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Adenosine Receptor

Adenosine Receptor

Adenosine Receptor related products

Structure Cat No. Product Name CAS No. Product Description
A2AAR antagonist 3 V127970 A2AAR antagonist 3 A2AAR antagonist 3 is a selective and potent A2A adenosine receptor (A2A AR) antagonist with an IC50 value of 1.57 nM.
A2AAR antagonist 4 V119241 A2AAR antagonist 4 A2AAR antagonist 4 is an orally effective A2A adenosine receptor antagonist with a Ki value of 0.36 nM and a KB value of 1 nM for human A2AAR.
A2AR-antagonist-1 V51753 A2AR-antagonist-1 2922920-71-4 A2AR-antagonist-1 (compound 38) is a potent cervical adenylate A2A receptor (A2AR) clamp antagonist (IC50=29 nM).
A2A受体拮抗剂1 V3128 A2A receptor antagonist 1 443103-97-7 A2A receptor antagonist 1 is a novel and potent antagonist of the adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
A3AR agonist 3 V103545 A3AR agonist 3 3032474-53-3 A3AR agonist 3 (Compound 15A) is an A3 adenosine receptor (A3AR) agonist with a Ki value of 2.27 nM for hA3 and an EC50 value of 0.20 nM for cAMP.
A3AR agonist 4 V92167 A3AR agonist 4 3032475-23-0 A3AR agonist 4 is a A3 adenosine receptor (A3AR) agonist (Ki 1.24 nM for hA3AR).
A3AR modulator 1 V79210 A3AR modulator 1 A3AR modulator 1 (MRS8054) is an orally bioactive A3AR (Adenosine Receptor) PAM (positive allosteric modulator).
CGS 21680 HCl V1482 CGS 21680 HCl 124431-80-7 CGS 21680 HCl (CGS21680; CGS-21680), the hydrochloride salt of CGS 21680,is a potent and specific agonist of adenosine A2 receptors with potential antideppressant activity.
DPTN dihydrochloride V75276 DPTN dihydrochloride 325767-87-1 DPTN is a potent and specific antagonist of human, mouse and rat A3AR with Kis of 1.65, 9.61 and 8.53 nM respectively.
MRS-3777 hemioxalate V75262 MRS-3777 hemioxalate 1186195-57-2 MRS-3777 hemioxalate is a selective adenosine A3 receptor blocker (antagonist).
MRS7935 V80840 MRS7935 MRS7935 (compound 15) is an A1AR positive allosteric modulator (PAM) with EC50 of about 2 μM.
N 0861 V101847 N 0861 141696-90-4 N-0861 is a novel selective A1 adenosine receptor antagonist that can inhibit the negative conduction effects (prolonged AH interval) and chest pain caused by adenosine, but has no significant effect on the increase in coronary blood flow velocity caused by adenosine.
SCH-58261 V2917 SCH-58261 160098-96-4 SCH-58261 (SCH58261; SCH 58261) is a novel, potent, selective and competitive antagonist of the adenosine A2A receptor with immunomodulatory and neuroprotective effects.
SYAF080 V145482 SYAF080 352692-70-7 SYAF080 is a human A₂B adenosine receptor (hA₂B AdoR) antagonist with a Ki value of 23.6 nM and a KB value of 25.2 nM.
XCC V84699 XCC 96865-83-7
Zaladenant V147289 Zaladenant 2246426-52-6 Zaladenant is an adenosine receptor antagonist with antitumor activity.
伊曲茶碱 V1483 Istradefylline (KW-6002) 155270-99-8 Istradefylline (formerly KW6002; KW 6002; KW-6002; Nourianz), a caffeine derivative, is an orally bioavailable and selective adenosine A2A receptor (A2AR) antagonist with anti-PD (Parkinson's disease) effects.
去甲肾上腺素 V13165 Norepinephrine (Levarterenol; L-Noradrenaline) 51-41-2 Norepinephrine (Levarterenol; L-Noradrenaline) is a potent and β1-selective adrenergic receptor agonist with EC50 of 5.37 μM.
盐酸托屈嗪 V16551 Todralazine hydrochloride 3778-76-5 Todralazine HCl (Ecarazine HCl) is an anti-hypertensive (blood pressure lowering) agent, a β2 adrenergic receptor (β2AR) blocker, and has antioxidant and free radical scavenging activities.
茶碱-7-乙酸 V3126 Acefylline 652-37-9 Acefylline (also known as Theophylline-7-acetic acid and Theophyllineacetic acid), is an antagonist of theadenosine receptor and an activator of the peptidylarginine deiminase (PAD).
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