| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V50422 | (E/Z)-Zotiraciclib citrate-TG-02 citrate; SB-1317 citrate | 1204918-73-9 | (E/Z)-Zotiraciclib citrate (TG02 citrate; SB1317 citrate is a novel and potent CDK2, JAK2, and FLT3 inhibitorwith the potential for the treatment of cancer. |
|
V41444 | (Rac)-Vepdegestrant | 2229711-08-2 | (Rac)-Vepdegestrant (ARV-471 racemate; ARV471) is a first-in-class, selective and orally bioavailable PROTAC-based Estrogen Receptor (AR) degrader. |
|
V41400 | Bay-3827 | 2377576-35-5 | BAY-3827 is a potent and specific AMPK inhibitor (antagonist) with IC50s of 1.4 nM (10 µM ATP) and 15 nM (2 mM ATP). |
|
V41447 | BIIB068 | 1798787-27-5 | BIIB068 (BIIB-068) is a novelreversible and orally bioavailable BTK inhibitor with the potential to be used for autoimmune diseases such as systemic lupus erythematosus (SLE). |
|
V37648 | BMVC-8C3O | 1301708-12-2 | BMVC-8C3O is a novel ligand of DNA G-quadruplexe (G4) that can induce topological conversion of non-parallel to parallel forms in human telomeric DNA G4s. |
|
V41389 | C-021 (CCR4 antagonist) | 864289-85-0 | C021 (C-021; CCR4 antagonist) is a novel and potent CCR4 antagonist with anti-inflammatory activity. |
|
V42163 | CCR6 antagonist 1 | 588674-64-0 | CCR6 antagonist 1 is a CCR6 antagonist with the potential tobe used in autoimmune diseases, e. |
|
V41588 | Compound 6q | Compound 6q is a novel and potent steroidal anti-inflammatory agent that has the potential to be used in the treatment of IBD (inflammatory bowel diseases). | |
|
V49209 | DDO-7263 | 2254004-96-9 | DDO-7263 is a 1,2,4-Oxadiazole analogue and a potent Nrf2-ARE activator. |
|
V41419 | gamma-Glu-Cys | 636-58-8 | Gamma-glutamylcysteine (amma-Glu-Cys) is a substrate for biosynthesis of L-glutathione by glutathione synthetase. |
|
V50576 | GRK6-IN-1 | 2677786-61-5 | GRK6-IN-1 (compound 18) is a potent inhibitor of G protein-coupled receptor kinase 6 (GRK6) with IC50 of 120 nM. |
|
V37640 | GS-441524 HCl | 2378280-82-9 | GS-441524 is an active metabolite of Remdesivir (GS-5734;Veklury) which is an FDA approved drug for treating the2019-nCoV (COVID-19 pandemic, CoronaVirus)infections. |
|
V44412 | MLN-3126 | 628300-71-0 | MLN3126 is an orally bioactive and potent CCR9 antagonist. |
|
V47181 | Mtb ATP synthase-IN-1 | 2642394-38-3 | Mtb ATP synthase-IN-1 (compound 6ab) is a potent inhibitor of Mycobacterium tuberculosis (TB) (Mtb) ATP synthesis, with MIC of Mtb of 0.452 ~ 0.499 μg/mL. |
|
V41464 | MYLS22 | 306959-01-3 | MYLS22 is a selective inhibitor of optic atrophy 1 (OPA1). |
|
V37656 | NS-3-008 HCl | 1172854-54-4 | NS-3-008 is a novel and orally bioactive transcriptional inhibitor of G0/G1 switch 2 (G0s2). |
|
V47326 | P2Y2R/GPR17 antagonist 1 | 2395016-49-4 | P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R and GPR17 antagonist (inhibitor) with IC50s of 3.17 µM and 1.67 µM for P2Y2R and GPR17, respectively. |
|
V44337 | SHMT-IN-2 | 2102681-49-0 | SHMT-IN-2 is an inhibitor of human SHMT1/2 which is aserine hydroxymethyltransferase (SHMT). |
|
V42907 | SRI-37240 | 883956-47-6 | SRI-37240 is a potent inhibitor of premature termination codons (PTCs). |
|
V37651 | VLX600 HCl | 1622945-04-3 | VLX600 is a novel Iron Chelator Targeting Both Proliferating and Quiescent Cancer Cells. |