Others 8

Angiogenesis

5-alpha Reductase ALK Bcr-Abl BTK EGFR FAK FLT3 HER-2 HIF Src Syk VDA VEGFR
Anti-infection

Antibiotic Arenavirus Bacterial CMV EBV Enterovirus Filovirus Fungal Gli HBV HCV HCV Protease HIV HSV Influenza Virus Parasite RABV Reverse Transcriptase RSV SARS-CoV TMV Virus Protease
Apoptosis

Apoptosis ASK Bcl-2 Caspase c-Myc c-RET Cytohesin DAPK Ferroptosis FKBP IAP Mdm2 p53 PD-1 PD-L1 PERK PKD Ras RIP kinase ROS Survivin Thymidylate Synthase TNF Receptor TNFa TRADD
Autophagy

Autophagy LRRK2 Mitophagy OGA ULK
Cell Cycle

Antifolate APC Aurora Kinase BMI-1 CDK Chk c-Myc Eukaryotic Initiation Factor G-quadruplex HDAC HSP Kinesin LIMK Mad2 Microtubule(Tubulin) Mps1 Nucleoside Antimetabolite/Analog Nur77 p21 PAK PERK PFKFB PLK PPAR Ras Rho ROCK SRPK TOPK Topoisomerase Wee1
Cytoskeletal Signaling

Arp2 3 Complex Bcr-Abl Cardiac Myosin Dynamin Gap Junction Protein HSP Integrin Kinesin Microtubule Associated MLCK Myosin PAK TACC3 Wntbeta-catenin
DNA Damage

ATM(ATR) CRISPR(Cas9) DNA alkylator DNA Stain DNA(RNA) Synthesis GAK HDAC HSP Nucleoside Antimetabolite(Analog) OGG1 p97 PARG PARP RAD51 RNR Sirtuin SMN Telomerase Topoisomerase
Endocrinology & Hormones

5-alpha Reductase ACE Adrenergic Receptor Androgen Receptor Aromatase Estrogenprogestogen Receptor Glucocorticoid Receptor GPR Mineralocorticoid Receptor RAAS THR TSH Receptor
Epigenetics

AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain EZH1 2 HDAC HIF Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MAT MicroRNA MLL Pim PKC Protein Arginine Deiminase Sirtuin Small Interfering RNA (siRNA) SMYD
GPCR & G Protein

5-HT Receptor Adenosine Receptor Adenylate Cyclase Adrenergic Receptor Angiotensin Receptor APJ Bombesin Receptor Bradykinin Receptor cAMP Cannabinoid Receptor CaSR CCK receptor CCR CGRP Receptor CRFR CXCR Dopamine Receptor EBI2 Endothelin Receptor Formyl Peptide Receptor Free Fatty Acid Receptor G protein-coupled Bile Acid Receptor GCGR GHSR GLP Receptor Glucagon Receptor GnRH Receptor GPCR19 GPR GPR109A Guanylate Cyclase Hedgehog(Smoothened) ROCK Histamine Receptor ICMT Leukotriene Receptor LPA Receptor LPL Receptor LTR mAChR Melanocortin Receptor Melatonin Receptor mGluR Motilin Receptor MRGPR MT Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor NPY receptor Opioid Receptor OX Receptor Oxytocin Receptor P2Y Receptor PAFR PAR PKD PKG Prostaglandin Receptor Ras RGS Protein S1P Receptor SGLT Sigma Receptor Somatostatin Receptor TAAR TSH Receptor Urotensin Receptor Vasopressin Receptor

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Others 8

Others 8 related products

Cat No.	Product Name	CAS No.	Product Description
V3542	GSK3004774	2138814-32-9	GSK3004774 is a novel, potent, nonabsorbable agonist ofCaSR, with anpEC50of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively.
V3593	GSK318689	1972617-87-0	GSK3186899 (also known as DDD-853651) is a novel and potent inhibitor of cdc-2-related kinase 12 (CRK12), with anEC50of 1.4 μM forL.
V3617	GSK3395879	2215852-91-6	GSK3395879 is a novel, potent, selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with anIC50of 1 nM for hTRPV4.
V3604	GSK376501A	1010412-80-2	GSK376501A is a novel,, potent and selective peroxisome proliferator-activated receptor gamma (PPARγ) modulator that has the potential for the treatment of type 2 diabetes mellitus.
V4394	INDACRINONE	57296-63-6	Indacrinone (MK196; Indacrynic acid; Indanone)is an investigational loop diuretic which can be used in patients of gout with hypertension as an antihypertensive because it decreases reabsorption of uric acid.
V4379	IPILIMUMAB	477202-00-9	Ipilimumab (trade name Yervoy; also known as MDX-010; BMS-734016) is a fully human monoclonal IgG1κ antibody against the cytotoxic T-lymphocyte antigen-4 (CTLA-4), which is an immune-inhibitory molecule expressed in activated T cells and in suppressor T regulatory cells.
V2120	JNJ-18038683	851373-91-6	JNJ-18038683 is a novel and potent antagonist of 5-Hydroxytryptamine Type 7 (5-HT7) receptor withpKisof 8.19, 8.20 for rat and human 5-HT7in HEK293 cells, respectively.
V2118	JNJ-47965567	1428327-31-4	JNJ-47965567 is a novel, potent,centrally permeable, high affinity and selective antagonist of the purinergic receptor P2X subtype 7 (P2X7), which is a ligand-gated ion channel.
V3546	KD-3010	934760-90-4	KD-3010 is a potent, orally bioactive, and selective agonist of peroxisome proliferator-activated receptordelta(PPARδ)that can be potentially used for the treatment of diabetes and obesity.
V4099	KMUP-1	81996-46-5	KMUP-1, a xanthine derivative, has been demonstrated to modulate K+-channel activity in smooth muscles and is a stimulator of the NO/sGC/cGMP pathway.
V4100	KMUP-3	421556-16-3	KMUP-3, a xanthine derivative, has been demonstrated to modulate K+-channel activity in smooth muscles and is a stimulator of the NO/sGC/cGMP pathway.
V4102	KT5823	126643-37-6	KT5823 (KT-5823),a staurosporine-related analog,is a selective inhibitor of protein kinase G (PKG) with anticancer activity.
V2591	L755507	159182-43-1	L-755,507 isidentified as a potent and selective β3 adrenergic receptor partial agonist with EC50 of 0.43 nM, it displayed > 1000-fold selective over β1- and β2-adrenoceptors (EC50 values are 0.43, 580 and > 10000 nM for activation of cloned human β3-, β1- and β2-adrenoceptors respectively).
V2251	LBQ-657 sodium	149709-44-4	Sacubitril (Desethyl Sacubitril) is an active inhibitor of neprilysin (NEP).
V3139	LLY-284	2226515-75-7	LLY-284 (LLY284) is a negative control and tool compound forLLY-283.
V2137	LY-309887	127228-54-0	LY309887 is a novel and potent inhibitor of glycinamide ribonucleotide formyltransferase (GARFT) withKiof 6.5 nM, and has antitumor activity.
V2141	LY285434	159748-08-0	LY285434 is an angiotensin II receptor blocker (antagonist).
V3809	LY3104607	1795232-22-2	LY3104607 is a potent, selective and orally available G Protein-Coupled Receptor 40 (GPR40) agonist with potential antidiabetic application.
V3905	MACIMORELIN	381231-18-1	Macimorelin (formerly known as UMV-1843;EP-1572;AEZS-130; JMV1843; trade name:Macrilen) is a synthetic small molecule agonist of growth hormone secretagogue receptor that has been approved to diagnose growth hormone deficiency.
V3904	MACIMORELIN ACETATE	945212-59-9	Macimorelin acetate (formerly AEZS-130; EP-1572; JMV-1843; trade name:Macrilen), the acetate salt form of Macimorelin, is a novel and potent synthetic small molecule growth hormone secretagogue receptor agonist approved in 2018 for use in the diagnosis of adult growth hormone deficiency.