| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V1168 | 5-hydroxymethyl tolterodine (PNU 200577) | 207679-81-0 | 5-hydroxymethyl tolterodine (Desfesoterodine, PNU 200577,PNU-200577, 5HMT, 5HM;5-HMT, 5-HM), the active metabolite of tolterodine which is a medicationused treat overactive bladder, is a novel and potent muscarinic receptor antagonist with a Kb of 0.84 nM. |
|
V1165 | LY2119620 | 886047-22-9 | LY2119620 (LY 2119620; LY-2119620) is a novel, potent, specific, high-affinity and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors, the so called positive allosteric modulator (PAM). |
|
V1191 | PNU-120596 (NSC-216666) | 501925-31-1 | PNU-120596 (PNU120596;NSC 216666;PNU 120596;NSC-216666)is a potent and selective PAM (positive allosteric modulator) of α7 nAChR (acetylcholine receptor) with an EC50 of 216 NM. |
|
V17279 | Butylscopolamine bromide | 149-64-4 | Butylscopolamine bromide is a potent antimuscarinic quaternary ammonium analogue acting as a competitive antagonist of mAChR (IC50: 55.3 ± 4.3 nM). |
|
V1185 | Gallamine Triethiodide | 65-29-2 | Gallamine Triethiodide (Flaxedil; Tricuran; Gallamoni jodidum; Gallaminii iodidum),a non-depolarising muscle relaxant, is a potent and cardioselective cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM. |
|
V1196 | Homatropine Bromide (Homatropine hydrobromide) | 51-56-9 | Homatropine Bromide (Equipin, Isopto Homatropine), the hydrobromide salt of Homatropine, is a potent muscarinic AChR (acetylcholine receptor) antagonist used before eye examinations (i.e. refraction), before and after certain eye surgeries, and for treating certain eye conditions (e.g., uveitis). |
|
V1172 | Pyridostigmine Bromide | 101-26-8 | Pyridostigmine Bromide (Mestinon; Regonol; Kalimin) is a parasympathomimetic and a reversible cholinesterase inhibitor used in the treatment of myasthenia gravis and to reverse the actions of muscle relaxants. |
|
V1160 | Tiotropium Bromide hydrate (BA-679 BR) | 139404-48-1 | Tiotropium Bromide hydrate (PUR-0200; BA-679BR; BA679BR;PUR0200; Spiriva), the monohydrate form of tiotropium bromide, is an anticholinergic and bronchodilator and a muscarinic receptor antagonist used as a long-acting bronchodilator for the management of chronic obstructive pulmonary disease (COPD). |
|
V1186 | Oxybutynin | 5633-20-5 | Oxybutynin (Ditropan, Lyrinel XL, Lenditro,Oxybutynin, Uripan) is a potent and competitive antagonist of the M1, M2, and M3 subtypes of the muscarinic acetylcholine receptor, used to relieve urinary and bladder difficulties. |
|
V25120 | Isoimperatorin | 482-45-1 | Isoimperatorin is a COX-2 inhibitor. |
|
V1181 | Tropicamide | 1508-75-4 | Tropicamide (formerlyRo-17683;Ro 1-7683; trade names Mydral; Mydriafair; Mydriaticum; Mydrum),an approved medication used to dilate the pupil and help with eye examination,is a potent anticholinergic and a muscarinic receptor isoform M4 antagonistwith important biological activity. |
|
V1190 | Orphenadrine Citrate | 4682-36-4 | Orphenadrine Citrate (BS-5930;BS5930; BS 5930; Disipal), the citrate salt ofOrphenadrine,is anuncompetitiveNMDA receptor antagonist and apotent skeletal muscle relaxant with antispastic and analgesic activities. |
|
V1171 | Darifenacin HBr (UK88525) | 133099-07-7 | Darifenacin HBr (formerly known as UK-88525;Emselex; Enablex),the hydrobromide salt ofDarifenacin, is a approved medication used to treat urinary incontinence and overactive bladder. |
|
V1162 | Pancuronium dibromide | 15500-66-0 | Pancuronium dibromide (OrgNA97; NA-97; Org NA 97; Pavulon),a neuromuscular relaxant used in euthanasia, is a bis-quaternary steroid and a competitive nicotinic acetylcholine receptor antagonist with an IC50 of5.5 nM. |
|
V1176 | Rocuronium Bromide (ORG 9426 Bromide) | 119302-91-9 | Rocuronium Bromide (ORG-9426; Zemuron; Esmeron; Esmeron; Esmerone) is a potent and competitive Nicotinic acetyl-choline receptors (AchR) antagonist, which is a non-depolarizing neuromuscular blocking agent used in anaesthesia required for surgery or mechanical ventilation. |
|
V1200 | L-Hyoscyamine (Daturine) | 101-31-5 | L-Hyoscyamine (Daturine), a natural tropane alkaloid and plant toxin, is the the levo-isomer of atropine and is used for controlling symptoms associated with disorders of the gastrointestinal (GI) tract. |
|
V1203 | Varenicline Tartrate (CP 526555-18) | 375815-87-5 | Varenicline Tartrate (CP-526555 18; CP 526555 18;Chantix; Champix), the tartrate salt of varenicline, is a potent partial agonist of nicotinic AChR (acetylcholine receptor) used for smoke-cessation and nicotine addiction. |
|
V1194 | Aclidinium Bromide (LAS 34273; LAS-W 330) | 320345-99-1 | Aclidinium Bromide (formerly LAS34273, LAS-W 330; brand names Tudorza Genuair;Eklira Genuair; Bretaris Genuair) is a potent, long-acting and inhalable muscarinic antagonist used as a maintenance treatment for chronic obstructive pulmonary disease (COPD). |
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