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GPR

GPR

GPR related products

Structure Cat No. Product Name CAS No. Product Description
(S)-CVN424 V75415 (S)-CVN424 1799968-74-3 (S)-CVN424 is a potent modulator of G protein-coupled receptor 6 (GPR6).
2-Oleoylglycerol (2-octadecenoic acid monoglyceride; 2-glyceryl monooleate) V70305 2-Oleoylglycerol (2-octadecenoic acid monoglyceride; 2-glyceryl monooleate) 3443-84-3 2-Oleoylglycerol is a naturally occurring lipid in the diet.
2-PCCA hydrochloride V77329 2-PCCA hydrochloride 2-PCCA HCl is a racemate and a GPR88 receptor agonist.
[Ala17]-MCH V70558 [Ala17]-MCH 359784-84-2 [Ala17]-MCH is an analog of MCH and is a ligand for MCHR1 (Ki=0.16 nM) with greater selectivity for MCHR2 (Ki=34 nM).
Ac-hMCH(6-16)-NH2 V70561 Ac-hMCH(6-16)-NH2 1053601-50-5 Ac-hMCH(6-16)-NH2 is a non-selective peptide agonist of MCH in human brain, with IC50s of 0.16 nM and 2.7 nM for MCH-1R and MCH-2R, respectively.
AF64394 V6494 AF64394 1637300-25-4 AF64394 is an inverse agonist of GPR3 with pIC50 of 7.3.
AMG-076 V70556 AMG-076 1001438-96-5 AMG-076 is an orally bioactive, selective MCHR1 antagonist.
APD 668 V3354 APD 668 832714-46-2 APD668 (also known as JNJ-28630368) is a novel and potent agonist of the pancreatic and GI-expressed orphan G-protein coupled receptor GPR119, with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119 respectively.
APD597 (JNJ38431055) V2826 APD597 (JNJ38431055) 897732-93-3 APD597 (formerly known as JNJ-38431055) is a novel potent and selective GPR119 agonist/modulator, which has the potential for the treatment of type 2 diabetes.
AR 231453 V29481 AR 231453 733750-99-7 AR231453 (AR-231453) is a potent, selective and orally bioavailable GPR119 agonist used as an antidiabetic agent.
AS1269574 V11653 AS1269574 330981-72-1 AS1269574 is a potent, orally bioactive GPR119 agonist with EC50 of 2.5 μM in HEK293 cells expressing human GPR119.
AZD1981 V1806 AZD1981 802904-66-1 AZD1981 is a novel potent and selective CRTh2 (Chemoattractant receptor-homologous molecule expressed on TH2 cells; DP2-Prostaglandin D2 receptor 2, ) receptor antagonist with IC50 of 4 nM,it displayed>1000-fold selectivity over more than 340 other enzymes and receptors, including DP1.
BI-9508 V86635 BI-9508 BI-9508 is a selective GPR88 agonist that crosses the blood-brain barrier.
BigLEN(mouse) V75408 BigLEN(mouse) 501036-69-7 BigLEN(mouse) is a potent and specific agonist of orphan G protein-coupled receptor 171 (GPR171) with a Kd of approximately 0.5 nM.
BigLEN(rat) V75407 BigLEN(rat) 369377-66-2 BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM.
BigLEN(rat) TFA V78421 BigLEN(rat) TFA BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM.
BRD5080 V130635 BRD5080 BRD5080 is a potent GPR65 positive allosteric modifier.
CID 2745687 V75409 CID 2745687 264233-05-8 CID 2745687 is a specific, reversible and competitive GPR35 antagonist (inhibitor) with Ki of 12.8 nM.
CID-16020046 V5220 CID-16020046 834903-43-4 CID-16020046 (CI-16020046) is a novel, potent and selective GPR55 (LPI receptor) antagonist / inverse agonist which can block GPR55-mediated endothelial wound healing and reverse LPI-inhibited platelet aggregation.
CID1231538 V75410 CID1231538 354126-20-8 CID1231538, a benzothiazole analog, is a potent GPR35 antagonist.
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