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Neurokinin Receptor

Neurokinin Receptor

Neurokinin Receptor related products

Structure Cat No. Product Name CAS No. Product Description
(1R,2S,3R)-Aprepitant V121316 (1R,2S,3R)-Aprepitant 1185502-97-9 (1R,2S,3R)-Aprepitant is a competitive human neurokinin-1 (NK-1) receptor antagonist.
(Trp7,β-Ala8)-Neurokinin A (4-10) V70807 (Trp7,β-Ala8)-Neurokinin A (4-10) 132041-95-3 (Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist.
(β-Ala8)-Neurokinin A (4-10) V70819 (β-Ala8)-Neurokinin A (4-10) 127633-71-0 (β-Ala8)-Neurokinin A (4-10) is a neuropeptide and a potent and specific NK-2 (Neurokinin Receptor) tachykinin receptor agonist (activator).
[Glp5,Sar9] Substance P (5-11) V70809 [Glp5,Sar9] Substance P (5-11) 77128-78-0 [Glp5,Sar9] Substance P (5-11) is an analog of Substance P.
GR 83074 V70806 GR 83074 141636-44-4 GR 83074 is a potent and specific NK-2 (Neurokinin Receptor) antagonist (inhibitor) with a pKB of 8.23.
GR 87389 V70793 GR 87389 141663-86-7 GR 87389 is a potent NK2 receptor antagonist.
GR 94800 TFA V79645 GR 94800 TFA GR 94800 TFA is a potent and specific peptide antagonist of neurokinin 2 (NK2) receptors with pKB values of 9.6, 6.4 and 6.0 for NK2, NK1 and NK3 receptors respectively.
Neurokinin A(4-10) TFA V76709 Neurokinin A(4-10) TFA Neurokinin A (4-10) TFA is a tachykinin NK2 receptor agonist (activator).
Neurotensin(8-13) TFA V94292 Neurotensin(8-13) TFA 2952825-79-3 Neurotensin (8-13) is the active fragment of neurotensin.
NK3R antagonist-1 V141405 NK3R antagonist-1 NK3R antagonist-1 is an orally effective neurokinin-3 receptor (NK3R) antagonist with an IC50 value of 53.61 nM.
RO4583298 V115455 RO4583298 825643-56-9 RO4583298 is a potent dual antagonist of NK1 (human and gerbil)/NK3 (human, cynomolgus monkey, gerbil and guinea pig) receptors.
RO5328673 V144259 RO5328673 1310817-94-7 RO5328673 is an orally effective, blood-brain barrier-crossing neurokinin receptor antagonist that effectively targets human NK3 receptors (Ki=0.4 nM, Ka=0.1 nM), human NK2 receptors (Ki=1.1 nM, Ka=0.9 nM), and guinea pig NK3 receptors (Ka=0.1 nM and 0.13 nM).
Senktide TFA V144777 Senktide TFA Senktide TFA is a potent, selective neuromodulatory K3 (NK3) receptor agonist (EC50 = 0.5-3 nM).
SLV-317 V86679 SLV-317 393183-40-9 SLV-317 is an orally active neurokinin-1 receptor antagonist.
Substance P (3-11) acetate V118516 Substance P (3-11) acetate Substance P (3-11) acetate is a peptide fragment of substance P (SP) that can cross the blood-brain barrier.
Substance P, free acid TFA V145384 Substance P, free acid TFA Substance P, free acid TFA is a natural analogue of substance P, but it lacks the biological activity of substance P.
Y1 receptor antagonist 1 formic V97448 Y1 receptor antagonist 1 formic Y1 receptor antagonist 1 formate (H 409-22 isomer formate) is the formate salt form of Y1 receptor antagonist 1.
γ-Neuropeptide (rabbit) V70805 γ-Neuropeptide (rabbit) 114882-65-4 γ-Neuropeptide (rabbit) can be extracted from rabbit intestine.
福沙吡坦二甲葡胺 V4400 FOSAPREPITANT DIMEGLUMINE 265121-04-8 Fosaprepitant dimeglumine (also known as L-758298 dimeglumine; MK0517 dimeglumine) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting.
罗拉吡坦盐酸盐水合物 V3304 Rolapitant HCl hydrate 914462-92-3 Rolapitant HCl hydrate (SCH619734; SCH-619734; SCH 619734; Varubi), the hydrochloride salt of Rolapitant, is a CNS penetreable and orally bioavailable antagonist of neurokinin (NK1) receptor (Ki = 0.66 nM) that was approved in 2015 to prevent delayed nausea and vomiting caused by cancer chemotherapy.
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