|
V5069
|
Metaxalone (AHR438;NSC170959) |
1665-48-1 |
Metaxalone(also known as AHR438; NSC170959) is a skeletal muscle relaxant prescribed for the short-term treatment of painful muscle spasmscaused by strains, sprains, and other musculoskeletal conditions. |
|
V5088
|
Methoxyamine HCl |
593-56-6 |
Methoxyamine HCl is a novel, potent and orally bioavailable small molecule inhibitor with potential adjuvant activity. |
|
V5137
|
Miconazole Nitrate |
228321-87-7 |
Miconazole Nitrate is a potent imidazole-based antifungal agent that is commonly used by topical administration to the skin or to mucous membranes to cure fungal infections. |
|
V5016
|
NSC-41589 |
6310-41-4 |
NSC-41589 is N-[2-(methylsulfanyl) phenyl]acetamide. |
|
V5041
|
NSC139021 (ERGi-USU) |
1147-56-4 |
NSC139021 (also known as ERGi-USU) is a novel, potent and highly selective inhibitor for the growth of ERG-positive cancer cells with IC50s ranging from 30 to 400 nM. |
|
V4875
|
Onalespib lactate |
1019889-35-0 |
Onalespib (formerly also known as AT13387; AT-13387) is an orally bioavailable small-molecule Hsp90 inhibitor (IC50 = 18 nM in A375 cells) with long-lasting anti-tumor activity. |
|
V4780
|
PCI-27483 |
871266-63-6 |
PCI-27483 is a novel, potent and reversible small-molecule inhibitor of activated factor VII (factor VIIa) with potential anticancer and antithrombotic activities. |
|
V2174
|
RETV804M inhibitor |
2414373-42-3 |
RET-IN-21 is a receptor tyrosine kinase (RET) inhibitor (antagonist) with IC50 of 4.4 μM and anti-tumor activity. |
|
V4811
|
Ro 10-5824 |
189744-46-5 |
Ro 10-5824 is a novel, potent and selectivepartial agonist of dopamine D4 receptorwithKiof 5.2 nM. |
|
V4611
|
SB-224289 HCL |
180083-23-2 |
SB-224289 hydrochloride is a novel, potent and selective5-HT1B receptorantagonist with anxiolytic effect with pKi of 8.2. |
|
V2164
|
SC-26196 |
218136-59-5 |
SC-26196 is a novel, potent and orally bioactive D6D (Delta6 desaturase) inhibitor with IC50 of 0.2 µM in a rat liver microsomal assay. |
|
V4670
|
SCH00013 |
217963-18-3 |
SCH00013 is a novel and potent Ca2+ sensitizer that elicits a moderate positive inotropic effect without significant alteration of Ca2+ transients. |
|
V4800
|
SJA710-6 |
1397255-09-2 |
SJA710-6 (a Hepatic Differentiation Inducer) is a novel, potent and cell-permeable small moleculeimidazopyridinamine compound that is able to induce the differentiation of rat MSCs (rMSCs) toward hepatocyte-like cells(~47% at 5 µM). |
|
V5053
|
SKI-II HCl |
1177741-83-1 |
SKI-II HCl is a substrate competitive, reversible, and highly specific inhibitor of sphingosine kinase. |
|
V4597
|
Sufugolix (TAK013) |
308831-61-0 |
Sufugolix (formerly known as TAK-013) is a novel, highly potent,non-peptide, selective and orally bioavailable luteinizing hormone-releasing hormone (LHRH) receptor antagonist with anticancer activity. |
|
V4906
|
Talampanel |
161832-65-1 |
Talampanel (also known as LY300164; LY-300164 and GYKI-53773) is a novel, potent, orally bioavailable and selective α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate (AMPA) receptor antagonis with anti-seizure activity. |
|
V5197
|
Teixobactin |
1613225-53-8 |
Teixobactin, a naturally occuring antibiotic discovered in a screen of uncultured bacteria, is a novel peptide-like secondary metabolite of some species of bacteria, that kills some gram-positive bacteria, and has the the potential to overcome drug resistance. |
|
V5058
|
TP-2857 |
1575491-01-8 |
TP-2857 is novel and potent antimicrobial compound. |
|
V4594
|
U83836E |
137018-55-4 |
U83836E is a novel and potent lipid peroxidation (LP) inhibitor. |
|
V4622
|
Zotiraciclib (SB1317) HCl |
1354567-82-0 |
Zotiraciclib (SB1317; TG02) HCl, the hydrochloride salt of SB1317, is a novel and potent small molecule inhibitor ofCDK2,JAK2, andFLT3 with the potential for the treatment of cancer. |