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Histamine Receptor

Histamine Receptor

Histamine Receptor related products

Structure Cat No. Product Name CAS No. Product Description
ABT-239 V4406 ABT-239 460746-46-7 ABT-239 is a novel, highly efficacious, non-imidazole class of H3R antagonist and a transient receptor potential vanilloid type 1 (TRPV1) antagonist/inverse agonist developed by Abbott with stimulant and nootropic effects, and has been investigated as a treatment for ADHD, Alzheimer's disease, and schizophrenia.
Aminopotentidine V97373 Aminopotentidine 140873-26-3 Aminopotentidine is a histamine H2 receptor antagonist with KB values of 220 and 280 nM for human and guinea pig H2 receptors, respectively.
Arpromidine V103940 Arpromidine 106669-71-0 Apromidine (BU-E-50) is a histamine H2 receptor agonist and histamine H1 receptor antagonist.
D-20133 V115308 D-20133 146764-26-3 D-20133 is an orally effective cetylphosphocholine analogue.
Elbanizine V107689 Elbanizine 110629-41-9 Albanizine inhibits histamine, bradykinin activity, histamine release from rat mast cells (IC50 0.26 μM), and IgE-mediated passive cutaneous anaphylaxis (PCA).
Fenspiride-d5 hydrochloride V135865 Fenspiride-d5 hydrochloride 1246815-28-0 Fenspiride-d5 hydrochloride is a deuterated fenspiride hydrochloride.
GSK189254A V2939 GSK189254A 720690-73-3 GSK189254A (also known as GSK189254) is a novel histamine H(3) receptor antagonist with high affinity for human (pK(i) = 9.59 -9.90) and rat (pK(i) = 8.51-9.17) H(3) receptors.
H3R antagonist 5 V137057 H3R antagonist 5 879368-27-1 H3R antagonist 5 is a selective histamine H3 receptor inverse agonist with an IC50 value of 0.54 nM and the ability to cross the blood-brain barrier.
Impromidine hydrochloride V94342 Impromidine hydrochloride 65573-02-6 Imoprodine is a potent histamine H2 receptor agonist.
JNJ-7777120 V1239 JNJ-7777120 459168-41-3 JNJ-7777120 (JNJ7777120; JNJ 7777120), an indole analog, is a potent and selective non-imidazole-based histamine H4R receptor antagonist that can reduce allergic and asthmatic symptoms.
N-ω-乙酰基组胺 V29682 N-Acetylhistamine 673-49-4 N-Acetylhistamine is a histamine metabolite.
Propiomazine maleate V109135 Propiomazine maleate 3568-23-8 Promethazine maleate is an effective oral antihistamine.
S 38093 V2789 S 38093 862896-30-8 S 38093 is a novel brain-penetrant antagonist (inverse agonist) of the H3 (histamine H3) receptor with Kiof 8.8, 1.44 and 1.2 µM for rat, mouse and human H3 receptors, respectively.
SCH 79687 V144669 SCH 79687 224585-45-9 SCH 79687 is an orally effective histamine H3 receptor antagonist with a Ki value of 1.9 nM in rats and 13 nM in guinea pigs.
Spinacetin V85156 Spinacetin 3153-83-1
Wy 45086 V147152 Wy 45086 87476-50-4 Wy 45086 is a histamine H2 receptor antagonist.
XmAb-7195 V147195 XmAb-7195 XmAb-7195 is a human monoclonal antibody (mAb) that targets IGH.
Zolantidine V117117 Zolantidine 104076-38-2 Zolantidine (SKF 95282) is a potent, selective, blood-brain barrier-crossing histamine H2 receptor antagonist.
σ1R/H3R ligand-1 V147782 σ1R/H3R ligand-1 σ1R/H3R ligand-1 is a dual σ1R/H3R antagonist with a Ki value of 8.8 nM for σ1R and 31.2 nM for H3R.
依匹斯汀 V29268 Epinastine (WAL801) 80012-43-7 Epinastine (also known as WAL-801CL HCl) is a potent antihistamine H1 without sedative activity and a mast cell stabilizer that is used in eye drops for the treatment of allergic conjunctivitis.
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