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Glucocorticoid Receptor

Glucocorticoid Receptor

Glucocorticoid Receptor related products

Structure Cat No. Product Name CAS No. Product Description
AL082D06 V2896 AL082D06 256925-03-8 AL082D06 (formerly known as D-06), is a nonsteroidal glucocorticoid receptor (GR) antagonist which is characterized by a tri-aryl methane core chemical structure.
Glucocorticoid receptor agonist-1 V67727 Glucocorticoid receptor agonist-1 2166375-82-0 Glucocorticoid receptor agonist-1 is a potent and specific glucocorticoid receptor agonist/activator with IC50 of 2.8 nM.
GSK9027 V67733 GSK9027 1229096-88-1 GSK9027 is a nonsteroidal glucocorticoid receptor (GR) agonist that behaves as a partial agonist on the 2× glucocorticoid response element (GRE) reporter system and achieves intrinsic activity relative to dexamethasone.
HP210 V67742 HP210 728039-52-9 HP210 is a selective glucocorticoid receptor modulator (SGRM).
SelDeg51 V144758 SelDeg51 3036372-80-9 SelDeg51 is a selective FKBP51 PROTAC degrader with a Kd value of 18 nM and a Dmax value of 90%.
Sesaminone V144806 Sesaminone 157207-93-7 Sesaminone is a lignan found in magnolia leaves.
Tegacorat V145722 Tegacorat 2409551-99-9 Tegacorat is a glucocorticoid receptor agonist with an EC50 < 100 nM.
Triamcinolone acetonide-d7 V146435 Triamcinolone acetonide-d7 Triamcinolone acetonide-d7 is a deuterated triamcinolone.
Win 45164 V147114 Win 45164 83880-39-1 Win 45164 is an orally effective glucocorticoid receptor ligand that inhibits the pituitary-adrenal axis.
丙酸倍氯米松 V1716 Beclomethasone dipropionate (Beclomethasone) 5534-09-8 Beclomethasone dipropionate (also called BDP;Clenil; Qvar; Beconase; alanase; Vancenase) is a topical anti-inflammatory corticosteroid approved for use in treatment of asthma and rhinitis.
曲安西龙 V1719 Triamcinolone 124-94-7 Triamcinolone (BRN2341955;Adcortyl; BRN-2341955; Aristocort),a long-acting synthetic corticosteroid, is an approved glucocorticoid medication with anti-inflammatory activities.
氟米松 V1720 Flumethasone (Flumetasone) 2135-17-3 Flumethasone (NSC-54702;RS-2177; U-10974;RS2177; BRN-5645455;NSC54702; Anaprime; Aniprime; Fluvet; Methagon; Cortexilar; Flucort; Flucorticin;Locacorten),a topically used corticosteroid, is a potent glucocorticoid receptor agonist with potential anti-inflammatory activity.
醋酸氟轻松 V1717 Fluocinolone Acetonide 67-73-2 Fluocinolone Acetonide (Flucort-N;Flucinar, Fluonid, Synandone, Jellin, Sinalar) is a topical and synthetic glucocorticoid withwith anti-inflammatory and immunomodulating properties.
醋酸泼尼松龙 V1718 Prednisolone Acetate (Omnipred) 52-21-1 Prednisolone Acetate (also called Omnipred; Prednisolone 21-acetate) is a synthetic corticosteroid drug approved for use as an immunosuppressant,anti-inflammatory, and anti-allergicagent.
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