members of the large family of G-protein-coupled receptors that resemble rhodopsin.
The V1a receptor stimulates hepatic glycogenolysis, platelet aggregation, coagulation factor release, and cell contraction and proliferation. It is expressed in both neuronal and non-neuronal tissues, including the heart. The pituitary gland is the primary site of the V1b receptor subtype, which is responsible for stimulating the release of adrenocorticotropic hormone. The G protein alpha-subunit of the Gαq family (αq, q11, q14, α15/16) is the mechanism by which the V1a and V1b AVP receptors activate phospholipase C-β, raising the levels of calcium and IP3 in cells. On the other hand, the V2 receptor subtype is primarily found in the kidney, where it activates adenylyl cyclase and mediates the anti-diuretic effects of AVP via the heterotrimeric G protein Gs.

Vasopressin Receptor related products

Structure Cat No. Product Name CAS No. Product Description
(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) V74547 (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) 73168-24-8 (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin (SKF 100273) is a vasopressin V1 receptor selective antagonist.
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) V74535 (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) 176714-12-8 (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) is a specific vasopressin receptor V1a antagonist agent, the pA2 value was 6.71.
(D-Arg8)-Inotocin V74540 (D-Arg8)-Inotocin 745816-74-4 (D-Arg8)-Inotocin is a specific and competitive vasopressin receptor V1aR antagonist (inhibitor) with a Ki of 1.3 nM.
(Phe2,Orn8)-Oxytocin acetate V77425 (Phe2,Orn8)-Oxytocin acetate (Phe2,Orn8)-Oxytocin acetate is a selective V1 vasopressin agonist.
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin V74534 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin 129520-65-6 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin is a potent vasopressin V1 receptor (VP V1R) antagonist.
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin acetate V86791 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin acetate (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin acetate is a potent vasopressin V1 receptor (VP V1R) antagonist.
[Asu1,6-Arg8]Vasopressin V74542 [Asu1,6-Arg8]Vasopressin 40944-53-4 [Asu1,6-Arg8]Vasopressin is a vasopressin agonist that enhances corticotropin-releasing factor (CRF)-induced cyclic AMP accumulation and ACTH release in cultured rat anterior pituitary cells.
[Deamino-Pen1,Val4,D-Arg8]-vasopressin V74538 [Deamino-Pen1,Val4,D-Arg8]-vasopressin 64158-84-5 [Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an arginine vasopressin (AVP) antagonist.
Antagonist G TFA V77957 Antagonist G TFA Antagonist G TFA is a potent vasopressin antagonist.
Balovaptan | RG7314 | Vasopressin Receptor V12273 Balovaptan 1228088-30-9 Balovaptan (RG7314; RG-7314; RO-5285119) is a novel potent andbrain-penetrant vasopressin 1a (hV1a) receptor antagonist with the potential to be used for autism.
Big Endothelin-1 (1-38), human V74531 Big Endothelin-1 (1-38), human 120796-97-6 Big Endothelin-1 (1-38), human is the precursor of endothelin-1.
Big Endothelin-1 (1-39), porcine V74537 Big Endothelin-1 (1-39), porcine 120796-99-8 Big Endothelin-1 (1-39), porcine is the precursor of endothelin-1.
d[Cha4]-AVP V74532 d[Cha4]-AVP 500170-27-4 d[Cha4]-AVP is a potent and specific vasopressin (AVP) V1b receptor agonist/activator with a Ki of 1.2 nM for the human V1b receptor.
d[Cha4]-AVP TFA V78994 d[Cha4]-AVP TFA d[Cha4]-AVP TFA is a potent and specific vasopressin (AVP) V1b receptor agonist/activator with a Ki of 1.2 nM for the human V1b receptor.
D[LEU4,LYS8]-VP V74541 D[LEU4,LYS8]-VP 42061-33-6 D[LEU4,LYS8]-VP is a selective agonist of vasopressin V1b receptor, with Kis of 0.16 nM, 0.52 nM and 1.38 nM for rat, human and mouse V1b receptor respectively.
D[LEU4,LYS8]-VP TFA V77111 D[LEU4,LYS8]-VP TFA D[LEU4,LYS8]-VP TFA is a selective agonist of vasopressin V1b receptor, with Kis of 0.16 nM, 0.52 nM and 1.38 nM for rat, human and mouse V1b receptor respectively.
Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin V74544 Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin 136105-89-0 Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin is a synthetic analog of antidiuretic hormone (AVP) and a weak agonist of antidiuretic receptors.
Dp[Tyr(methyl)2,Arg8]-Vasopressin V74536 Dp[Tyr(methyl)2,Arg8]-Vasopressin 67269-08-3 Dp[Tyr(methyl)2,Arg8]-Vasopressin is a non-selective peptide arginine vasopressin Vlb receptor blocker (antagonist).
Endolide F V86793 Endolide F Endolide F (Compound 2) is a proline-containing lactone.
Enuvaptan (BAY-2327949) V74543 Enuvaptan (BAY-2327949) 2145062-48-0 Enuvaptan (BAY-2327949) is a vasopressin receptor blocker (antagonist) with potential for studying renal and cardiovascular diseases.
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