Adrenergic receptors are a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.These receptors are found on numerous cells, and when a catecholamine binds to one of these receptors, the sympathetic nervous system is typically stimulated. The fight-or-flight response, which entails dilating the pupils of the eyes, mobilizing energy, and rerouting blood flow away from skeletal muscle to non-essential organs, is controlled by the sympathetic nervous system.There are numerous subtypes of the two main groups of adrenergic receptors, and. The receptor subtypes 1 and 2 exist. There are three subtypes of receptors: 1, 2, and 3. They are all associated with Gs proteins, which are associated with adenylate cyclase. Thus, antagonist binding increases the level of the second messenger cAMP inside of the cell. The cAMP-dependent protein kinase (PKA), one of cAMP's downstream effectors, mediates some intracellular processes after hormone binding.
| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V87631 | (Rac)-Nebivolol-d2,15N | (Rac)-Nebivolol-d2,15N is 15N and deuterium labeled (Rac)-Nebivolol. | |
|
V84080 | (Rac)-Nebivolol-d4 hydrochloride ((Rac)-R 065824-d4 hydrochloride) | 2701283-32-9 | |
|
V86520 | 5,6-Epoxyeicosatrienoic acid | 87173-80-6 | 5,6-Epoxyeicosatrienoic acid (5,6-EET; (±)5,6-EpETrE) is a fully racemic form of the enantiomer biosynthesized from arachidonic acid by cytochrome P450 enzymes. |
|
V89031 | ADRA2A antagonist 1 | ADRA2A antagonist 1 (compd 4n) is a potent and selective ADRA2A antagonist with IC50 of 18 nM. | |
|
V87770 | Amitraz-d6 | 2734300-36-6 | Amitraz-d6 (BTS-27419-d6) is the deuterated derivative of Amitraz. |
|
V86143 | Apraclonidine dihydrochloride (ALO 2145 dihydrochloride) | 73217-88-6 | |
|
V85241 | BAY-6096 | 2313483-41-7 | |
|
V87767 | BRL-37344 | 90730-96-4 | BRL-37344 is a specific β3-adrenergic receptor agonist. |
|
V87814 | Cirazoline | 59939-16-1 | Cirazoline (LD 3098) is a dual agonist of presynaptic imidazoline receptors (R(i-pre)) and α-adrenergic receptors (R(α)). |
|
V90532 | Guanfacine-13C,d5 hydrochloride | Guanfacine-13C,d5 hydrochloride is a 13C-labeled deuterated form of Guanfacine hydrochloride. | |
|
V89800 | Guanfacine-15N13,13C2 | Guanfacine-15N3,13C2 is 15N and 13C labeled Guanfacine. | |
|
V87813 | Harmane-d4 | 2012598-89-7 | Harmane-d4 is deuterium-labeled Harmane. |
|
V86519 | Heptaminol | 372-66-7 | Heptaminol is a fatty amine with pressor properties and is a potential antihypotensive agent. |
|
V86521 | Idazoxan | 79944-58-4 | Idazoxan is a potent α2 adrenergic receptor (α2AR) antagonist and potential I2 imidazoline receptor (imidazoline receptor) agonist. |
|
V90641 | Isoprenaline-d7 hydrochloride | 2517584-04-0 | Isoprenaline-d7 (hydrochloride) is a deuterated isoprenaline (hydrochloride). |
|
V3338 | L-765314 | 189349-50-6 | L-765314 (L-765,314) is a novel, potent and selectiveα1b adrenergic receptorantagonist withKis of 5.4 nM and 2.0 nM for rat and human α1b adrenergic receptor, respectively. |
|
V89030 | Mabuterol hydrochloride | 54240-36-7 | Mabuterol hydrochloride is a selective and orally active beta-2 adrenergic receptor (ADRB2) agonist. |
|
V90632 | Medetomidine-13C,d3 hydrochloride | 1216630-06-6 | Medetomidine-13C,d3 (hydrochloride) is a deuterated Medetomidine (hydrochloride). |
|
V88928 | Mirtazapine-d4 hydrochloride | 1215587-73-7 | Mirtazapine-d4 hydrochloride is a deuterated mitazapine. |
|
V88574 | Olanzapine-d4 | 1252611-62-3 | Olanzapine-d4 (LY170053-d4) is deuterium-labeled Olanzapine. |
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