| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V75381 | BMS-604992 free base (EX-1314 free base) | 760944-56-7 | BMS-604992 (EX-1314) free base is a selective, orally bioactive, small molecule growth hormone secretagogue receptor (GHSR) agonist. |
|
V86608 | Cortistatin-8 | 485803-62-1 | Cortistatin-8 (CST-8; PCFWKTCK) is a neuropeptide and a GHS-R1a antagonist that counteracts the secretion of ghrelin in response to gastric acid and modulates ghrelin release from somatotrophs in vitro. |
|
V75366 | Emoghrelin | 928262-58-2 | Emoghrelin is extracted from Polygonum multiflorum and stimulates the secretion of growth hormone through activation of ghrelin receptors. |
|
V136609 | GHSR-1a agonist-1 | 3060887-25-1 | GHSR-1a agonist-1 is an orally potent growth hormone secretagogue receptor 1a (GHSR-1a) agonist with an EC50 of 0.49 nM. |
|
V75378 | PF-6870961 | 2857112-06-0 | PF-6870961 is an inverse agonist of GHSR1a with Kis of 73.6 nM (human GHSR), 239 nM (rat GHSR) and 217 nM (dog GHSR). |
|
V145947 | Tezusomant | 2802416-72-2 | Tezusomant is a growth hormone receptor antagonist. |
|
V4686 | Anamorelin | 249921-19-5 | Anamorelin (formerly also known as RC-1291 and ONO-7643) is a novel, potent, and orally bioavailable ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay. |