G protein-coupled Bile Acid Receptor

ADC Related

ADC Antibody ADC Cytotoxin ADC Linker ADCs Drug-Linker Conjugates for ADC
Angiogenesis

5-alpha Reductase ALK Bcr-Abl BTK EGFR FAK FLT3 HER-2 HIF Src Syk VDA VEGFR
Anti-infection

Antibiotic Arenavirus Bacterial CMV EBV Enterovirus Filovirus Fungal Gli HBV HCV HCV Protease HIV HSV Influenza Virus Parasite RABV Reverse Transcriptase RSV SARS-CoV TMV Virus Protease
Apoptosis

Apoptosis ASK Bcl-2 Caspase c-Myc c-RET Cytohesin DAPK Ferroptosis FKBP IAP Mdm2 p53 PD-1 PD-L1 PERK PKD Ras RIP kinase ROS Survivin Thymidylate Synthase TNF Receptor TNFa TRADD
Autophagy

Autophagy LRRK2 Mitophagy OGA ULK
Cell Cycle

Antifolate APC Aurora Kinase BMI-1 CDK Chk c-Myc Eukaryotic Initiation Factor G-quadruplex HDAC HSP Kinesin LIMK Mad2 Microtubule(Tubulin) Mps1 Nucleoside Antimetabolite/Analog Nur77 p21 PAK PERK PFKFB PLK PPAR Ras Rho ROCK SRPK TOPK Topoisomerase Wee1
Cytoskeletal Signaling

Arp2 3 Complex Bcr-Abl Cardiac Myosin Dynamin Gap Junction Protein HSP Integrin Kinesin Microtubule Associated MLCK Myosin PAK TACC3 Wntbeta-catenin
DNA Damage

ATM(ATR) CRISPR(Cas9) DNA alkylator DNA Stain DNA(RNA) Synthesis GAK HDAC HSP Nucleoside Antimetabolite(Analog) OGG1 p97 PARG PARP RAD51 RNR Sirtuin SMN Telomerase Topoisomerase
Endocrinology & Hormones

5-alpha Reductase ACE Adrenergic Receptor Androgen Receptor Aromatase Estrogenprogestogen Receptor Glucocorticoid Receptor GPR Mineralocorticoid Receptor RAAS THR TSH Receptor
Epigenetics

AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain EZH1 2 HDAC HIF Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MAT MicroRNA MLL Pim PKC Protein Arginine Deiminase Sirtuin Small Interfering RNA (siRNA) SMYD

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G protein-coupled Bile Acid Receptor

G protein-coupled Bile Acid Receptor related products

Cat No.	Product Name	CAS No.	Product Description
V125529	3-MPPI	133399-65-2	3-MPPI is a G protein-coupled receptor (GPCR) ligand with high selectivity for α1-adrenergic receptors. Its Ki value for α1-adrenergic receptors is 0.21 nM, and its Ki value for 5-HT1A receptors is 50 nM.
V144068	RG-239	1199222-56-4	RG-239 is an orally effective TGR5 agonist with an EC50 value of 120 nM, which is significantly better than betulinic acid (EC50 = 1.04 μM).
V145277	SSTR5/TGR5-modulator-1	3069267-46-2	SSTR5/TGR5-modulator-1 is an orally effective dual-target small molecule that exhibits balanced activity against both human TGR5 and human SSTR5 in vitro.
V15922	TC-G 1005	1415407-60-1	TC-G 1005 (TC-G-1005; TCG1005) is a novel, oral and potent TGR5 (GPBAR1) agonist with glucose-lowering effects.
V145971	TGR5 agonist 10	3081614-92-5	TGR5 agonist 10 is a selective, allosteric, and orally effective Takeda G protein-coupled receptor 5 (TGR5) agonist with EC50 values of 0.8 μM for human TGR5 and 0.6 μM for mouse TGR5.
V145972	TGR5 agonist 7		TGR5 agonist 7 is an intestinal-restricted, orally effective G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) agonist with an EC50 < 1 μM.
V2862	TGR5 Receptor Agonist	1197300-24-5	TGR5 Receptor Agonist is a novel, potent andsynthetic small molecule agonist of TGR5 (G-protein coupled receptor19, GPCR19), it showed improved potency in the U2-OS cell assay with pEC50 of 6.8 and in melanophore cells with pEC50 of 7.5.