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mAChR

mAChR

mAChR related products

Structure Cat No. Product Name CAS No. Product Description
(-)-Vesamicol (AH5183) V85954 (-)-Vesamicol (AH5183) 112709-59-8
(Rac)-5-Hydroxymethyl Tolterodine-d14 ((Rac)-Desfesoterodine-d14; (Rac)-PNU-200577-d14) V70549 (Rac)-5-Hydroxymethyl Tolterodine-d14 ((Rac)-Desfesoterodine-d14; (Rac)-PNU-200577-d14) 1185071-13-9 (Rac)-5-Hydroxymethyl Tolterodine-d14 is the deuterated form of (Rac)-5-Hydroxymethyl Tolterodine.
Arecaidine-propargyl ester tosylate V84784 Arecaidine-propargyl ester tosylate 147202-94-6
Atropine methyl nitrate V86661 Atropine methyl nitrate 52-88-0 Atropine methyl bromide, a muscarinic receptor (mAChR) antagonist, is a quaternary ammonium salt of atropine and is the active molecule used for pupil dilation during ophthalmic examinations.
AZD-2115 V83201 AZD-2115 AZD-2115 is a muscarinic antagonist/beta 2 agonist (MABA).
Baogongteng A ((-)-Bao Gong Teng A) V84978 Baogongteng A ((-)-Bao Gong Teng A) 74239-84-2
BQCA V4096 BQCA 338747-41-4 BQCA, a benzylquinolone carboxylic acid, is a potent, highly selective positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR).
Dexetimide hydrochloride V94275 Dexetimide hydrochloride 21888-96-0 Dexrazoxane hydrochloride ((+)-benzamide hydrochloride) is an antimuscarinic drug with activity in suppressing antipsychotic-induced parkinsonism.
Dimethyl-W84 dibromide V101368 Dimethyl-W84 dibromide 402475-33-6 Dimethyl-W84 (dibromide) can modulate the M2 muscarinic acetylcholine receptor.
Eucatropine V70517 Eucatropine 100-91-4 Eucatropine is a potent muscarinic acetylcholine receptor (mAChR) inhibitor (antagonist) with IC50 of 0.583 μM.
Eucatropine hydrochloride V135450 Eucatropine hydrochloride 536-93-6 Eucatropine hydrochloride is a potent muscarinic acetylcholine receptor (mAChR) inhibitor with an IC50 value of 0.583 μM.
G-Protein antagonist peptide TFA V76963 G-Protein antagonist peptide TFA G-Protein antagonist peptide TFA is a truncated substance P-related peptide that competes with receptors for G protein binding.
M1/M2/M4 muscarinic agonist 2 V79209 M1/M2/M4 muscarinic agonist 2 M1/M2/M4 muscarinic agonist 2 (compound 43) is a muscarinic mAChR M1/M2/M4 agonist/activator with EC50s of 30 nM, 200 nM and 6.2 nM respectively.
M3/PDE4 modulator-1 V80656 M3/PDE4 modulator-1 M3/PDE4 modulator-1 (compound 10f) is a bifunctional molecule that is an M3 mAChR antagonist and a PDE4 inhibitor.
Milameline hydroiodide V93074 Milameline hydroiodide Miramelline (CI 979) hydroiodide is a muscarinic receptor agonist that improves cognitive abilities.
Muscarinic M4 modulator-1 V140525 Muscarinic M4 modulator-1 3082186-91-9 Muscarinic M4 modulator-1 is a positive allosteric modulator of the muscarinic M4 receptor.
p-F-HHSiD hydrochloride V103154 p-F-HHSiD hydrochloride 175615-76-6 pF-HHSiD (p-fluorohexahydrosilicinol) hydrochloride is a selective M3 mAChR antagonist.
PF-06764427 V114367 PF-06764427 1842371-08-7 PF-06764427 is a selective M1 muscarinic acetylcholine receptor positive allosteric modulator.
Propantheline-d3 bromide (Propantheline-d3 bromide) V70522 Propantheline-d3 bromide (Propantheline-d3 bromide) 64717-35-7 Propantheline-d3 (bromide) is the deuterated form of Propantheline bromide.
RS-86 V115495 RS-86 3576-73-6 RS-86 is a potent, centrally acting, selective muscarinic acetylcholine receptor agonist.
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