| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V129699 | Axareotide | 2126833-17-6 | Axareotide is a somatostatin analogue. |
|
V70061 | BIM-23056 TFA | 1426173-61-6 | BIM 23056 TFA is a linear octapeptide and a potent sst3 and sst5 somatostatin receptor antagonist (inhibitor) with Kis of 10.8 and 5.7 respectively. |
|
V115388 | BIM-23197 | 168016-90-8 | BIM-23197 is a selective SST2 agonist (IC50 = 0.19 nM). |
|
V141584 | NOTA-TATE | 709043-21-0 | NOTA-TATE is a somatostatin receptor 2 (SSTR2) binder. |
|
V70051 | Paltusotine (CRN00808) | 2172870-89-0 | Paltusotine (CRN00808) is an orally bioactive, non-peptide selective somatostatin type 2 (SST2) receptor agonist. |
|
V96651 | Paltusotine hydrochloride | 2172875-40-8 | Paltusotine hydrochloride (CRN00808) is an orally active, non-peptide selective somatostatin type 2 (SST2) receptor agonist. |
|
V76656 | Pasireotide ditrifluoroacetate (Pasireotide ditrifluoroacetate; SOM230 ditrifluoroacetate; Pasireotide TFA salt) | Pasireotide (SOM230) ditrifluoroacetate is a long-acting cyclohexanide somatostatin analogue that can increase the agonist activity of somatostatin receptors, with pKi of 8.2/9.0 for sst1/2/3/4/5 respectively. | |
|
V51075 | PRL-2915 | 209006-18-8 | PRL 2915 is a potent human somatostatin subtype 2 receptor blocker (antagonist) (hsst2) with Ki of 12 nM. |
|
V145274 | SST1 receptor antagonist-1 | 868057-23-2 | SST1 receptor antagonist-1 is a selective somatostatin receptor 1 (SST1) antagonist with pKd values of 9.11 for rSST1 and 8.79 for hSST1. |
|
V145275 | SST1 receptor antagonist-2 | 524743-70-2 | SST1 receptor antagonist-2 is a piperazine derivative and a somatostatin receptor 1 (SST1) antagonist. |
|
V145276 | SSTR4 agonist 5 | 2761347-44-6 | SSTR4 agonist 5 is an orally potent somatostatin receptor 4 (SSTR4) agonist with an EC50 value of 0.228 nM. |
|
V103243 | SSTR4 agonist-1 | 1638588-92-7 | SSTR4 agonist-1 (Compound 47) is a selective agonist of somatostatin receptor 4 (SSTR4) with EC50 of 4.7 nM. |