| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V105029 | ABCG2-IN-4 | 2559759-63-4 | ABCG2-IN-4 (compound K31) is an orally available ABCG2 inhibitor that reduces the release of protoporphyrin IX (PPIX) from erythrocytes into plasma and prevents phototoxicity. |
|
V117213 | ABCG2-IN-5 | 190323-50-3 | ABCG2-IN-5 (compound 10) is a selective ABCG2 inhibitor with an IC50 value of 0.34 µM. |
|
V115602 | Ac22(Az8)2 | 2377858-65-4 | Ac22(Az8)2 is a selective BCRP inhibitor (EC50: 1-2 nM). |
|
V74159 | Ac32Az19 | 2760674-72-2 | Ac32Az19 is a potent, nontoxic, and selective BCRP inhibitor (antagonist) with EC50 of 13 nM in BCRP-overexpressing HEK293/R2 cells. |
|
V3037 | KS176 | 1253452-78-6 | KS176 is a novel potent and highly selective/specific inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter with IC50 values of 0.59 and 1.39 μM in Pheo A and Hoechst 33342 assays respectively. |
|
V13718 | RG 14620 | 136831-49-7 | RG 14620 (RG-14620),a non-phenolic tyrphostin analog, is a novel and potent EGFR inhibitor (IC50 = 3 μM) with anticancer activity. |