| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V112402 | 2'-Hydroxybiphenyl-3-carboxylic acid | 893736-72-6 | 2'-Hydroxybiphenyl-3-carboxylic acid is an inhibitor of β-lactamase oxa-48 (IC50 = 50 µM; Kd = 1750 µM). |
|
V110473 | 3-Cyanochromone | 50743-17-4 | 3-Cyanoxychrome (compound fragment 1) is a dual inhibitor of NDM-1 and VIM-2, with KD values of 181 μM and 999 μM, respectively. |
|
V116335 | CB-618 | 1463520-70-8 | CB-618 is a β-lactamase inhibitor. |
|
V115972 | Ciprofloxacin prodrug-1 | 2418537-98-9 | Ciprofloxacin prodrug-1 (compound 35) is a β-lactamase-activated prodrug. |
|
V120072 | D-CS319 | 1770826-25-9 | D-CS319 is a potent metallo-β-lactamase (MBL) inhibitor with IC50 values of 2.0 and 3.0 μM for IMP-1 and IMP-78, respectively. |
|
V107888 | Doxazosin impurity 12 | 2066-93-5 | Doxazosin impurity 12 is a CTX-M β-lactamase inhibitor with a Ki value of 0.7 mM for CTX-M. |
|
V114397 | KSP-1007 | 2380240-20-8 | KSP-1007 is a broad-spectrum β-lactamase inhibitor based on bicyclic borate esters. |
|
V114494 | LN-1-255 sodium | 247115-03-3 | LN-1-255 sodium is a β-lactamase inhibitor. |
|
V118762 | MBL-IN-6 | MBL-IN-6 (compound 6d) is a metallo-β-lactamase (MBL) inhibitor with a Ki value of 2.6 μM for NDM-1 and 0.08 μM for VIM-2. | |
|
V88213 | Metallo-β-lactamase-IN-13 | 1802366-23-9 | Metallo-β-lactamase-IN-13 (Compound 13i) is a pan-metallo-β-lactamase inhibitor. |
|
V88216 | Metallo-β-lactamase-IN-14 | 1802367-43-6 | Metallo-β-lactamase-IN-14 (Compound 17e) is a Metallo-β-Lactamase inhibitor. |
|
V88214 | Metallo-β-lactamase-IN-15 | 1804934-57-3 | Metallo-β-lactamase-IN-15 (Compound ±13) is a potent MBL inhibitor with IC50 values of 0.29 μM, 0.088 μM and 0.063 μM for NDM-1, IMP-1 and VIM-2, respectively. |
|
V115729 | ML121 | 1212185-26-6 | ML121 is a selective and potent VIM-2 inhibitor with an IC50 of 54 nM and a Ki of 148 nM. |
|
V84317 | N-Cbz-D-Cysteine (Cbz-D-Cys) | 156916-81-3 | |
|
V84188 | N-Cbz-L-Cysteine (Cbz-cysteine) | 53907-29-2 | |
|
V118339 | NDM-1-IN-10 | 3044733-61-8 | NDM-1-IN-10 (compound CS-23) is an irreversible covalent New Delhi metallo-β-lactamase-1 (NDM-1) inhibitor with an IC50 of 36 nM. |
|
V111246 | NDM-1-IN-11 | NDM-1-IN-11 is a potent covalent inhibitor of NDM-1 with an IC50 value of 1.12 μM. | |
|
V111178 | NDM-1-IN-12 | NDM-1-IN-12 (compound 10c) is an NDM-1 metallo-β-lactamase inhibitor with an IC50 value of 9 nM. | |
|
V119428 | NDM-1-IN-9 | NDM-1-IN-9 (compound M7) is an orally effective NDM-1 inhibitor with a Ki value of 3.95 nM. | |
|
V111839 | rel-Avibactam sodium | 1383814-68-3 | rel-Avibactam (NXL-104) sodium is a β-lactamase inhibitor with broad-spectrum antibacterial activity. |