| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V2975 | B-Raf IN 1 | 950736-05-7 | B-Raf IN 1 is a novel, potent and selective B-Raf inhibitor with IC50 of 24 nM; it is equally potent against c-Raf with IC50 of 25 nM. |
|
V2989 | BT-11 | 1912399-75-7 | This product is discontinued due to commercial reason. |
|
V3271 | CB-1158 analog | 1345810-21-0 | CB-1158 analog (CB-1158, INCB01158 or Numidargistat analog) is a potent and orally bioavailable small-molecule inhibitor of the arginase with potential immunomodulating activities. |
|
V3167 | HDM201 R Enantiomer | 1448867-42-2 | HDM201 R Enantiomer is the R enantiomer of HDM201 (also called NVP-HDM201, HDM stands for human double minute 2 homolog). |
|
V2911 | HUHS015 | 1453097-13-6 | HUHS015 is a novel and potent inhibitor of PCA-1/ALKBH3 (prostate cancer antigen-1/AlkB Homolog 3) both in vitro and in vivo that was discovered from the optimization of a hit compound identified during random screening using a recombinant PCA-1/ALKBH3. |
|
V3040 | JWH-133 | 259869-55-1 | JWH-133 is a synthetic cannabinoid and a potent & selective agonist of the CB2 receptor with a Ki of 3.4nM and selectivity of ~ 200x for CB2 over CB1 receptors. |
|
V3188 | LGD-3303 | 917891-35-1 | LGD-3303is a potent,selective, orally bioavailable, and non-sterdoidal androgen receptor modulator (SARM) with anabolic effects on muscle and cortical bone not observed with bisphosphonates. |
|
V3259 | Mavorixafor (AMD-070) HCl | 880549-30-4 | Mavorixafor HCl (also known as AMD-1107, AMD070, X4P-001) is a potent, selective and orally bioavailable antagonist ofCXCR4 with anti-HIV activity. |
|
V3353 | MRK-016 HCl | 783331-24-8 | MRK-016 HCl (MRK016; MRK 016) is a novel, potent, orally bioactive and selective negative allosteric modulator (inverse agonist) of α5 subunit-containing GABAA with nootropic properties. |
|
V2948 | PF-3274167 | 900510-03-4 | Cligosiban (formerly known as PF-3274167) is a novel, potent, selective and high-affinity nonpeptideantagonist of oxytocin receptor(OTR) with Ki of 9.5 nM. |
|
V2947 | PF-915275 | 857290-04-1 | PF-915275 (PF915275) is a novel and selective inhibitor of human 11β-hydroxysteroid dehydrogenase type 1 (11betaHSD1) with Ki of<1 nM and good pharmacokinetics.11betaHSD1 play a key role in ligand-induced activation of the GR through the production of cortisol. |
|
V2955 | Ro 48-8071 fumarate | 189197-69-1 | Ro 48-8071 fumarate is an orally bioavailable inhibitor of OSC (Oxidosqualene cyclase) with IC50of ~6.5 nM. |
|
V3372 | Tirasemtiv | 1005491-05-3 | Tirasemtiv (also known as CK2017357) is a novel small-molecule activator of fast-skeletal-troponin, it is being developed as a potential treatment for diseases and conditions associated with aging, muscle weakness and wasting or neuromuscular dysfunction. |
|
V3021 | UNC1079 | 1418741-86-2 | UNC1079, the piperidine analog of UNC1021, is a structurally similar but significantly less potent inhibitor for use as a negative control in cellular studies. |
|
V2977 | Cebranopadol | 863513-91-1 | Cebranopadol (also known as GRT-6005) is a novel, first in class compound with potent agonist activity on ORL-1 (opioid receptor like -1) and the well established mu opioid receptor. |
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