| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V2985 | BD 1047 dihydrobromide | 138356-21-5 | BD1047 dihydrobromide (BD-1047) is a selective functional antagonist of sigma receptors (σ receptors) with antipsychotic activity and may be used for schizophrenia. |
|
V108977 | CM304 free base | 1350296-21-7 | CM304 free base (FTC-146) is a potent S1R antagonist. |
|
V70032 | Rimcazole dihydrochloride (BW 234U dihydrochloride) | 75859-03-9 | Rimcazole (BW 234U) di-HCl is a carbazole analogue that acts partially as a sigma receptor antagonist. |
|
V144465 | S1R agonist 3 | 401501-66-4 | S1R agonist 3 is a highly potent, selective, and blood-brain barrier-penetrating σ-1 receptor (S1R) agonist with a Ki value of 1.5 nM. |
|
V144893 | Sigma-2 Receptor ligand 1 | Sigma-2 Receptor ligand 1 is a highly selective Sigma-2 receptor ligand with a Ki value of 40 nM. | |
|
V93033 | UMB24 | 1033-69-8 | UMB24 is a potent σ2 receptor antagonist with Ki values of 170 nM and 322 nM for σ2 and σ1 receptors, respectively. |
|
V147783 | σ1R-IN-1 | σ1R-IN-1 is a potent σ-1R inhibitor with an IC50 of 110 nM. | |
|
V0097 | Cutamesine (SA 4503; AGY 94806) | 165377-43-5 | Cutamesine (SA-4503; AGY-94806) is a selective and potent sigma-1 (σ1) receptor agonist with an IC50of 17.4 nM in guinea pig brain membranes, 100-fold less selective for the sigma 2 receptor. |
|
V2813 | Cutamesine (SA-4503) dihydrochloride | 165377-44-6 | SA4503 dihydrochloride (also known asAGY94806 dihydrochloride andCutamesine dihydrochloride), is a potent sigma-1 (σ1) receptor agonist with an IC50of 17.4 nM in guinea pig brain membranes. |
|
V3703 | Siramesine | 147817-50-3 | Siramesine (Formerly known as Lu-28-179) is a potent and selective agonist of sigma-2 receptor. |
|
V2908 | Siramesine HCl | 224177-60-0 | Formerly known as Lu-28-179, siramesine HCl is a potent and selective sigma-2 receptor agonist with anticancer effects. |