yingweiwo

Adrenergic Receptor

Adrenergic Receptor

The catecholamines, in particular norepinephrine and epinephrine, are targets of the G protein-coupled receptor class known as adrenergic receptors. These receptors are found on numerous cells, and when a catecholamine binds to one of these receptors, the sympathetic nervous system is typically stimulated. The fight-or-flight response is controlled by the sympathetic nervous system, which causes the eye pupils to dilate, the body to mobilize energy, and the blood supply to skeletal muscle to be diverted from non-essential organs.There are numerous subtypes of the two main groups of adrenergic receptors, and. The receptor subtypes 1 and 2 exist. There are three subtypes of receptors: 1, 2, and 3. They are all associated with Gs proteins, which are associated with adenylate cyclase. Thus, antagonist binding increases the level of the second messenger cAMP inside of the cell. The cAMP-dependent protein kinase (PKA), one of cAMP's downstream effectors, mediates some intracellular processes after hormone binding.

Adrenergic Receptor related products

Structure Cat No. Product Name CAS No. Product Description
(+)-Sotalol ((S)-Sotalol) V71347 (+)-Sotalol ((S)-Sotalol) 30236-32-9 (+)-Sotalol ((S)-Sotalol) is the S-isomer of Sotalol.
(-)-Scopolamine (Atroscine) V71260 (-)-Scopolamine (Atroscine) 138-12-5 (-)-Scopolamine (Atroscine) is an isomer of Scopolamine.
(Des-His6)-ACTH (1-24) (human, bovine, rat) V71318 (Des-His6)-ACTH (1-24) (human, bovine, rat) 1926163-11-2 (Des-His6)-ACTH (1-24) (human, bovine, rat) is an analog of adrenocorticotropic hormone (ACTH).
(R)-(+)-Atenolol V71238 (R)-(+)-Atenolol 56715-13-0 (R)-(+)-Atenolol is the less active enantiomer of (R,S)-atenolol.
(R)-9-Hydroxy Risperidone-d4 V79234 (R)-9-Hydroxy Risperidone-d4 (R)-9-Hydroxy Risperidone-d4 is the deuterium labelled form of (R)-9-Hydroxy Risperidone.
(R)-Carvedilol V40138 (R)-Carvedilol 95093-99-5 (R)-Carvedilol is an optically active and R-enantiomer of Carvedilol, which is a nonselective ß-adrenergic blocker with a1-blocking activity.
(R)-Metoprolol-d7 (Metoprolol d7) V71303 (R)-Metoprolol-d7 (Metoprolol d7) 1292907-84-6 (R)-Metoprolol-d7 is the deuterium labelled form of Metoprolol.
(R,R)-Reboxetine mesylate ((R,R)-FCE20124 mesylate; (R,R)-PNU155950E mesylate) V70516 (R,R)-Reboxetine mesylate ((R,R)-FCE20124 mesylate; (R,R)-PNU155950E mesylate) 105017-39-8 (R,R)-Reboxetine mesylate is an antidepressant with good bioavailability.
(rac)-Dobutamine-d4 hydrochloride V71297 (rac)-Dobutamine-d4 hydrochloride 1246815-74-6 (rac)-Dobutamine-d4 ( HCl) is the deuterated racemate of Dobutamine HCl.
(rac)-Dobutamine-d6 hydrochloride V71323 (rac)-Dobutamine-d6 hydrochloride 1246818-96-1 (rac)-Dobutamine-d6 ( HCl) is the deuterated racemate of Dobutamine HCl.
(rac)-Nebivolol-d4 (Nebivolol-d4) V71355 (rac)-Nebivolol-d4 (Nebivolol-d4) 1219407-55-2 (rac)-Nebivolol-d4 is the deuterated racemate of Nebivolol.
(Rac)-Talinolol-d5 V71312 (Rac)-Talinolol-d5 1215343-94-4 (Rac)-Talinolol-d5 is the racemic deuterated form of Talinolol.
(Rac)-Zenidolol (ICI118551) hydrochloride V71276 (Rac)-ICI-118551 hydrochloride 1217094-53-5 (Rac)-ICI-118551 HCl is a selective beta2-adrenergic receptor antagonist.
(RS)-Butyryltimolol V71345 (RS)-Butyryltimolol 2320274-78-8 (RS)-Butyryltimolol is the racemate of Butyryltimolol.
(S)-(-)-Propranolol hydrochloride ((S)-(-)-Propranolol hydrochloride) V71344 (S)-(-)-Propranolol hydrochloride ((S)-(-)-Propranolol hydrochloride) 4199-10-4 (S)-(-)-Propranolol HCl is an adrenergic receptor (β-adrenergic receptor) antagonist (inhibitor) with log Kds of -8.16, -9.08 and -6.93 for β1, β2, and β3 respectively.
(S)-Metoprolol-d7 (Metoprolol d7) V71267 (S)-Metoprolol-d7 (Metoprolol d7) 1292906-91-2 (S)-Metoprolol-d7 is the deuterium labelled form of Metoprolol.
(S)-Terazosin V37874 (S)-Terazosin 109351-33-9 S)-Terazosin is the S-enantiomer of Terazosin,which is a selective α1-adrenoceptor antagonist used for treatment of symptoms of BPH (benign prostatic hyperplasia, an enlarged prostate).
(±)-N-Methylcolaurine V71313 (±)-N-Methylcolaurine 1472-62-4 (±)-N-Methylcolaurine is a selective α2-adrenergic receptor blocker (antagonist).
(±)-Penbutolol-d9 hydrochloride ((Rac)-Penbutolol-d9 (hydrochloride); (±)-Isopenbutolol-d9 (hydrochloride)) V71279 (±)-Penbutolol-d9 hydrochloride ((Rac)-Penbutolol-d9 (hydrochloride); (±)-Isopenbutolol-d9 (hydrochloride)) 1346605-01-3 (±)-Penbutolol-d9 (HCl) is a deuterium-labeled (±)-Penbutolol HCl.
2-Methoxyidazoxan monohydrochloride (RX821002 hydrochloride) V71237 2-Methoxyidazoxan monohydrochloride (RX821002 hydrochloride) 109544-45-8 2-Methoxyidazoxan mono HCl (RX821002 HCl) is a selective alpha 2r adrenergic receptor antagonist (inhibitor) with little or no antagonism to imidazoline.
Contact Us