|
V60051
|
4-(Methylhydroxyphosphinyl)-2-oxobutyric acid
|
79778-02-2 |
|
|
V3441
|
ARN272
|
488793-85-7 |
ARN272 is a novel, potentinhibitor ofanandamide transport. |
|
V3424
|
CID-797718
|
370586-05-3 |
CID797718 is novel potent and selective PKD (Protein kinase D) inhibitor. |
|
V60046
|
Cystathionine-γ-lyase-IN-1
|
2165706-30-7 |
Cystathionine-γ-lyase-IN-1 is a selective cystathionine-γ-lyase (CSE) inhibitor (antagonist) with IC50 of 6.3 μM. |
|
V3407
|
Eleclazine
|
1443211-72-0 |
Eleclazine (also known as GS-6615) is a novel late Na+ current inhibitor with IC50 value of 0.7 uM. |
|
V3536
|
GSK 525768A
|
1260530-25-3 |
GSK 525768A is the inactive enantiomer of GSK525762A, and has no activity towards BET. |
|
V3555
|
GSK-J2
|
1394854-52-4 |
GSK-J2 is the isomer of GSK-J1 without any specific activity. |
|
V3550
|
GSK2807
|
2245255-65-4 |
GSK2807 (GSK-2807) is a novel, potent, selective and SAM-competitive inhibitor ofSMYD3(SET And MYND Domain Containing 3) with anticancer activity. |
|
V3600
|
GSK2838232
|
1443461-21-9 |
GSK2838232, a betulin derivative, is a novel and potent inhibitor of human immune virus (HIV) maturation that is being developed for the treatment of chronic HIV infection. |
|
V3554
|
GSK598809
|
1310803-30-5 |
GSK598809 is a novel, potent and selective dopamine D3 Receptor(DRD3)antagonist with apKiof 8.9. |
|
V3423
|
kb-NB77-78
|
1350622-33-1 |
kb-NB77-78 is a CID797718 analog but without PKD (Protein kinase D) inhibitory activity. |
|
V3547
|
KRN 7000
|
158021-47-7 |
KRN 7000 is a novel, potent and selective synthetic α-galactosylceramide whichactivates NKT immune cells byassociation with the antigen-presenting CD1d protein. |
|
V3404
|
TPT-260
|
769856-81-7 |
TPT-260 (also known as TPU260 and R55) is a thiophene thiourea derivative with molecule weight 260.00 in free base form; There is no formal name yet, it is temporally called as TPT-260. |
|
V3390
|
Salmeterol (GR33343X)
|
18910-65-1 |
Salmeterol (AHR-3929;GR33343X; AHR3929;GR-33343G;Salmetedur, Serevent) is a potent and long-acting β2-adrenergic receptor agonist with anti-inflammatory effects (Kiof 1.5 nM for WT β2AR). |
|
V3513
|
Garenoxacin mesylate (BMS284756)
|
223652-82-2 |
Garenoxacin mesylate(formerly known asT-3811ME;BMS-284756; tradename: Geninax), themesylate salt ofGarenoxacin, is a novel and orally bioavailable quinolone antibiotic effective against both Gram-positive and Gram-negative bacterial infections. |
|
V60050
|
Collagenase I, from Clostridium histolyticum
|
9001-12-1 |
Collagenase is an enzyme that disrupts the peptide bonds of collagen. |
|
V3401
|
Afobazole (CM 346; Fabomotizole)
|
173352-21-1 |
Fabomotizole (also known as CM346; CM-346;Fabomotizole; trade name: Afobazole) is a novel and selective anxiolytic drug thatproduces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions. |