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V78447
|
Biotin-NeurokininA |
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Biotin-NeurokininA is a biotinylated NeurokininA. |
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V70790
|
Ditryptophenaline ((-)-Ditryptophenaline) |
64947-43-9 |
Ditryptophenaline ((-)-Ditryptophenaline) is a metabolite of Aspergillus flavus. |
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V70788
|
Eledoisin (Eledone peptide) |
69-25-0 |
Eledoisin (Eledone peptide) is a specific agonist of NK2 and NK3 receptors. |
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V38701
|
Eprazinone diHCl |
10402-53-6 |
Eprazinone diHCl, the dihydrochloride salt of Eprazinone, is a novel and potent neurokinin 1 receptor (NK1R) ligand with mucolytic, secretolytic, and bronchialantispasmodic activities. |
|
V4399
|
FOSAPREPITANT |
172673-20-0 |
Fosaprepitant (also known as L-758298; MK0517) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting. |
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V4400
|
FOSAPREPITANT DIMEGLUMINE |
265121-04-8 |
Fosaprepitant dimeglumine (also known as L-758298 dimeglumine; MK0517 dimeglumine) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting. |
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V70783
|
Fosnetupitant chloride monohydrochloride (Pronetupitant chloride monohydrochloride) |
1643757-72-5 |
Fosnetupitant chloride mono HCl (Pronetupitant chloride mono HCl) is an NK1 antagonist (inhibitor) with pKis of 9.5 and 6.1 for human NK1 and NK3 receptors, respectively. |
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V70801
|
Gly-Leu-Met-NH2 |
4652-64-6 |
Gly-Leu-Met-NH2 is the C-terminal tripeptide of Substance P (Substance P). |
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V70786
|
GR 64349 |
137593-52-3 |
GR 64349 is a potent and selective peptide antagonist of the neurokinin 2 (NK2) receptor with EC50 of 3.7 nM measured in rat colon. |
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V79644
|
GR 64349 TFA |
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GR 64349 is a potent and selective peptide antagonist of the neurokinin 2 (NK2) receptor with EC50 of 3.7 nM measured in rat colon. |
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V70806
|
GR 83074 |
141636-44-4 |
GR 83074 is a potent and specific NK-2 (Neurokinin Receptor) antagonist (inhibitor) with a pKB of 8.23. |
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V70793
|
GR 87389 |
141663-86-7 |
GR 87389 is a potent NK2 receptor antagonist. |
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V79645
|
GR 94800 TFA |
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GR 94800 TFA is a potent and specific peptide antagonist of neurokinin 2 (NK2) receptors with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors respectively. |
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V79751
|
Hemokinin 1, human TFA |
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Hemokinin 1, human TFA is a selective full agonist of the tachykinin neurokinin 1 (NK1) receptor. |
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V70814
|
Imnopitant |
290297-57-3 |
Imnopitant is an NK1 receptor blocker (antagonist) (WO2020132716, compound 1). |
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V15365
|
Maropitant (CJ11,972; CJ-11972) |
147116-67-4 |
Maropitan (CJ11972; CJ11972) is a novel, potent, selective and orally bioactive antagonist of neurokinin (NK1) receptor. |
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V70810
|
MDL 29913 |
135721-56-1 |
MDL 29913 cyclic peptide is a competitive NK2 tachykinin receptor selective antagonist (inhibitor) with a pA2 value of 8.66. |
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V76775
|
Men 10376 TFA (Neurokinin-2 receptor antagonist TFA) |
|
Men 10376 TFA is a potent and specific tachykinin NK-2 receptor antagonist (inhibitor) with a Ki of 4.4 μM for rat intestinal NK-2 receptors. |
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V70817
|
MLGFFQQPKPR-NH2 |
1802883-75-5 |
MLGFFQQPKPR-NH2 is a Substance P reverse sequence peptide. |
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V78372
|
Monohydroxy Netupitant-d6 |
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Monohydroxy Netupitant-d6 is the deuterium labelled form of Monohydroxy Netupitant. |