GPR

GPR

GPR related products

Structure Cat No. Product Name CAS No. Product Description
V70306 PSN 375963 hydrochloride 1781834-82-9 PSN 375963 HCl is a potent GPR119 agonist/activator with EC50 of 8.4 and 7.9 μM in humans and mice, respectively.
V76546 RTI-13951-33 hydrochloride RTI-13951-33 HCl is a specific, BBB (blood-brain barrier) permeable (penetrable) GPR88 agonist/activator with EC50 of 25 nM in GPR88 cAMP functional assays.
V15926 TC-H 106 937039-45-7 Pimelic Diphenylamide 106 is a slow, tight-binding class I HDAC inhibitor (inhibits HDAC1, 2, and 3, IC50s 150 nM, 760 nM, and 370 nM, respectively) with no activity against class II HDACs.
V1807 Timapiprant (OC000459) 851723-84-7 Timapiprant (formerly known as OC000459; OC-000459) is a novel, potent, selective, and orally bioactive prostanoid receptor 2 (DP2- also known as CRTH2)) antagonist with IC50 of 13 nM.
V70308 Zelatriazin (TAK-041; NBI-1065846) 1929519-13-0 Zelatriazin (TAK-041; NBI-1065846) is a potent and specific GPR139 agonist/activator with EC50 of 22 nM.
V75419 ZQ-16 376616-73-8 ZQ-16 is a potent and specific GPR84 agonist/activator with EC50 of 0.213 μM.
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