The ion channel known as the calcium channel exhibits selective permeability to calcium ions. Although there are ligand-gated calcium channels as well, it is sometimes referred to as a voltage-dependent calcium channel. Even though the concentration of Na+ outside of cells is 70 times higher than that of Ca2+, voltage-gated calcium (CaV) channels catalyze a rapid, highly selective influx of Ca2+ into cells. A side effect of some calcium channel blockers is that they slow your heart rate, which helps to lower blood pressure, treat angina, and regulate irregular heartbeats.
| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
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V71504 | Catharanthine Sulfate (vinblastine sulfate; (+)-3,4-Didehydrocoronaridine Sulfate) | 153230-94-5 | Catharanthine Sulfate ((+)-3,4-Didehydrocoronaridine Sulfate) is an alkaloid in Catharanthus roseus. |
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V71525 | Cav 3.2 inhibitor 1 | 2878598-59-3 | Cav 3.2 inhibitor 1 is a T-type calcium channel inhibitor (antagonist) with low binding affinity to dopamine receptor (D2 receptor). |
|
V71493 | Cav 3.2 inhibitor 2 | 2878598-92-4 | Cav 3.2 inhibitor 2 is an inhibitor (blocker/antagonist) of Cav3.2 T-type Ca2+ channels, with IC50 of 0.09339 μM at a constant potential of -80mV. |
|
V71489 | Cav 3.2 inhibitor 3 | 2878598-69-5 | Cav 3.2 inhibitor 3 (Compound 4) is a potent Cav3.2 T-type Ca2+ channel inhibitor (antagonist) with IC50 of 0.1534 μM and low binding affinity to D2 receptors. |
|
V71524 | Cav 3.2 inhibitor 4 | 1416984-93-4 | Cav 3.2 inhibitor 4 (compound 21) is a potent, peripherally restricted and selective T-type calcium channel (Cav3.2) inhibitor (antagonist) with IC50 of 0.6 μM. |
|
V71477 | CaV1.3 antagonist-1 | 1391385-57-1 | CaV1.3 antagonist-1 is a potent and selective CaV1.3 L-type calcium channel antagonist (inhibitor) with IC50 of 1.7 μM. |
|
V71482 | Cavα2δ-IN-1 | 2416957-09-8 | Cavα2δ-IN-1 is selective for voltage-gated calcium channels, with a Ki of 6 nM for Cavα2δ-1 and greater than 10000 nM for Cavα2δ-2. |
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V71532 | Cavα2δ1&NET-IN-1 | 2314361-39-0 | Cavα2δ1&NET-IN-1 (Compound 59S) is a dual (bifunctional) inhibitor of voltage-gated calcium channel α2δ-1 subunit (Cavα2δ-1) and norepinephrine transporter (NET). |
|
V71514 | Cavα2δ1&NET-IN-2 | 2143586-17-6 | Cavα2δ1&NET-IN-2 (Compound 45CS) is a dual (bifunctional) inhibitor of voltage-gated calcium channel α2δ-1 subunit (Cavα2δ-1) and norepinephrine transporter (NET). |
|
V71520 | Cavα2δ1&NET-IN-3 | 2143584-82-9 | Cavα2δ1&NET-IN-3 (example 216) is an inhibitor (blocker/antagonist) of voltage-gated calcium channel (VGCC) subunit α2δ and norepinephrine transporter (NET). |
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V78822 | Clevidipine-d7 (clevidipine d7) | Clevidipine-d7 is the deuterated form of Clevidipine. | |
|
V71483 | Crisugabalin (HSK16149) | 2209104-84-5 | Crisugabalin (HSK16149) is a novel voltage-gated calcium channel (VGCC) α2δ subunit ligand. |
|
V78947 | Cyclic ADP-ribose ammonium (cADPR ammonium) | Cyclic ADP-ribose ammonium (cADPR ammonium) is a potent calcium mobilization second messenger synthesized from NAD+ by ADP-ribosyl cyclase. | |
|
V71537 | Diltiazem-(acetoxy-d3) (hydrochloride) | 1217860-13-3 | Diltiazem-(acetoxy-d3) ( HCl) is the deuterated form of Diltiazem HCl. |
|
V71518 | Diltiazem-d3 hydrochloride (Diltiazem d3 hydrochloride (hydrochloride)) | 1217623-80-7 | Diltiazem-d3 ( HCl) is the deuterium labelled form of Diltiazem HCl. |
|
V79175 | DL-Phenylalanine-d5 hydrochloride (2-Amino-3-phenylpropionic acid-d5 (hydrochloride)) | DL-Phenylalanine-d5 ( HCl) is the deuterated form of DL-Phenylalanine. | |
|
V79176 | Drotaverine-d10 hydrochloride | Drotaverine-d10 ( HCl) is the deuterium labelled form of Drotaverine HCl. | |
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V2837 | Ebselen | 60940-34-3 | Ebselen (formerly SPI-1005;PZ-51; DR-3305;CCG-39161), is an organoselenium-based small molecule biochemical compound with potential anti-inflammatory, anti-oxidant, and cytoprotective activity. |
|
V71517 | Etiracetam-d3 (UCB 6474-d3) | 2714408-84-9 | Etiracetam-d3 is the deuterated form of Etiracetam. |
|
V79401 | Fenoverine-d8 (Spasmopriv-d8) | Fenoverine-d8 is the deuterium labelled form of Fenoverine. |
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