The ion channel known as the calcium channel exhibits selective permeability to calcium ions. Although there are ligand-gated calcium channels as well, it is sometimes referred to as a voltage-dependent calcium channel. Even though the concentration of Na+ outside of cells is 70 times higher than that of Ca2+, voltage-gated calcium (CaV) channels catalyze a rapid, highly selective influx of Ca2+ into cells. A side effect of some calcium channel blockers is that they slow your heart rate, which helps to lower blood pressure, treat angina, and regulate irregular heartbeats.
Structure | Cat No. | Product Name | CAS No. | Product Description |
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V71513 | Menthol-d4 | 1217765-02-0 | Menthol-d4 is the deuterium labelled form of Menthol. |
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V71538 | MMK1 | 271246-66-3 | MMK1 is a potent and specific human formyl peptide receptor-like 1 (FPRL-1/FPR2) agonist/activator with EC50s of <2 nM and >10000 nM for FPRL-1 and FPR1, respectively. |
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V80794 | MMK1 TFA | MMK1 TFA is a potent and specific human formyl peptide receptor-like 1 (FPRL-1/FPR2) agonist/activator with EC50s of <2 nM and >10000 nM for FPRL-1 and FPR1, respectively. | |
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V80860 | Myoregulin (MLN peptide) | Myoregulin (MLN peptide) is a member of the regulin family. | |
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V80861 | Myoregulin TFA (MLN peptide TFA) | Myoregulin (MLN peptide) TFA is a member of the regulin family. | |
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V80865 | Myr-TAT-CBD3 | Myr-TAT-CBD3 is a CRMP2-CaV2.2 interaction inhibitor. | |
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V71516 | N-Desalkylflurazepam (Norfludiazepam) | 2886-65-9 | N-Desalkylflurazepam (Norfludiazepam) is a long-acting metabolite of benzodiazepines such as Flurazepam. |
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V71536 | Ned-K | 2250019-90-8 | Ned-K is a niacin adenine dinucleotide phosphate (NAADP) antagonist. |
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V101127 | Nemadipine B | 79925-38-5 | Nemadipine B is a calcium channel blocker and EGL-19 antagonist. |
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V71508 | Nemadipine-A | 54280-71-6 | Nemadipine-A is a specific inhibitor of the EGL-19 Ca2+ channel. |
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V102930 | Niguldipine monohydrochloride | 119934-51-9 | Niguldipine monohydrochloride is a calcium channel blocker with inhibitory effects on P-glycoprotein and can be used in tumor research. |
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V71505 | Norverapamil-d7 hydrochloride ((±)-Norverapamil-d7 (hydrochloride); D591-d7 (hydrochloride)) | 1216413-74-9 | Norverapamil-d7 ( HCl) is a deuterium labelled form of Norverapamil. |
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V107902 | O-Desmethylcarvedilol | 72956-44-6 | O-Desmethylcarvedilol (desmethylcarvedilol) is the active metabolite of carvedilol and a non-selective β-adrenergic receptor (β-AR) antagonist. |
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V102288 | Oxodipine | 90729-41-2 | Osodipine, a dihydropyridine calcium channel blocker, inhibits KCl-induced constriction of the rabbit aorta and reduces cardiac force during weak ventricular contraction in rats. |
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V76662 | PACAP-38 (31-38), human, mouse, rat TFA | PACAP-38 (31-38), human, mouse, rat TFA is a PAC1 receptor agonist/activator. | |
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V81035 | Palmitoylglycine-d31 (N-palmitoylglycine-d31) | Palmitoylglycine-d31 is the deuterated form of Palmitoylglycine. | |
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V94236 | Palonidipine hydrochloride | 96515-74-1 | Palonidipine hydrochloride is a calcium antagonist used to treat angina pectoris and hypertension. |
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V96880 | PD-0299685 | 313651-33-1 | PD-0299685 is a potent Ca2+ channel α2δ ligand. |
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V102955 | PDDHV | 179469-40-0 | PDDHV is a calcium uptake inducer that can induce 45Ca2+ influx by stimulating the vanilloid receptor VR1. |
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V80048 | PptT-IN-4 | 2948309-57-5 | PptT-IN-4 (Compound 3a) is a PptT inhibitor (IC50= 0.71 μM). |