| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V70785 | Substance P(1-7) TFA | 2828433-22-1 | Substance P(1-7) TFA is a fragment of the neuropeptide substance P (SP). |
|
V70796 | Substance P-Gly-Lys-Arg | 123148-51-6 | Substance P-Gly-Lys-Arg, known also as β-Preprotachykinin (58-71), is an analog of Substance P (Substance P). |
|
V116226 | TKA-731 | 210776-01-5 | TKA-731 is an NK1 receptor antagonist. |
|
V116183 | UK-224671 | 178309-91-6 | UK-224671 is a potent, selective NK2 receptor antagonist. |
|
V114363 | Vestipitant mesylate | 334476-64-1 | Vestipitant (GW597599) mesylate is a selective, orally effective NK1 receptor antagonist that can cross the blood-brain barrier. |
|
V99674 | WIN 66306 | 151928-32-4 | WIN 66306 is a cyclic heptapeptide isolated from Aspergillus sp. |
|
V97448 | Y1 receptor antagonist 1 formic | Y1 receptor antagonist 1 formate (H 409-22 isomer formate) is the formate salt form of Y1 receptor antagonist 1. | |
|
V102731 | YM-49598 iodide | 476494-44-7 | YM-49598 iodide is a tachykinin NK-1 receptor antagonist. |
|
V112052 | Zalsenertant tetraxetan | 1613265-38-5 | Zalsenertant tetraxetan (IPN-01087) is a DOTA-coupled neurotensin receptor type 1 (NTSR1) antagonist. |
|
V70805 | γ-Neuropeptide (rabbit) | 114882-65-4 | γ-Neuropeptide (rabbit) can be extracted from rabbit intestine. |
|
V4357 | VAPREOTIDE | 103222-11-3 | Vapreotide (trade name: Sanvar) is a synthetic somatostatin analog and a NK1R antagonist with an IC50 of 330 nM. |
|
V26404 | Netupitant | 290297-26-6 | Netupitant (formerly CID-6451149; AGE-94200; Ro 67-3189)is an orally bioavailable neurokinin 1 (NK1) receptor antagonist with potential antiemetic activity. |
|
V38701 | Eprazinone diHCl | 10402-53-6 | Eprazinone diHCl, the dihydrochloride salt of Eprazinone, is a novel and potent neurokinin 1 receptor (NK1R) ligand with mucolytic, secretolytic, and bronchialantispasmodic activities. |
|
V4399 | FOSAPREPITANT | 172673-20-0 | Fosaprepitant (also known as L-758298; MK0517) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting. |
|
V4400 | FOSAPREPITANT DIMEGLUMINE | 265121-04-8 | Fosaprepitant dimeglumine (also known as L-758298 dimeglumine; MK0517 dimeglumine) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting. |
|
V3303 | Rolapitant | 552292-08-7 | Rolapitant (formerly SCH-619734; SCH619734; tradename: Varubi) is a selective,CNS penetrant and orally bioactiveneurokinin (NK1) receptor antagonist (Ki = 0.66 nM) with antiemetic activity. |
|
V3304 | Rolapitant HCl hydrate | 914462-92-3 | Rolapitant HCl hydrate (SCH619734; SCH-619734; SCH 619734; Varubi), the hydrochloride salt of Rolapitant, is a CNS penetreable and orally bioavailable antagonist of neurokinin (NK1) receptor (Ki = 0.66 nM) that was approved in 2015 to prevent delayed nausea and vomiting caused by cancer chemotherapy. |
|
V4358 | VAPREOTIDE ACETATE | 849479-74-9 | Vapreotide acetate (trade name: Sanvar) is a synthetic somatostatin analog and a NK1R antagonist with an IC50 of 330 nM. |
|
V4330 | APREPITANT | 170729-80-3 | Aprepitant (formerly known as MK-0869; MK-869; L-754030; trade name: Emend) is a novel, selective and high-affinity small molecule antagonist of neurokinin 1 receptor with a Kd of 86 pM. |
|
V15365 | Maropitant (CJ11,972; CJ-11972) | 147116-67-4 | Maropitan (CJ11972; CJ11972) is a novel, potent, selective and orally bioactive antagonist of neurokinin (NK1) receptor. |