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Drug Metabolite

Drug Metabolite

Drug metabolites are created when a drug is metabolized into a different form that still has therapeutic effects. Active metabolites can be produced by drug metabolism redox reactions like heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations. In some rare circumstances, conjugation reactions can also produce an active metabolite. 

Drug Metabolite related products

Structure Cat No. Product Name CAS No. Product Description
N-De-2,4-difluorobenzyl dolutegravir V107666 N-De-2,4-difluorobenzyl dolutegravir 1485081-26-2 N-De-2,4-difluorobenzyl dolutegravir is a metabolite of the HIV integrase inhibitor dolutegravir.
N-Demethyl Mifepristone (RU 42633) V67748 N-Demethyl Mifepristone (RU 42633) 104004-96-8 N-Demethyl Mifepristone (RU 42633) is the bioactive metabolite of Mifepristone.
N-Demethylerythromycin A (N-Demethylerythromycin A) V72220 N-Demethylerythromycin A (N-Demethylerythromycin A) 992-62-1 N-Demethylerythromycin A is a metabolite of Erythromycin A.
N-Depropylpropafenone V107798 N-Depropylpropafenone 86383-21-3 N-despropylpropafenone is the active metabolite of propafenone, which is metabolized by the CYP450 enzyme system (mainly CYP2D6). It has a certain antiarrhythmic effect by blocking sodium ion channels and delaying the depolarization process of myocardial cells.
N-Desalkyludenafil V72170 N-Desalkyludenafil 319491-68-4 N-Desalkyludenafil is a metabolite of Udenafil.
N-Desethyl Sunitinib hydrochloride (SU-12662 hydrochloride) V76713 N-Desethyl Sunitinib hydrochloride (SU-12662 hydrochloride) N-Desethyl Sunitinib (SU-12662) ( HCl) is a metabolite of Sunitinib.
N-Desmethyl clomipramine V91139 N-Desmethyl clomipramine 303-48-0 Desmethylclomipramine (Norclomipramine) is a metabolite of clomipramine and can be used in neurological research.
N-Desmethyl imatinib mesylate (Norimatinib mesylate; Imatinib metabolite N-Desmethyl imatinib mesylate) V72277 N-Desmethyl imatinib mesylate (Norimatinib mesylate; Imatinib metabolite N-Desmethyl imatinib mesylate) 404844-03-7 N-Desmethyl imatinib mesylate (Norimatinib mesylate) is a metabolite of Imatinib.
N-Desmethyl rosiglitazone V102724 N-Desmethyl rosiglitazone 257892-31-2 N-desmethylrosiglitazone (SB 237216) is a metabolite of rosiglitazone, produced by the demethylation reaction of the cytochrome P450 enzyme system in liver microsomes, and has a certain PPARγ agonist effect.
N-Desmethyl zopiclone-d8 V72239 N-Desmethyl zopiclone-d8 1189805-43-3 N-Desmethyl zopiclone-d8 is the deuterium labelled form of Norzopiclone.
N-Desmethyl-U-47700 V103003 N-Desmethyl-U-47700 67579-73-1 N-Demethyl-U-47700 is the major metabolite of U-47700 (opioid agonist).
N-Methyl Palbociclib (impurity of palbociclib) V72153 N-Methyl Palbociclib (impurity of palbociclib) 571189-51-0 N-Methyl Palbociclib is an impurity of Palbociclib.
N-Methyl pemetrexed (Pemetrexed Impurity A) V72229 N-Methyl pemetrexed (Pemetrexed Impurity A) 869791-42-4 N-Methyl pemetrexed is an impurity in Pemetrexed.
N-Methyl-4-pyridone-3-carboxamide V72129 N-Methyl-4-pyridone-3-carboxamide 769-49-3 N-Methyl-4-pyridone-3-carboxamide is a metabolite of caffeopyridine.
N-Nitrosoglyphosate sodium (N-Nitroso-N-(phosphonoMethyl)glycine sodium; Glyphosate-N-nitroso sodium) V72226 N-Nitrosoglyphosate sodium (N-Nitroso-N-(phosphonoMethyl)glycine sodium; Glyphosate-N-nitroso sodium) 56516-71-3 N-Nitrosoglyphosate sodium is a degradation product of nitrosamines and a synthetic impurity in glyphosate herbicides.
N-去乙基舒尼替尼 V30776 N-Desethyl Sunitinib (SU-11662) 356068-97-8 N-Desethyl Sunitinib(SU-11662) is a major metabolite of sunitinib which is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Kis of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively.
N-去甲基伊伐布雷定盐酸盐 V33434 Ivabradine metabolite N-Demethyl Ivabradine hydrochloride 1246638-08-3 Ivabradine metabolite N-Demethyl Ivabradine hydrochloride is the N-demethylated metabolite of ivabradine (S-16257; S16257; S 16257;Corlentor; Coralan;Procoralan;Coraxan; Ivabid; Bradia), which is a cardiac pacemaker current (If) inhibitor and a medication approved in 2015 for the management of stable heart-related chest pain and heart failure.
Netupitant N-oxide-d6 V78373 Netupitant N-oxide-d6 Netupitant N-oxide-d6 is the deuterium labelled form of Netupitant N-oxide.
Nicorandil pyridine oxide V107580 Nicorandil pyridine oxide 107833-98-7 Nicorandil oxypyridine is a metabolite of sulfonylurea receptor 2B (SUR2B) that binds to nicorandil, an activator of the ATP-sensitive potassium channel Kir6.2 (SUR2B/Kir6.2) and a nitric oxide donor.
Nirvanol V106578 Nirvanol 631-07-2 Nirvanol (ethylphenylhydantoin), a metabolite of mephenytoin, exerts anticonvulsant effects in the maximal electroshock (MES) epilepsy mouse model.
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