Adrenergic receptors are a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.These receptors are found on numerous cells, and when a catecholamine binds to one of these receptors, the sympathetic nervous system is typically stimulated. The fight-or-flight response, which entails dilating the pupils of the eyes, mobilizing energy, and rerouting blood flow away from skeletal muscle to non-essential organs, is controlled by the sympathetic nervous system.There are numerous subtypes of the two main groups of adrenergic receptors, and. The receptor subtypes 1 and 2 exist. There are three subtypes of receptors: 1, 2, and 3. They are all associated with Gs proteins, which are associated with adenylate cyclase. Thus, antagonist binding increases the level of the second messenger cAMP inside of the cell. The cAMP-dependent protein kinase (PKA), one of cAMP's downstream effectors, mediates some intracellular processes after hormone binding.
| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V101112 | (-)-Isoproterenol hydrochloride | 5984-95-2 | (-)-Isoproterenol (L-isoproterenol; Proternol L) hydrochloride is a β-adrenergic receptor agonist. |
|
V87631 | (Rac)-Nebivolol-d2,15N | (Rac)-Nebivolol-d2,15N is 15N and deuterium labeled (Rac)-Nebivolol. | |
|
V84080 | (Rac)-Nebivolol-d4 hydrochloride ((Rac)-R 065824-d4 hydrochloride) | 2701283-32-9 | |
|
V101375 | (S)-Atenolol | 93379-54-5 | (S)-Atenolol is a potent β-adrenergic receptor blocker. |
|
V102882 | (±)-4-Hydroxy propranolol β-D-glucuronide | 94731-13-2 | |
|
V102678 | (±)-Penbutolol | 36507-48-9 | |
|
V107164 | 2,3-MDMA hydrochloride | 168968-01-2 | |
|
V92173 | 3,4-Dihydro-6,7-isoquinolinediol | 4602-83-9 | 3,4-Dihydro-6,7-isoquinolinediol (compound 7) is a β2-AR agonist with EC50 of 106.9 μM in CH-K1/GA1S cells. |
|
V101068 | 4-Hydroxy nebivolol hydrochloride | 2717115-85-8 | 4-Hydroxynebivolol (4-OH nebivolol) hydrochloride is the active β-blocking hydrolytic metabolite of nebivolol. |
|
V86520 | 5,6-Epoxyeicosatrienoic acid | 87173-80-6 | 5,6-Epoxyeicosatrienoic acid (5,6-EET; (±)5,6-EpETrE) is a fully racemic form of the enantiomer biosynthesized from arachidonic acid by cytochrome P450 enzymes. |
|
V102915 | 5-Hydroxy propranolol | 81907-82-6 | |
|
V102470 | A 80426 mesylate | 152148-64-6 | |
|
V98017 | Aclidinium | 727649-81-2 | Aclidinium bromide is a long-acting muscarinic antagonist and long-acting β2-adrenergic receptor (β2-AR) agonist with bronchodilatory effects. |
|
V89031 | ADRA2A antagonist 1 | ADRA2A antagonist 1 (compd 4n) is a potent and selective ADRA2A antagonist with IC50 of 18 nM. | |
|
V94737 | Amibegron | 121524-08-1 | Amibegron is a selective β3-adrenergic receptor agonist with an EC50 of 3.5 nM for rat colonic β-adrenergic receptors; Amibegron has anxiolytic and antidepressant effects. |
|
V87770 | Amitraz-d6 | 2734300-36-6 | Amitraz-d6 (BTS-27419-d6) is the deuterated derivative of Amitraz. |
|
V86143 | Apraclonidine dihydrochloride (ALO 2145 dihydrochloride) | 73217-88-6 | Apraclonidine (ALO 2145) dihydrochloride is a selective α2 and weak α1 receptor agonist |
|
V102471 | Azepexole hydrochloride | 147663-20-5 | |
|
V85241 | BAY-6096 | 2313483-41-7 | |
|
V94462 | Bedoradrine | 194785-19-8 | Bedoradrine is a highly selective β2-adrenergic agonist with activity in suppressing asthma and chronic obstructive pulmonary disease (COPD). |
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