| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V4243 | AZD6482 S-isomer | 1173900-37-2 | AZD6482 S-isomer, is an isomer of AZD6482 which is a novel, potent, selective and ATP competitive PI3Kβ inhibitor with IC50 of 10 nM, 8-, 87- and is 109-fold more selective to PI3Kβ than PI3Kδ, PI3Kα and PI3Kγ in cell-free assays. |
|
V4062 | Protein degrader 1 TFA | 1631137-51-3 | Protein degrader 1 TFA (trifluoroacetic acid salt) is a novel and potent small molecule ligand forVHL (Von Hippel-Lindau), anE3 ligasewhich has been targeted in many PROTACs (proteolysis-targeting chimeras). |
|
V4042 | R(+)-SKF-38393A | 81702-42-3 | R(+)-SKF-38393A (the R-isomer of SKF3839A) is a novel potent and selective dopamine D1 receptor agonist with IC50 of 110 nM,the (+)-enantiomer is the active isomer. |
|
V4041 | SKF38393 | 67287-49-4 | SKF38393 (also known as SKF-38393A) is a novel potent and selective dopamine D1 receptor agonist with IC50 of 110 nM,the (+)-enantiomer is the active isomer. |
|
V4161 | Diroximel fumarate | 1577222-14-0 | Diroximel fumarate (also known as ALKS 8700) is a novel compound that is taken orally and rapidly converted into monomethyl fumarate (MMF). |
|
V4046 | Irosustat | 288628-05-7 | Irosustat (formerlyknown as STX64, BN83495 or 667 coumate) is a novel potent and irreversibleinhibitor of steroid sulfatasewith anIC50of 8 nM and has the potential for treating breast cancer. |
|
V4148 | Fenebrutinib (GDC-0853) HCl | 2128304-54-9 | Fenebrutinib HCl (formerly known RG-7845; GDC-0853 hydrochloride) is an orally bioavailable, and noncovalent (reversible) brutons tyrosine kinase (BTK) inhibitor (Ki = 0.91 nM) with anticancer and anti-inflammatory activity. |