Others 8

Angiogenesis

5-alpha Reductase ALK Bcr-Abl BTK EGFR FAK FLT3 HER-2 HIF Src Syk VDA VEGFR
Anti-infection

Antibiotic Arenavirus Bacterial CMV EBV Enterovirus Filovirus Fungal Gli HBV HCV HCV Protease HIV HSV Influenza Virus Parasite RABV Reverse Transcriptase RSV SARS-CoV TMV Virus Protease
Apoptosis

Apoptosis ASK Bcl-2 Caspase c-Myc c-RET Cytohesin DAPK Ferroptosis FKBP IAP Mdm2 p53 PD-1 PD-L1 PERK PKD Ras RIP kinase ROS Survivin Thymidylate Synthase TNF Receptor TNFa TRADD
Autophagy

Autophagy LRRK2 Mitophagy OGA ULK
Cell Cycle

Antifolate APC Aurora Kinase BMI-1 CDK Chk c-Myc Eukaryotic Initiation Factor G-quadruplex HDAC HSP Kinesin LIMK Mad2 Microtubule(Tubulin) Mps1 Nucleoside Antimetabolite/Analog Nur77 p21 PAK PERK PFKFB PLK PPAR Ras Rho ROCK SRPK TOPK Topoisomerase Wee1
Cytoskeletal Signaling

Arp2 3 Complex Bcr-Abl Cardiac Myosin Dynamin Gap Junction Protein HSP Integrin Kinesin Microtubule Associated MLCK Myosin PAK TACC3 Wntbeta-catenin
DNA Damage

ATM(ATR) CRISPR(Cas9) DNA alkylator DNA Stain DNA(RNA) Synthesis GAK HDAC HSP Nucleoside Antimetabolite(Analog) OGG1 p97 PARG PARP RAD51 RNR Sirtuin SMN Telomerase Topoisomerase
Endocrinology & Hormones

5-alpha Reductase ACE Adrenergic Receptor Androgen Receptor Aromatase Estrogenprogestogen Receptor Glucocorticoid Receptor GPR Mineralocorticoid Receptor RAAS THR TSH Receptor
Epigenetics

AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain EZH1 2 HDAC HIF Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MAT MicroRNA MLL Pim PKC Protein Arginine Deiminase Sirtuin Small Interfering RNA (siRNA) SMYD
GPCR & G Protein

5-HT Receptor Adenosine Receptor Adenylate Cyclase Adrenergic Receptor Angiotensin Receptor APJ Bombesin Receptor Bradykinin Receptor cAMP Cannabinoid Receptor CaSR CCK receptor CCR CGRP Receptor CRFR CXCR Dopamine Receptor EBI2 Endothelin Receptor Formyl Peptide Receptor Free Fatty Acid Receptor G protein-coupled Bile Acid Receptor GCGR GHSR GLP Receptor Glucagon Receptor GnRH Receptor GPCR19 GPR GPR109A Guanylate Cyclase Hedgehog(Smoothened) ROCK Histamine Receptor ICMT Leukotriene Receptor LPA Receptor LPL Receptor LTR mAChR Melanocortin Receptor Melatonin Receptor mGluR Motilin Receptor MRGPR MT Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor NPY receptor Opioid Receptor OX Receptor Oxytocin Receptor P2Y Receptor PAFR PAR PKD PKG Prostaglandin Receptor Ras RGS Protein S1P Receptor SGLT Sigma Receptor Somatostatin Receptor TAAR TSH Receptor Urotensin Receptor Vasopressin Receptor

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Others 8

Others 8 related products

Cat No.	Product Name	CAS No.	Product Description
V3608	Echinocandin B	54651-05-7	Echinocandin B is a novel and potent cyclic hexapeptide echinocandin antibioticoriginallyisolated from Aspergillus nidulans var.
V3855	Ehp-inhibitor	861249-77-6	Ehp inhibitor is a novel and potent inhibitor of EHP.
V3611	Enantiomer of Sofosbuvir		Enantiomer of Sofosbuvir is the isomer/enantiomer of Sofosbuvir(also known as PSI-7977, GS-7977; tradenames Sovaldi and Virunon) is a HCV NS5B polymerase inhibitor that is used for the treatment of chronic hepatitis C virus (HCV) infection.
V3618	Epelsiban	872599-83-2	Epelsiban (also known asGSK557296; GSK-557296) is a novel, potent, selective and orally bioavailableoxytocin receptorantagonist, with apKiof 9.9 for human oxytocin receptor.
V3638	Epetraborole R-Mandelate	1234563-15-5	Epetraborole R-Mandelate (also known as GSK2251052 and AN3365) is a novel, potent and selective leucyl-tRNA synthetase (LeuRS) inhibitor, which inhibits protein synthesis by binding to the terminal adenosine ribose (A76) of leucyl-tRNA synthetase.
V2104	Flavoxate sulfate	15301-69-6	Flavoxate sulfate (Rec-7-0040; DW61) is a potent anticholinergic (AChR) agent that binds and inhibits muscarinic receptors, thereby suppressing the micturition reflex and increases urinary bladder capacity by modifying the micturition center in the brain stem.
V3587	Foretinib-Based PROTAC 7	2230821-68-6	Foretinib-Based PROTAC 7 is a novel, potent and selective VHL-recruiting PROTAC that induces the degradation of c-Met in a dose- and time-dependent fashion in MDA-MB-231 cells.
V3897	Fosnetupitant	1703748-89-3	Fosnetupitant (07PNET; 07-PNET; Fosnetupitant chloride; Akynzeo), the prodrug of netupitant,is a novel and potentantagonist of neurokinin receptor usedin combination with palonosetron to prevent nausea and vomiting caused by chemotherapy.
V3507	Fosravuconazole	351227-64-0	Fosravuconazole (formerly known as E-1224, BEF-1224, and BMS-379224) is an azole-based antifungal agent that can be potentially used for the treatment of fungal infections.
V2128	GNE-0723	1883518-31-7	GNE 0723 is a novel, potent, brain permeable positive allosteric modulator (PAM) and GluN2A subunit-selective ofNMDAR, with anEC50of 21 nM for GluN2A, 7.4 and 6.2 μM for GluN2C and GluN2D, respectively.
V2125	GNE-207	2158266-58-9	GNE-207 is a novel, potent, selective and orally bioavailable inhibitor of the bromodomain ofCBP.
V2131	GNE-371	1926986-36-8	GNE-371 is a novel, potent and selective chemical probe for the second bromodomains of human transcription-initiation-factorTFIIDsubunit 1 and transcription-initiation-factorTFIIDsubunit 1-like with anIC50of 10 nM for TAF1(2).
V2126	GNE-493	1033735-94-2	GNE-493 is a novel, potent, selective, and orally bioavailable dualpan-PI3-kinase/mTORinhibitor withIC50s of 3.4 nM, 12 nM, 16 nM, 16 nM and 32 nM for PI3Kα, PI3Kβ, PI3Kδ, PI3Kγ and mTOR.
V2130	GNE-5729	2026635-66-3	GNE 5729 is a novel, potent, brain permeable positive allosteric modulator (PAM) and GluN2A subunit-selective ofNMDAR with anEC50of 37 nM for GluN2A, 4.7 and 9.5 μM for GluN2C and GluN2D, respectively.
V2123	GNE-6468	1677668-27-7	GNE-6468 is a novel, potent and selectiveRORγ (RORc)agonists with anEC50value of 13 nM in HEK-293 cells.
V2133	GNE684		GNE684 is a novel and potent inhibitor ofreceptor interacting protein 1 (RIP1), it inhibits human RIP1 potently over than mouse and rat withIC50s of 21 nM, 189 nM and 691 nM, respectively.
V2122	GNF179	1261114-01-5	GNF179, an optimized 8,8-dimethylimidazolopiperazine analog,is a novel, potent and orally bioavailable antiparasitic agent that exhibited the potency(4.8 nM against the multidrug resistant strain W2) in vitro metabolic stability and in vivo oral bioavailability.
V3539	GSK-269984A	892664-04-9	GSK-269984A is a novel and potentProstaglandin E2 Receptor 1 (EP1)antagonist with apIC50of 7.9.
V2062	GSK1379725A	1802251-00-8	GSK1379725A (AU1) is the first small molecule selective for BPTF over Brd4, as an inhibitor ofBrd4and a selective BPTF ligand with Kdof 2.8 μM.
V3592	GSK2973980A	1414797-35-5	GSK2973980A is a novel, potent and selective inhibitor ofAcyl-CoA:diacylglycerol acyltransferase 1 (DGAT1)with anIC50of 3 nM.