Drug Metabolite

Angiogenesis

5-alpha Reductase ALK Bcr-Abl BTK EGFR FAK FLT3 HER-2 HIF Src Syk VDA VEGFR
Anti-infection

Antibiotic Arenavirus Bacterial CMV EBV Enterovirus Filovirus Fungal Gli HBV HCV HCV Protease HIV HSV Influenza Virus Parasite RABV Reverse Transcriptase RSV SARS-CoV TMV Virus Protease
Apoptosis

Apoptosis ASK Bcl-2 Caspase c-Myc c-RET Cytohesin DAPK Ferroptosis FKBP IAP Mdm2 p53 PD-1 PD-L1 PERK PKD Ras RIP kinase ROS Survivin Thymidylate Synthase TNF Receptor TNFa TRADD
Autophagy

Autophagy LRRK2 Mitophagy OGA ULK
Cell Cycle

Antifolate APC Aurora Kinase BMI-1 CDK Chk c-Myc Eukaryotic Initiation Factor G-quadruplex HDAC HSP Kinesin LIMK Mad2 Microtubule(Tubulin) Mps1 Nucleoside Antimetabolite/Analog Nur77 p21 PAK PERK PFKFB PLK PPAR Ras Rho ROCK SRPK TOPK Topoisomerase Wee1
Cytoskeletal Signaling

Arp2 3 Complex Bcr-Abl Cardiac Myosin Dynamin Gap Junction Protein HSP Integrin Kinesin Microtubule Associated MLCK Myosin PAK TACC3 Wntbeta-catenin
DNA Damage

ATM(ATR) CRISPR(Cas9) DNA alkylator DNA Stain DNA(RNA) Synthesis GAK HDAC HSP Nucleoside Antimetabolite(Analog) OGG1 p97 PARG PARP RAD51 RNR Sirtuin SMN Telomerase Topoisomerase
Endocrinology & Hormones

5-alpha Reductase ACE Adrenergic Receptor Androgen Receptor Aromatase Estrogenprogestogen Receptor Glucocorticoid Receptor GPR Mineralocorticoid Receptor RAAS THR TSH Receptor
Epigenetics

AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain EZH1 2 HDAC HIF Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MAT MicroRNA MLL Pim PKC Protein Arginine Deiminase Sirtuin Small Interfering RNA (siRNA) SMYD
GPCR & G Protein

5-HT Receptor Adenosine Receptor Adenylate Cyclase Adrenergic Receptor Angiotensin Receptor APJ Bombesin Receptor Bradykinin Receptor cAMP Cannabinoid Receptor CaSR CCK receptor CCR CGRP Receptor CRFR CXCR Dopamine Receptor EBI2 Endothelin Receptor Formyl Peptide Receptor Free Fatty Acid Receptor G protein-coupled Bile Acid Receptor GCGR GHSR GLP Receptor Glucagon Receptor GnRH Receptor GPCR19 GPR GPR109A Guanylate Cyclase Hedgehog(Smoothened) ROCK Histamine Receptor ICMT Leukotriene Receptor LPA Receptor LPL Receptor LTR mAChR Melanocortin Receptor Melatonin Receptor mGluR Motilin Receptor MRGPR MT Receptor Neurokinin Receptor Neuropeptide Y Receptor Neurotensin Receptor NPY receptor Opioid Receptor OX Receptor Oxytocin Receptor P2Y Receptor PAFR PAR PKD PKG Prostaglandin Receptor Ras RGS Protein S1P Receptor SGLT Sigma Receptor Somatostatin Receptor TAAR TSH Receptor Urotensin Receptor Vasopressin Receptor

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Drug Metabolite

Drug metabolites are created when a drug is metabolized into a different form that still has therapeutic effects. Active metabolites can be produced by drug metabolism redox reactions like heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations. In some rare circumstances, conjugation reactions can also produce an active metabolite.

Drug Metabolite related products

Cat No.	Product Name	CAS No.	Product Description
V72260	Iloperidone metabolite Hydroxy Iloperidone-d3 (P88-d3; Hydroxy Iloperidone-d3)	1504554-02-2	Iloperidone metabolite Hydroxy Iloperidone-d3 is the deuterium labelled form of Iloperidone metabolite Hydroxy Iloperidone.
V72174	Imatinib Impurity E	1365802-18-1	Imatinib Impurity E is an impurity in Imatinib.
V72243	Iso-Sagittatoside A	503456-08-4	Iso-Sagittatoside A is a potent metabolite of Erxian Tang (EXD), a traditional Chinese medicine prescription for menopausal syndrome.
V72219	Isokotanin B	154160-09-5	Isokotanin B is a metabolite of dicoumarin extracted from the sclerotia of Aspergillus alliaceus.
V72182	Ivabradine impurity 1	1428869-91-3	Ivabradine impurity 1 is an impurity of Ivabradine.
V72269	Ivabradine impurity 2 (Ivabradine impurity 19)	73954-34-4	Ivabradine impurity 2 is an impurity of Ivabradine.
V33434	Ivabradine metabolite N-Demethyl Ivabradine hydrochloride	1246638-08-3	Ivabradine metabolite N-Demethyl Ivabradine hydrochloride is the N-demethylated metabolite of ivabradine (S-16257; S16257; S 16257;Corlentor; Coralan;Procoralan;Coraxan; Ivabid; Bradia), which is a cardiac pacemaker current (If) inhibitor and a medication approved in 2015 for the management of stable heart-related chest pain and heart failure.
V72180	IYPTNGYTR	1431957-72-0	IYPTNGYTR, a deamidation-sensitive characteristic peptide, is the deamidation product of Trastuzumab.
V76874	IYPTNGYTR acetate		IYPTNGYTR acetate, a deamidation-sensitive characteristic peptide, is the deamidation product of Trastuzumab.
V72128	Labetalone hydrochloride	96441-14-4	Labetalone HCl is an impurity of Labetalol.
V72107	Linsidomine hydrochloride (SIN-1 chloride)	16142-27-1	SIN-1 (chloride) is the bioactive metabolite of moxidomine, which can relax blood vessels and inhibit platelet aggregation.
V72247	Lurasidone Metabolite 14283-d8	2070009-43-5	Lurasidone Metabolite 14283-d8 is the deuterium labelled form of Lurasidone Metabolite 14283.
V76806	Lurasidone metabolite 14326 hydrochloride (lurasidone hydrochloride)		Lurasidone metabolite 14326 ( HCl) is an bioactive metabolite of the atypical antipsychotic active molecule Lurasidone.
V80636	Lurasidone Metabolite 14326-d8		Lurasidone Metabolite 14326-d8 is the deuterium labelled form of Lurasidone Metabolite 14326.
V40035	m-Nifedipine	21881-77-6	m-Nifedipine is an impurity of Nifedipine (Bay-1040; BAY-a-1040; Cordipin; Corinfar) which is an approved dihydropyridine calcium channel blocker (CCB) used as antihypertensive drug.
V38232	Mebeverine acid	475203-77-1	Mebeverine acid (Mebeverine metabolite Mebeverine acid) is a secondary metabolite (SM, chemical compound) of Mebeverine.
V34673	Mebeverine alcohol (Mebeverine metabolite)	14367-47-6	Mebeverine alcohol is a major metabolite of Mebeverine which is a musculotropic antispasmodic drug.
V32648	meta-Fexofenadine (meta-MDL-16455	479035-75-1	meta-Fexofenadine (meta-MDL-1645; meta-MDL16455) is an impurity of Fexofenadine (Allegra;MDL-16455A; MDL16455A; Telfast), which is a histamine H1 receptor antagonist (antihistamine) approved for the treatment of allergy including hay fever, nasal congestion, and urticaria.
V21871	Molsidomine	25717-80-0	Molsidomine is anorally bioactive and long acting vasodilator acting as anNO donor and annexin A2 inhibitor.
V72215	Mono(5-carboxy-2-ethylpentyl) phthalate (MECPP)	40809-41-4	Mono(5-carboxy-2-ethylpentyl) phthalate (MECPP) is a metabolite of Di-(2-ethylhexyl) phthalate (DEHP).