| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V73372 | 5-Amino-8-hydroxyquinoline (5A8HQ) | 13207-66-4 | 5-Amino-8-hydroxyquinoline (5A8HQ) is a potential anticancer candidate active molecule with good proteasome inhibitory activity |
|
V87690 | Ac-RLR-AMC TFA | Ac-RLR-AMC (Ac-Arg-Leu-Arg-AMC) TFA is a fluorescent substrate for the 26S proteasome (Ex/Em: 380/440-460 nm). | |
|
V84788 | ARI-3144 | 1426305-25-0 | |
|
V118625 | Az-NC-002 | 1356828-49-3 | Az-NC-002 is a proteasome trypsin-like site (β2) and immunoproteasome β2i specific active probe. |
|
V130063 | Berberine-amide-m-PhBA chloride | Berberine-amide-m-PhBA chloride is a selective anti-breast cancer drug. | |
|
V118624 | Biotin-(Oaa)3-epoxomicin | 247068-92-4 | Biotin-(Oaa)3-cyclooxymycin (compound 13) is the biotinylated active form of cyclooxymycin. |
|
V118594 | Biotin-epoxomicin | 1334608-28-4 | Biotin-labeled cyclooxygenin is a biotin-labeled cyclooxygenin. |
|
V106750 | Bortezomib impurity A | 289472-80-6 | Bortezomib impurity A is a metabolite of the 20S proteasome inhibitor bortezomib. |
|
V73368 | Enzyme-IN-1 | 868540-02-7 | Enzyme-IN-1 (compound 1) is a bioactive peptide-based N-terminal nucleophile (Ntn) hydrolase inhibitor. |
|
V94368 | Immunoproteasome activator 1 | 901728-48-1 | Immunoproteasome activator 1 (Compound A) is a selective immunoproteasome activator that increases the presentation of a single MHC-I-bound peptide by more than 100-fold. |
|
V110763 | INVA8001 | 1312993-34-2 | INVA8001 (ASB17061) is a highly selective, orally effective chymotrypsin inhibitor with IC50 values of 0.02 μM for human chymotrypsin and 0.03 μM for mouse mast cell protease-4 (mMCP-4). |
|
V105970 | Phepropeptin C | 396729-25-2 | Phepropeptin C is a microbial secondary metabolite and proteasome inhibitor with IC50 of 12.5 μg/mL. |
|
V143847 | RAPRMT5 | 2721998-42-9 | RAPRMT5 is a PRMT5 CAP-TAC (protease complex targeting chimera) degrader. |
|
V109931 | UR238 | 2728747-80-4 | UR238 is a proteasome inhibitor. |
|
V73387 | Z-Leu-Leu-Glu-βNA (Z-Leu-Leu-Glu-β-naphthylamide) | 75873-85-7 | Z-Leu-Leu-Glu-βNA (Z-Leu-Leu-Glu-β-naphthylamide) is a substrate for the determination of 20S proteasome glutamyl peptide hydrolase activity. |
|
V81804 | β5i-IN-1 | β5i-IN-1 is a potent selective inhibitor of β5i with IC50 of 8.463 nM. | |
|
V4408 | Alicapistat | 1254698-46-8 | Alicapistat (also known as ABT957; ABT-957) is a novel, potent,selective and orally bioactive inhibitor of humancalpains 1and2whose overactivation has been linked to Alzheimer disease (AD). |