| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V136432 | FXR DUBTAC IN-1 | 3081876-96-9 | FXR DUBTAC IN-1 is a chimeric molecule (DUBTAC) that targets deubiquitinase. It targets FXR and has a Ka value of 2.12 × 10⁻⁵ M for FXR. |
|
V136647 | GK13R | GK13R is a less active enantiomer of GK13S. | |
|
V51255 | IU1-248 | 2307472-03-1 | IU1-248 is an analogue of IU1 and a potent and specific USP14 inhibitor (antagonist) with IC50 of 0.83 μM. |
|
V138205 | IU2-6 | 1356074-25-3 | IU2-6 is a USP14 deubiquitinase inhibitor. |
|
V140440 | MS7131 | The MS7131 is a USP1 recruiting DUBTAC. | |
|
V146812 | USP1-IN-11 | USP1-IN-11 is a selective, reversible, non-competitive USP1 (ubiquitin-specific protease 1) inhibitor. | |
|
V146813 | USP1-IN-12 | 2961035-60-7 | USP1-IN-12 is a potent and orally effective USP1 inhibitor with an IC50 value of 0.00366 µM. |
|
V146814 | USP1-IN-13 | 2974433-50-4 | USP1-IN-13 is a potent and orally effective USP1 inhibitor with an IC50 value of 1.02 nM. |
|
V146815 | USP1-IN-16 | 3084671-46-2 | USP1-IN-16 is a USP1 inhibitor with an IC50 value of 0.002 μM for USP1-UAF1. |
|
V146816 | USP1-IN-17 | USP1-IN-17 is an orally effective inhibitor of the USP1/UAF1 complex. | |
|
V146811 | USP10-IN-1 | 904448-58-4 | USP10-IN-1 is a USP10 inhibitor. |
|
V51241 | Usp22i-S02 | 309735-96-4 | USP22 inhibitor |
|
V146817 | USP25/28-IN-2 | 2165322-95-0 | USP25/28-IN-2 is a selective dual USP25/USP28 inhibitor with an IC50 value of 0.9 μM and a Ka value of 0.9 μM for USP28, and an IC50 value of 0.88 μM for USP25. |
|
V146819 | USP7 activator 1 | 868940-26-5 | USP7 Activator 1 (compound MS-8) activates USP7 by binding to the allosteric C-terminal binding pocket of USP7. |
|
V146820 | USP7 Ligand-Linker Conjugates 1 | 3098774-65-0 | USP7 Ligand-Linker Conjugates 1 is a target protein ligand-linker conjugate containing a USP7 ligand and a PROTAC linker that recruits E3 ligases. |
|
V146821 | USP7-IN-17 | 1174836-23-7 | USP7-IN-17 is a potent USP7 inhibitor. |
|
V146823 | USP7-IN-19 | USP7-IN-19 is a USP7 inhibitor. | |
|
V51247 | USP8-IN-3 | 2477651-10-6 | deubiquitinase USP8 inhibitor |
|
V147324 | ZHAWOC8655 | 1257657-02-5 | ZHAWOC8655 is a USP18 inhibitor with an IC50 of 14.1 μM for hUSP18. |