|
V4763
|
Vecabrutinib |
1510829-06-7 |
Vecabrutinib (formerlySNS-062; FP-182, BSK-4841 and BIIB-062) is a novel, potent, and reversible/noncovalent BTK and ITK inhibitor with Kd of 0.3 nM and 2.2 nM, respectively; Vecabrutinib shows an IC50 of 24 nM for ITK. |
|
V4767
|
VHL Ligand 3 |
1448189-98-7 |
(S,R,S)-AHPC-Boc (VH032-Boc) is a ligand used to recruit von-Hippel-Lindau (VHL) proteins. |
|
V4707
|
VZ185 |
2306193-61-1 |
VZ185 is a potent, fast, and selective degrader of BRD9 and of its close homolog BRD7. |
|
V4998
|
Way 100135 |
133025-23-7 |
WAY-100135 (WAY100135) is a novel and potent serotonergic drug of the phenylpiperazine family for scientific research. |
|
V4996
|
WAY-151932 |
220460-92-4 |
WAY-151932 (also known as VNA-932; WAY-VNA 932)is a novel and potent vasopressin V2-receptor agonist with IC50of 80.3 nM and 778 nM in human-V2binding and V1abinding assay. |
|
V4995
|
WAY-163909 |
428868-32-0 |
WAY-163909 is a novel, potent and selective 5-HT(2C) receptor agonist with a Kiof 10.5±1.1 nM. |
|
V5002
|
WAY-204688 (SIM-688) |
796854-35-8 |
WAY-204688 (WAY204688; WAY 204688;SIM688; SIM-688) is a novel, potent, selective and orally bioactive agonist of estrogen receptor (ER-α) and also an inhibitor ofNF-κBtranscriptional activity with anti-inflammatory effects. |
|
V4997
|
WAY127093B racemate |
145743-63-1 |
WAY127093B racemate, the racemic mixture of WAY127093B, is a novel, potent and orally bioavailable phosphodiesterase IV inhibitor in guinea pigs and rats. |
|
V4939
|
WU-07047 |
1702378-78-6 |
WU-07047 (WU07047) is a novel and potent inhibitor of Gαq/11, it is a simplified analog of the selective Gαq/11 inhibitor YM-25489. |
|
V4733
|
Xantocillin |
580-74-5 |
Xanthocillin (also known as xanthocillin X or ophthocillin) is a marine product isolated from Penicillium commune, it was reported to be able to induceautophagythrough inhibition of theMEK/ERKpathway. |
|
V4938
|
YM-254890 |
568580-02-9 |
YM-254890 (YM254890),a cyclic depsipeptide discovered from Chromobacterium sp. |
|
V4889
|
Zatosetron maleate |
123482-23-5 |
Zatosetron maleate is a potent and specific 5HT3 receptor blocker (antagonist). |