| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V89083 | 17-Epiestriol | 1228-72-4 | 17-Epiestriol is an estrogen metabolite and a selective estrogen receptor (ER) β agonist. |
|
V125335 | 3-Cl-Pyridine-amide-acrylaldehyde-piperazine | 3-Cl-Pyridine-amide-acrylaldehyde-piperazine is a synthetic intermediate for LO-4-25. | |
|
V8411 | AC-262536 | 870888-46-3 | AC-262536 (AC262536) is anovel selective androgen receptor modulator (SARM) with beneficial anabolic effects. |
|
V93122 | Androgen receptor antagonist 12 | 6605-17-0 | Androgen receptor antagonist 12 (Compound EF2) is an orally active androgen receptor (AR) antagonist (IC50: 0.30 μM). |
|
V88176 | Androgen receptor-IN-4 | 2759137-87-4 | Androgen Receptor-IN-4 (Compound 206) is an androgen receptor inhibitor that can be used in the study of Kennedy's disease. |
|
V129322 | AR antagonist 13 | AR antagonist 13 is an androgen receptor antagonist with an inhibition rate of over 71.5% at a concentration of 10 μM. | |
|
V117158 | AR antagonist 17 | 3064715-04-1 | AR antagonist 17 is a selective, orally active, blood-brain barrier resistant androgen receptor (AR) antagonist (IC50 = 0.010 μM) that effectively blocks AR dimerization and nuclear translocation, exhibiting potent activity in various castration-resistant prostate cancer (CRPC) cells. |
|
V85093 | AR antagonist 5 | 2902679-53-0 | |
|
V101111 | AZ'3137 | 2960179-55-7 | AZ'3137 (Compound 22) is an orally active PROTAC-based androgen receptor (AR) degrader with a DC50 value of 22 nM. |
|
V41443 | Bavdegalutamide (ARV-110) | 2222112-77-6 | Bavdegalutamide (ARV110; ARV-110) is an orally bioavailable PROTAC-based Androgen Receptor (AR) degrader (DC₅₀ = ~1 nM) with potentialanticancer activity. |
|
V132526 | C-Terminally encoded peptide 1 | C-Terminally Encoded Peptide 1 is a small molecule secreted peptide hormone. | |
|
V131323 | CDPP-2PF6 | ||
|
V116219 | Ch-319 | 2589088-07-1 | Ch-319 is a triphenyltin(IV) carboxylate derivative. |
|
V132133 | CP61 | 1631984-43-4 | CP61 is a cyclic peptide with dual CtBP1/CtBP2 inhibitory activity. |
|
V97765 | FL442 | 1431166-12-9 | FL442 is an androgen receptor (AR) modulator. |
|
V115700 | Galeterone hydrochloride | 1239339-17-3 | Galactone hydrochloride (TOK-001) is a potent oral biodegrader that degrades androgen receptor (AR) and its splice variant (AR-V), as well as serine/threonine protein kinases Mnk1/2 that interact with MAP kinase. |
|
V109012 | ITRI-90 | 2798907-16-9 | ITRI-90 is an orally effective androgen receptor (AR) protein degrader. |
|
V3518 | KX-826 | 1272719-00-2 | This product is discontinued due to commercial reason. KX826( also known as Pyrilutamide ) is an androgen receptor (AR) antagonist and a potential first-in-class topical drug for the treatment of androgenetic alopecia (AGA) and acne vulgaris. |
|
V4852 | LY-2452473 | 1029692-15-6 | LY2452473 is a novel, potent, selective and orally bioavailable androgen receptor modulator (SARM) with potential tissue-selective androgenic/anti-androgenic activity. |
|
V141430 | NLX-219 | 2170404-93-8 | NLX-219 is a selective 5-HT1A receptor agonist with a pKi value of 10.21. |