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V26404
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Netupitant |
290297-26-6 |
Netupitant (formerly CID-6451149; AGE-94200; Ro 67-3189)is an orally bioavailable neurokinin 1 (NK1) receptor antagonist with potential antiemetic activity. |
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V70787
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Netupitant-d6 (Netupitant D6; CID-6451149-d6) |
2070015-31-3 |
Netupitant-d6 is a deuterium labelled form ofNetupitant (CID-6451149), a highly efficient, selective, orally bioactive Neurokinin-1 receptor (NK1) antagonist. |
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V70784
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Neurokinin A TFA (Substance K TFA; Neurokinin α TFA; Neuromedin L TFA) |
2828433-19-6 |
Neurokinin A TFA (Substance K TFA) is a bioactive peptide neurotransmitter of the tachykinin family that acts through the NK-2 receptor. |
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V76709
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Neurokinin A(4-10) TFA |
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Neurokinin A (4-10) TFA is a tachykinin NK2 receptor agonist (activator). |
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V70804
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Neurokinin Receptor (393-407), rat (SPR393-407) |
153607-26-2 |
Neurokinin Receptor (393-407), rat (SPR393–407) is a fragment of the rat neurokinin 1 receptor (NK1R). |
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V70799
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NK1 receptor antagonist 2 |
579475-17-5 |
NK1 receptor antagonist 2 is an NK1 receptor antagonist. |
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V70792
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NK3R-IN-1 |
2854331-14-7 |
NK3R-IN-1 (compound 16x) is an imidazopiperazine analogue and an orally bioactive Neurokinin Receptor NK3R inhibitor. |
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V4278
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Pavinetant |
941690-55-7 |
AZD2624 (also known as AZD-4901, MLE-4901, AZ-12472520, and AZD-2624) is a novel, potent, selective and orally bioactive neurokinin-3 receptor (NK3R) antagonist. |
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V70812
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Phyllomedusin |
26145-48-2 |
Phyllomedusin, a tachykinin decapeptide, is an NK1 receptor agonist (activator). |
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V70808
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QWF Peptide |
126088-82-2 |
QWF Peptide (Compound 4a) is a substance P antagonist (inhibitor) with IC50 of 0.09 μM. |
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V3303
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Rolapitant |
552292-08-7 |
Rolapitant (formerly SCH-619734; SCH619734; tradename: Varubi) is a selective,CNS penetrant and orally bioactiveneurokinin (NK1) receptor antagonist (Ki = 0.66 nM) with antiemetic activity. |
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V3304
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Rolapitant HCl |
914462-92-3 |
Rolapitant HCl (SCH619734; SCH-619734; SCH 619734; Varubi), the hydrochloride salt of Rolapitant, is a CNS penetreable and orally bioavailable antagonist of neurokinin (NK1) receptor (Ki = 0.66 nM) that was approved in 2015 to prevent delayed nausea and vomiting caused by cancer chemotherapy. |
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V4618
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SB 222200 |
174635-69-9 |
SB-222200 is a novel, potent, selective, reversible, brain penetrant and competitive antagonist of human NK-3 receptor with Ki of 4.4 nM. |
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V76487
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Spantide I TFA |
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Spantide I TFA is an analogue of substance P and a selective neurokinin-1 receptor (NK1 receptor) antagonist. |
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V76473
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Substance P (5-11) (TFA) |
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Substance P (5-11) TFA TFA is the C-terminal heptapeptide of Substance P (Substance P), a neuropeptide that binds to the NK-1 tachykinin receptor. |
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V70794
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Substance P (6-11) |
51165-07-2 |
Substance P (6-11) is the C-terminal hexapeptide amide of Substance P (Substance P). |
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V70785
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Substance P(1-7) TFA |
2828433-22-1 |
Substance P(1-7) TFA is a fragment of the neuropeptide substance P (SP). |
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V70796
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Substance P-Gly-Lys-Arg |
123148-51-6 |
Substance P-Gly-Lys-Arg, known also as β-Preprotachykinin (58-71), is an analog of Substance P (Substance P). |
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V4357
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VAPREOTIDE |
103222-11-3 |
Vapreotide (trade name: Sanvar) is a synthetic somatostatin analog and a NK1R antagonist with an IC50 of 330 nM. |
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V4358
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VAPREOTIDE ACETATE |
849479-74-9 |
Vapreotide acetate (trade name: Sanvar) is a synthetic somatostatin analog and a NK1R antagonist with an IC50 of 330 nM. |