Progesterone receptor (PR) is a member of the steroid/thyroid hormone-retinoid receptor superfamily of ligand-activated nuclear transcription factors.
The development, differentiation, and maintenance of female reproductive tissue depends heavily on progesterone receptor.The ability of the progesterone receptor to bind to a wide range of ligands results in a wide range of transcriptional responses, including full agonism, full antagonism, and several mixed profiles in between. Progesterone receptors, such as progesterone, cause the PR ligand binding domain (LBD) to change its conformation, which in turn controls subsequent gene regulatory cascades.
Human PR-A and PR-B are two different types of progesterone receptors that mediate the biological response to progesterone in humans.
| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V114533 | Anordrin | 56470-64-5 | Anordlin is a type of birth control pill. |
|
V115691 | EC 313 | 1249398-29-5 | EC 313 is a selective progesterone receptor modulator. |
|
V118660 | EIDD-036 | 211302-60-2 | EIDD-036 is a C-20 oxime progesterone derivative that can cross the blood-brain barrier and bind to the progesterone receptor (PR), with an IC50 value of 171 nM. |
|
V109480 | Hydroxyprogesterone caproate-d8 | Hydroxyprogesterone hexanoate-d8 (17α-hydroxyprogesterone hexanoate-d8) is a deuterated derivative of hydroxyprogesterone hexanoate. | |
|
V109488 | Medroxyprogesterone acetate-d7 | Medroxyprogesterone acetate-d7 is a deuterated derivative of medroxyprogesterone acetate. | |
|
V109715 | Melengesterol | 5633-18-1 | Merenprogesterone is a steroidal progestin belonging to the 17α-hydroxyprogesterone class and is an anti-tumor drug. |
|
V111341 | Brofoxine | 21440-97-1 | Brofoxine is a progesterone receptor modulator with anxiolytic effects. |
|
V83993 | 17α-Ethynyl-19-nor-Δ-5(6)-androsten-17β-ol-3-one (delta-5(6)-Norethindrone) | 22933-71-7 | |
|
V67772 | 17α-Hydroxyprogesterone-13C3 (17-Hydroxyprogesterone-13C3; 17-OHP-13C3) | 1356154-92-1 | 17α-Hydroxyprogesterone-13C3 is a 13C (carbon 13)-labeled 17α-Hydroxyprogesterone. |
|
V67766 | 17α-Hydroxyprogesterone-d8 (17-Hydroxyprogesterone-d8; 17-OHP-d8) | 850023-80-2 | 17α-Hydroxyprogesterone-d8 is the deuterium labelled form of 17α-Hydroxyprogesterone. |
|
V77901 | Altrenogest-d5 (Allyltrenbolone-d5; Allyltrenbolone-d5; RU2267-d5) | Altrenogest-d5 is the deuterium labelled form of Altrenogest. | |
|
V67604 | ARD-61 | 2316837-08-6 | ARD-61 is a highly efficient and specific PROTAC androgen receptor (AR) degrader. |
|
V110533 | CPAG-1 | 2094991-62-3 | CPAG-1 is a small molecule progesterone receptor membrane component 2 (PGRMC2) activator. |
|
V67773 | Drospirenone-d4 | 2376035-94-6 | Drospirenone-d4 is the deuterium labelled form of Drospirenone. |
|
V79659 | Dydrogesterone-d6 (dydrogesterone d6) | Dydrogesterone-d6 is the deuterated form of Dydrogesterone. | |
|
V65080 | Gestodene-d6 (SHB 331-d6; WL 70-d6) | 1542211-40-4 | Gestodene-d6 is the deuterated form of Gestodene. |
|
V67771 | Medroxyprogesterone-d3 (17α-Hydroxy-6α-methylprogesterone-d3; U8840-d3) | 162462-69-3 | Medroxyprogesterone-d3 is the deuterium labelled form of Medroxyprogesterone. |
|
V67765 | Melengestrol acetate | 2919-66-6 | Melengestrol acetate is a progesterone analogue that works as an orally bioactive corticosteroid that promotes endometrial proliferation, maintenance of pregnancy, and delayed menstrual activity. |
|
V78844 | Melengestrol acetate-d2 | Melengestrol acetate-d2 is the deuterium labelled form of Melengestrol acetate. | |
|
V76777 | Melengestrol acetate-d3 | Melengestrol acetate-d3 is the deuterium labelled form of Melengestrol acetate. |
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