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Adrenergic Receptor

Adrenergic Receptor

Adrenergic receptors are a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.These receptors are found on numerous cells, and when a catecholamine binds to one of these receptors, the sympathetic nervous system is typically stimulated. The fight-or-flight response, which entails dilating the pupils of the eyes, mobilizing energy, and rerouting blood flow away from skeletal muscle to non-essential organs, is controlled by the sympathetic nervous system.There are numerous subtypes of the two main groups of adrenergic receptors, and. The receptor subtypes 1 and 2 exist. There are three subtypes of receptors: 1, 2, and 3. They are all associated with Gs proteins, which are associated with adenylate cyclase. Thus, antagonist binding increases the level of the second messenger cAMP inside of the cell. The cAMP-dependent protein kinase (PKA), one of cAMP's downstream effectors, mediates some intracellular processes after hormone binding.

Adrenergic Receptor related products

Structure Cat No. Product Name CAS No. Product Description
(-)-Isoproterenol hydrochloride V101112 (-)-Isoproterenol hydrochloride 5984-95-2 (-)-Isoproterenol (L-isoproterenol; Proternol L) hydrochloride is a β-adrenergic receptor agonist.
(1R,2S)-Dihydrobupropion V116575 (1R,2S)-Dihydrobupropion 292055-72-2 (1R,2S)-dihydrobupropion is a norepinephrine-dopamine reuptake inhibitor and one of the active metabolites of bupropion.
(2S,3S)-Zenidolol hydrochloride V112149 (2S,3S)-Zenidolol hydrochloride 1236034-74-4 (2S,3S)-Zenidolol ((2S,3S)-ICI-118551) hydrochloride is a β2-adrenergic receptor (β2AR) antagonist with a pKi value of 7.51 for β1AR and 9.27 for β2AR.
(Rac)-Nebivolol-d2,15N V87631 (Rac)-Nebivolol-d2,15N (Rac)-Nebivolol-d2,15N is 15N and deuterium labeled (Rac)-Nebivolol.
(Rac)-Nebivolol-d4 hydrochloride ((Rac)-R 065824-d4 hydrochloride) V84080 (Rac)-Nebivolol-d4 hydrochloride ((Rac)-R 065824-d4 hydrochloride) 2701283-32-9
(S)-Atenolol V101375 (S)-Atenolol 93379-54-5 (S)-Atenolol is a potent β-adrenergic receptor blocker.
(S)-Doxazosin V113025 (S)-Doxazosin 104874-86-4 (S)-Doxazosin is a long-acting selective α1-adrenergic receptor antagonist.
(S)-Trimetoquinol hydrochloride V110173 (S)-Trimetoquinol hydrochloride 18559-59-6 (S)-Trimethylquinolone hydrochloride (compound 1) is a potent, nonselective, nonclassical β-adrenergic agonist and a nonprostaglandin A2/prostaglandin H2 antagonist.
(±)-4-Hydroxy propranolol β-D-glucuronide V102882 (±)-4-Hydroxy propranolol β-D-glucuronide 94731-13-2 (±)-4-Hydroxypropranolol β-D-glucuronide is a metabolite of the β-adrenergic receptor antagonist 4-hydroxypropranolol.
(±)-Penbutolol V102678 (±)-Penbutolol 36507-48-9 (±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of penbutolol.
(±)-WB 4101 V115621 (±)-WB 4101 613-67-2 (±)-WB 4101 is a highly selective α1-adrenergic receptor inhibitor.
2,3-MDMA hydrochloride V107164 2,3-MDMA hydrochloride 168968-01-2 2,3-MDMA hydrochloride is a norepinephrine transporter and serotonin transporter inhibitor with IC50 values of 6.2 μM and 82 μM, respectively.
3,4-Dihydro-6,7-isoquinolinediol V92173 3,4-Dihydro-6,7-isoquinolinediol 4602-83-9 3,4-Dihydro-6,7-isoquinolinediol (compound 7) is a β2-AR agonist with EC50 of 106.9 μM in CH-K1/GA1S cells.
4-Hydroxy nebivolol hydrochloride V101068 4-Hydroxy nebivolol hydrochloride 2717115-85-8 4-Hydroxynebivolol (4-OH nebivolol) hydrochloride is the active β-blocking hydrolytic metabolite of nebivolol.
5,6-Epoxyeicosatrienoic acid V86520 5,6-Epoxyeicosatrienoic acid 87173-80-6 5,6-Epoxyeicosatrienoic acid (5,6-EET; (±)5,6-EpETrE) is a fully racemic form of the enantiomer biosynthesized from arachidonic acid by cytochrome P450 enzymes.
5-Hydroxy propranolol V102915 5-Hydroxy propranolol 81907-82-6 5-Hydroxypropranolol is a metabolite of propranolol and can be used to study the β-adrenergic receptor blocking effect.
A 131701 V114283 A 131701 181490-18-6 A131701 is a selective α1a receptor (human α1a receptor Ki value: 0.22 nM) and α1d adrenergic receptor antagonist.
A 80426 mesylate V102470 A 80426 mesylate 152148-64-6 A 80426 mesylate is an alpha2-adrenergic receptor antagonist.
Acepromazine-d6 hydrochloride V110620 Acepromazine-d6 hydrochloride 1173022-70-2 Acepromazine-d6 hydrochloride is a deuterated acepromazine hydrochloride.
Aclidinium V98017 Aclidinium 727649-81-2 Aclidinium bromide is a long-acting muscarinic antagonist and long-acting β2-adrenergic receptor (β2-AR) agonist with bronchodilatory effects.
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