| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V2724 | 10074-G5 | 413611-93-5 | 10074-G5 is a potent inhibitor of c-Myc-Max dimerization and interaction with an IC50 of 146 μM and with anticancer activities. |
|
V1587 | 10058-F4 | 403811-55-2 | 10058-F4 (10058F4; 10058 F4) is a novel potent and selective c-Myc inhibitor with potential antineoplastic activity. |
|
V129674 | AV-9606-129 | 783309-48-8 | AV-9606-129 is a USP28 inhibitor with an IC50 < 1 μM. |
|
V113262 | Hydroxyrubicin | 73113-90-3 | Hydroxyrubicin is an anti-tumor drug. |
|
V138437 | KI-CDK9d-32 | 3054009-82-1 | KI-CDK9d-32 is a highly selective and highly active CDK9 PROTAC degrader (DC50: 0.89 nM). |
|
V138459 | KL4-219A | KL4-219A is a selective covalently binding degrader of the oncogenic transcription factor MYC. | |
|
V142853 | PLK1-IN-13 | 3038489-48-1 | PLK1-IN-13 is a selective, orally active PLK1 inhibitor (IC50: 0.27 nM). |
|
V144393 | RS47 | 301655-16-3 | RS47 is a selective RelB inhibitor with a Kd value of 1.1 μM. |
|
V144811 | SF-3-030 | 1883721-73-0 | SF-3-030 is a highly effective, selective, and non-ATP-competitive ERK1/2 inhibitor. |
|
V144824 | SGI-1776-VHL-02 | 3013618-84-0 | SGI-1776-VHL-02 is a stereoselective PIM PROTAC degrader. |
|
V144825 | SGI-1776-VHL-02-epimer | 3013618-85-1 | SGI-1776-VHL-02-epimer is the epimer control compound of SGI-1776-VHL-02. |
|
V145297 | STAT3-IN-53 | 3113051-34-3 | STAT3-IN-53 is a STAT3 inhibitor with a Kd value of 6.16 μM. |
|
V145469 | SVC112 | SVC112 is a translation elongation inhibitor that prevents EF2 from cyclically dissociating from the ribosome, thereby inhibiting the elongation step of translation. | |
|
V146201 | TNIK-IN-10 | 3112758-72-9 | TNIK-IN-10 is a TNIK inhibitor with an IC50 value of 0.49 nM for human TNIK. |
|
V146695 | TZ1104 | TZ1104 is a PROTAC-based CDK7 degrader with a half-maximal lethal concentration (DC50) of 0.88 nM. | |
|
V147039 | VTX-0811 | VTX-0811 is a human IgG4 monoclonal antibody (mAb) that targets PSGL1/CD162. | |
|
V147087 | WDR5-MYC-IN-2 | 3062125-47-4 | WDR5-MYC-IN-2 is a WDR5-MYC protein-protein interaction (PPI) inhibitor with an IC50 of 0.59 μM. |
|
V147205 | XY25026 | XY25026 is an orally effective LRH-1 inhibitor with an IC50 value of 0.28 μM. | |
|
V147206 | XY25028 | XY25028 is an orally effective LRH-1 inhibitor with an IC50 of 0.30 μM. | |
|
V147220 | Y-99 | 2034334-74-0 | Y-99 is a PORCN inhibitor with an IC50 value of 155.4 nM for the Wnt/β-catenin signaling pathway. |