|
V0050
|
TG-101209
|
936091-14-4 |
TG101209 is a novel, potent, orally bioactive and selective small molecule JAK2 inhibitor with IC50 of 6 nM. |
|
V0048
|
Regorafenib (BAY73-4506)
|
755037-03-7 |
Regorafenib (also known as BAY 73-4506; BAY-73-4506) is a potent andorally bioavailable multi-kinase inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 values of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM in cell-free assays, respectively. |
|
V0071
|
Regorafenib HCl (BAY-73-4506)
|
835621-07-3 |
Regorafenib HCl, the hydrochloric acid salt of regorafenib (also known as BAY 73-4506), is a potent inhibitor of multi-kinase including VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 values of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM in cell-free assays, respectively. |
|
V0072
|
Regorafenib monohydrate (BAY73-4506)
|
1019206-88-2 |
Regorafenib monohydrate(also known as BAY 73-4506 monohydrate), the hydrated form ofRegorafenib, is an orally bioavailable multi-kinase inhibitor targeting kinases such as VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 values of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM in cell-free assays, respectively. |