| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V4914 | GNE-616 | 2349371-81-7 | GNE-616 is a novel, highly potent, metabolically stable, orally bioavailable, and subtype selectiveNav1.7inhibitor with Kiof 0.79 nM andKdof 0.38 nM for hNav1.7. |
|
V4554 | GNE-8505 | 1620573-48-9 | GNE-8505 is a novel, potent and orally bioavailable inhibitor ofDual leucine zipper kinase (DLK). |
|
V4558 | GNE-955 | 1527523-39-2 | GNE-955 is a novel, potent and orally bioavailable panPim kinaseinhibitor withKis of 0.018, 0.11, 0.08 nM for Pim1, Pim2, Pim3, respectively. |
|
V4758 | GS-6207 | 2189684-45-3 | GS-6207 (CA inhibitor 1) is a novel and potentHIVcapsid inhibitor that inhibits HIV virus and has the potential for HIV treatment. |
|
V2196 | GSK-973 | 2138473-38-6 | GSK973 is a selective oral bioavailable inhibitor of BET family BD2s, with pIC50 of 7.8 and a pKd of 8.7 for BRD4 BD2. |
|
V4570 | GSTO-IN-2 | 1202710-57-3 | GSTO-IN-2 is a novel and potent glutathione S-transferaseinhibitor withIC50s of 3.6, 16.3, and 1.4 μM for GSTA2, GSTM1, and GSTP1-1. |
|
V4723 | Guaiapate | 852-42-6 | Guaiapate is a cough suppressant. |
|
V4917 | GW 766994 | 408303-43-5 | GW766994 (GW-766994) is a novel, potent, specific and orally bioavailablesmall molecule antagonist of the CCR3 (chemokine receptor-3) receptor. |
|
V4925 | GW-274150 | 210354-22-6 | GW-274150 is a novel, potent, arginine-competitive,highly selective, NADPH-dependent, and long-acting inhibitor of inducible nitric oxide synthase (iNOS) activity in rat and mouse models of renal I/R. |
|
V4919 | GW-311616 | 198062-54-3 | GW311616 (GW-311616), thefree base form of GW311616A, is a novel, potent, intracellular, orally bioavailable, long duration inhibitor of human neutrophil elastase(HNE) with IC50 of 22 nM. |
|
V4927 | GW-406381 | 221148-46-5 | GW406381 is a novel, potent and highly selectivecyclooxygenase-2 (COX-2)inhibitor that is able to attenuate spontaneous ectopic discharge in sural nerves of rats following chronic constriction injury. |
|
V4922 | GW5638 | 155701-61-4 | Etacstil formerly also known as GW-5638 and DPC-974) is a novel and potent estrogen receptor ligand which is similar to tamoxifen. |
|
V4920 | GW7604 | 195611-82-6 | GW7604 is an antiestrogen. |
|
V5110 | Iberin (NSC-321801) | 505-44-2 | Iberin (NSC 321801), a sulfoxide analog of sulforaphane, is a naturally occurring antioxidant that is a member of isothiocyanate family. |
|
V4746 | IMD-0560 | 439144-66-8 | IMD-0560 is a novel and potent IKK inhibitor which suppresses heart failure and chronic remodeling after myocardial ischemia via MMP alteration. |
|
V4599 | Imiglitazar | 250601-04-8 | Imiglitazar (also known as TAK559; proposed tradename Pargluva) is a novel, potent and dual human peroxisome proliferator-activated receptor PPARα and PPARγ1 agonist with EC50 values of 67 and 31 nM and with hypoglycemic activity. |
|
V4627 | Inarigivir | 475650-36-3 | Inarigivir (formerly also known as ORI-9020; SB-9000) is a novel and potent dinucleotide which can significantly reduce liver HBV DNA in transgenic mice expressing hepatitis B virus. |
|
V5006 | ITIC | 1664293-06-4 | ITIC, athermally stable electron-accepting small molecule used for organic photovoltaic applications (OPV), is anon-fullerene acceptor that canundergo a glass-crystal transition considerably below its high Tg of 180 °C. |
|
V4508 | JNJ-47117096 HCl | 1610536-69-0 | JNJ-47117096 HCl (also known as MELK-T1), identified from a fragment-based drug design, is a novel, potent and selectiveMELK (maternal embryonic leucine zipper kinase)inhibitor with anIC50of 23 nM, it also effectively inhibitsFlt3, with anIC50of 18 nM. |
|
V4500 | JNJ-49153390 | JNJ-49153390 is a novel and potent inhibitor of respiratory syncytial virus (RSV). |
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