| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V67685 | (Rac)-Zearalanone-d6 | 1795020-90-4 | (Rac)-Zearalanone-d6 is the racemic deuterated form of Zearalenone. |
|
V118717 | 14-3-3σ/ERα stabilizer-2 | 14-3-3σ/ERα stabilizer-2 (compound 41) is a covalent 14-3-3σ/ERα stabilizer with a Kd value of 10.1 nM. | |
|
V106522 | 2-Ethylhexyl diphenyl phosphate | 1241-94-7 | 2-Ethylhexyl diphenyl phosphate is an organophosphorus flame retardant (OPFRs) and a PPARG agonist (EC20: 2.04 µM). |
|
V67691 | 3'-Hydroxymirificin | 168035-02-7 | 3'-Hydroxymirificin (compound 3) is a naturally occurring compound obtained from the roots of Pueraria lobata. |
|
V109447 | 3-Chlorobisphenol A | 74192-35-1 | 3-Chlorobisphenol A is a chlorinated derivative of bisphenol A and is an endocrine disruptor. |
|
V126521 | 4-sec-Butylphenol | 99-71-8 | 4-sec-Butylphenol is an androgen receptor ligand with a pIC50 value of 4.07 for the androgen receptor. |
|
V126525 | 4-tert-Octylphenol monoethoxylate | 2315-67-5 | 4-tert-Octylphenol monoethoxylate is an alkylphenol ethoxylate (APE) and a degradation product of nonionic surfactants such as 4-tert-octylphenol polyethoxylate. |
|
V93836 | ADX61623 | 1067189-44-9 | ADX61623 is a potent negative allosteric modulator (NAM) of the follicle-stimulating hormone receptor (FSHR). |
|
V110360 | ADX68692 | 1067191-08-5 | ADX68692 is an orally effective follicle-stimulating hormone (FSH) receptor negative allosteric modulator with a log IC50 value of -5.71. |
|
V128969 | Anticancer agent 276 | Anticancer agent 276 is a multi-target anticancer drug. | |
|
V101569 | Antiproliferative agent-51 | Antiproliferative agent-51 (Compound 18h) inhibits estrogen receptor α (ERα)-mediated transcription with IC50 of 1.6 nM. | |
|
V2554 | AZD9496 | 1639042-08-2 | AZD9496 is a novel, potent, orally bioavailable, and selective estrogen receptor (ERα) downregulator and antagonist with an IC50 of 0.28 nM and a Ki of 0.7 nM. |
|
V67699 | Bazedoxifene-d4 acetate (TSE-424-d4 acetate) | 1795027-71-2 | Bazedoxifene-d4 (acetate) is the deuterated form of Bazedoxifene. |
|
V130809 | BY13 | BY13 is an SRC-3 PROTAC degrader with a half-maximal lethal concentration (DC50) of 0.031 μM. | |
|
V2996 | DY131 (GSK-9089) | 95167-41-2 | DY131 (also known as GSK-9089) is a novel selective agonist at estrogen-related receptors ERRβ and ERRγ with minimal activity at ERRα, ERα and ERβ at concentrations up to 30 μM. |
|
V114277 | ER degrader 12 | 2376991-14-7 | ER degrader 12 (Example 1) is an estrogen receptor (ER) degrader with IC50 values of 2.3 nM and 80.2 nM for ERα and ERβ, respectively (TR-FRET assay). |
|
V114262 | ER degrader 13 | 2839847-93-5 | ER degrader 13 (compound 37) is an estrogen receptor (ER) degrader. |
|
V67679 | ER degrader 5 | 2913192-47-7 | ER degrader 5 is a potent estrogen receptor (ER) degrader. |
|
V135196 | ER ligand-10 | 1075742-56-1 | ER ligand-10 is a weak ligand for ERα and ERβ and exhibits weak estrogenic activity. |
|
V119066 | ER ligand-12 | ER ligand-12 is an estrogen receptor (ER) ligand that can be used to synthesize PROTACs, such as PROTAC ER degrader-2. |