| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V88105 | 4-Cyano-3-methylisoquinoline | 161468-32-2 | 4-Cyano-3-methylisoquinoline is a protein kinase A (PKA) inhibitor with IC50 in the micromolar range. |
|
V1847 | 8-Bromo-cAMP sodium | 76939-46-3 | 8-Bromo-cAMP sodium is a potent and cell permeable cyclic AMP (cAMP) analog and a PKA activator. |
|
V130684 | BRP | BRP is a 12-peptide derived from BRINP2 that can cross the blood-brain barrier. | |
|
V2841 | CCG215022 | 1813527-81-9 | CCG215022 is a potent GRK2 and GRK5 inhibitor that exhibited nanomolar IC50 values against both GRK2 and GRK5 and good selectivity against other closely related kinases such as GRK1 and PKA. |
|
V69106 | GEM-231 (HYBO-165) | 255810-66-3 | GEM231 is an antisense oligonucleotide targeting PKA-I (RIα regulatory subunit of cAMP-dependent protein kinase type I) mRNA. |
|
V136966 | GSK-3α/β-IN-1 | 1574354-24-7 | GSK-3α/β-IN-1 is a GSK-3α/β inhibitor with IC50 values of 0.265 μM for GSK-3α and 0.255 μM for GSK-3β. |
|
V76627 | PKA Inhibitor Fragment (6-22) amide TFA (PKI-(6-22)-amide TFA) | PKA Inhibitor Fragment (6-22) amide TFA is an inhibitor (blocker/antagonist) of cAMP-dependent protein kinase A (PKA) with a Ki of 2.8 nM. | |
|
V88094 | PKA RII peptide TFA | PKA RII peptide TFA is a PKA substrate that can be used to detect calcineurin activity after phosphorylation at serine residues. | |
|
V88121 | SMO-IN-4 | 1567963-99-8 | SMO-IN-4 (Compound 24) is a potent and orally active smoothened antagonist (IC50: 24 nM). |
|
V88118 | Sp-8-Br-PET-cGMPS | 172806-21-2 | Sp-8-Br-PET-cGMPS is a membrane-permeable PKG agonist, a membrane-permeable retinal cGMP-gated ion channel inhibitor, and an activator of cGMP-dependent protein kinases I α and I β. |
|
V69123 | Sp-8-CPT-cAMPS | 129693-13-6 | Sp-8-CPT-cAMPS, a cAMP analog, is a potent and specific activator of cAMP-dependent protein kinase A PKA I and PKA II. |
|
V88099 | Sp-cAMPS-AM | 152218-24-1 | Sp-cAMPS-AM is a cAMP analog. |
|
V145932 | Tetramisole | 5036-02-2 | Tetramisole is an orally effective selective inward rectifying potassium channel agonist with an EC50 value of approximately 30 μM for the Kir2.1 subunit. |