Prostaglandin Receptor

Prostaglandin Receptor

Prostaglandin receptor, a sub-family of cell surface seven-transmembrane receptors, are the G-protein-coupled receptors.Ten distinct prostaglandin receptors on different cell types are currently known. G-protein-coupled receptors are a subclass of cell surface seven-transmembrane receptors that prostaglandins bind to. The following are the names of these receptors: FP-FP, IP1-2-IP1, IP2 receptors, TP-TP receptor, EP1-4-EP1, EP2, EP3, and EP4 receptors. A class of lipid molecules known as prostaglandins, which are produced enzymatically from fatty acids and resemble hormones, play vital roles in the bodies of animals. Ten distinct prostaglandin receptors on different cell types are currently known.

Prostaglandin Receptor related products

Structure Cat No. Product Name CAS No. Product Description
V74464 (+)-Fluprostenol 54276-17-4 (+)-Fluprostenol is a potent agonist of PTGER2.
V74493 (+)-Oxypeucedanin methanolate 52939-12-5 (+)-Oxypeucedanin methanolate (compound 9) is a naturally occurring compound that can inhibit prostaglandin E2 production.
V74496 (8-epi)-BW 245C 65705-83-1 (8-epi)-BW 245C is the C-8 diastereomer of BW 245C.
V74478 (S)-Butaprost free acid 433219-55-7 (S)-Butaprost (free acid) is a potent and selective EP2 receptor agonist (activator).
V74485 11-Deoxy Prostaglandin E2 35536-53-9 11-Deoxy Prostaglandin E2 is an EP4 selective agonist/activator with EC50 of 0.66 nM.
V84325 12(S)-HPEPE 103239-14-1
V83666 13,14-Dihydro-15-keto prostaglandin D2 (DK-PGD2; 15-Oxo-13,14-dihydro-PGD2; 13,14-Dihydro-15-keto-PGD2) 59894-07-4
V84195 15(S)-HpEPE 125992-60-1
V74482 15-Keto latanoprost 135646-98-9 15-Keto latanoprost is a metabolite of Latanoprost, an intraocular pressure-lowering agent.
V74488 19(S)-HETE 115461-40-0 19(S)-HETE is an arachidonic acid metabolite produced by cytochrome P450 enzymes.
V74458 1a,1b-Dihomo prostaglandin E1 (1a,1b-Dihomo PGE1) 23452-98-4 1a,1b-Dihomo prostaglandin E1 (1a,1b-Dihomo PGE1) is a class of prostaglandin compounds.
V10518 AH6809 33458-93-4 AH6809 (AH-6809) is a novel and potent DP/EP prostanoid receptor antagonist with a Ki of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively, and with a Ki of 350 nM for mouse EP2 receptor.
V2425 Alprostadil (PGE1; Prostaglandin-E1) 745-65-3 Alprostadil (also known as Prostaglandin-E1) is a naturally occurring prostaglandin and a potent vasodilator used in the treatment of infants with congenital heart defects to maintain the patency of the ductus arteriosus until palliative or corrective surgery can be performed.
V3450 AMG-009 1027847-67-1 AMG-009 is a novel, potent, orally bioactive, small molecule antagonist of prostaglandin D2, with IC50 of 3 nM and 12 nM for CRTH2 (chemoattractant receptor-homologous molecule expressed on Th2 cells) and DP (D prostanoid) receptors, respectively.
V74494 AMX12006 2639775-01-0 AMX12006 is a specific and orally bioactive EP4 antagonist (inhibitor) with IC50 of 4.3 nM.
V74463 AZ12672857 945396-55-4 AZ12672857 is an orally bioactive inhibitor of EphB4 (IC50=1.3 nM) and Src kinase.
V74474 BAY-6672 2247517-53-7 BAY-6672 is a potent and specific human prostaglandin F (FP) receptor blocker (antagonist) with IC50 of 11 nM.
V74476 BAY-6672 hydrochloride 2247520-31-4 BAY-6672 HCl is a potent and specific human prostaglandin F (FP) receptor blocker (antagonist) with IC50 of 11 nM.
V74469 BGC-20-1531 free base (PGN 1531 free base) 736183-35-0 BGC-20-1531 (PGN 1531) free base is a potent and specific prostaglandin EP4 receptor antagonist (inhibitor) with a pKB value of 7.6.
V84541 Bima SA (Bimatoprost serinol amide) 1175838-84-2
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