| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V56638 | 17β-HSD10-IN-2 | 2316765-79-2 | 17β-HSD10-IN-2 (compound 11) is a benzothiazuride-based inhibitor that targets 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10), a multifunctional mitochondrial enzyme. |
|
V55746 | Anemonin (Pulsatilla camphor; Anemonine; trans-Anemonin) | 508-44-1 | Anemonin (Pulsatilla camphor), a selective iNOS inhibitor, is also a PKC-θ inhibitor. |
|
V56731 | B-Raf IN 15 | 832107-31-0 | BRAF V600E/CRAF-IN-3 (Compound 7) is a BRAF inhibitor. |
|
V56739 | BE1218 | 2893967-40-1 | BE1218 is a liver X receptor (LXR) inverse agonist with IC50s of 9 nM and 7 nM for LXRα and LXRβ, respectively. |
|
V56676 | CEE321 | 2098545-89-0 | CEE321 is a potent pan-JAK inhibitor (IC50 = 54 nM) in enzymatic and cellular assays. |
|
V56586 | CGS20625 | 111205-55-1 | CGS-20625 is an anti-anxiety drug for scientific research. |
|
V52255 | CHR-6494 TFA | 1458630-17-5 | CHR-6494 TFA is a potent and specific haspin inhibitor (antagonist) with IC50 of 2 nM. |
|
V56816 | CYP4Z1-IN-1 | 2760611-38-7 | CYP4Z1-IN-1 (compound 7c) is a potent inhibitor of CYP4Z1 with IC50 of 41.8 nM. |
|
V56777 | DPTIP | 351353-48-5 | DPTIP is a potent, BBB (blood-brain barrier) permeable/penetrable neutral sphingomyelinase (N-SMase 2) (exosome inhibitor) with IC50 of 30 nM. |
|
V56596 | Gcase activator 2 | 2759897-35-1 | Gcase activator 2 (compound 14) is a pyrrole[2,3-b]pyrazine and a β-glucocerebrosidase (Gcase) activator (EC50=3.8 μM). |
|
V56687 | GSK251 | 2125968-05-8 | GSK251 is a highly efficient, selective, orally bioavailable PI3Kδ inhibitor (antagonist) with a novel binding mode. |
|
V56712 | GW438014 free base | 469861-48-1 | GW438014A is a selective NPY-Y5 receptor antagonist. |
|
V56746 | HaloPROTAC3 | 1799506-07-2 | HaloPROTAC3 is a degrader of HaloTag fusion proteins. |
|
V56749 | HUN39963 | 893739-96-3 | HUN39963, also known as LDH-IN-2, is an inhibitor (blocker/antagonist) of glycolate oxidase. |
|
V56794 | MAO-B-IN-19 | 152897-41-1 | MAO-B-IN-19) is a selective MAO-B inhibitor (antagonist) with IC50 of 0.67 μM. |
|
V56805 | Moracin M | 56317-21-6 | Moracin M is a phosphodiesterase 4 inhibitor extracted from Morus alba. |
|
V56799 | NCGC00135472 | 862811-76-5 | NCGC00135472 is an agonist of the human Resolvin D1 receptor DRV1 and has pro-resolving function. |
|
V56641 | NCRW0005-F05 | 342779-66-2 | NCRW0005-F05 is a potent GPR139 antagonist (inhibitor) with IC50 of 0.21 μM. |
|
V56677 | NSC243928 | 59988-01-1 | NSC243928 mesylate is a human lymphocyte antigen 6 (LY6) binder that also works as a cell growth inhibitor and has anti-cancer effect. |
|
V56664 | Nurr1 agonist 2 | 742058-34-0 | Nurr1 agonist 2 (Compound 7) is a Nurr1 agonist (EC50= 0.07 μM). |