| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
|
V93135 | (R,R)-Suntinorexton | (R,R)-Suntinorexton is an isomer of Suntinorexton. | |
|
V69902 | (S,S)-J-113397 | 256640-46-7 | (S,S)-J-113397 is an enantiomer of J-113397. |
|
V69917 | [(pF)Phe4]Nociceptin(1-13)NH2 | 380620-88-2 | [(pF)Phe4]Nociceptin(1-13)NH2 is a highly efficient and selective NOP receptor (OP4) agonist/activator with pKi of 10.68 and pEC50 of 9.31. |
|
V69907 | [D-Ala2]-Met-Enkephalinamide | 61090-95-7 | [D-Ala2]-Met-Enkephalinamide is an opioid peptide and a potent opioid agonist. |
|
V69954 | Ac-RYYRIK-NH2 | 200959-48-4 | Ac-RYYRIK-NH2 is a potent ORL1 partial agonist that works as an endogenous ligand of ORL1 in CHO cells (Kd=1.5 nM). |
|
V102759 | Alvimopan metabolite hydrochloride | 170098-43-8 | Alvimopan metabolite hydrochloride is a peripherally restricted opioid receptor antagonist that inhibits the amplitude of electrically evoked contractions and spontaneous mechanical activity in the guinea pig ileum. |
|
V104966 | AP-238 | 140924-11-4 | AP-238 is a novel synthetic opioid (NSO) that acts as an agonist at the μ-opioid receptor (MOR) with an EC50 of 248 nM. |
|
V84961 | AT-035 | 2099680-55-2 | |
|
V86695 | Atoxifent | Atoxifent is a μ-opioid receptor agonist (EC50=0.39 nM), which is found in brain regions that control pain, mood, habit learning, and cognition. | |
|
V86698 | Bilaid A | 2393865-97-7 | Bilaid A is a μ-opioid receptor agonist extracted from Penicillium with a Ki value of 3.1 μM. |
|
V130425 | BNTX maleate | 864461-31-4 | BNTX maleate is a δ1-opioid receptor antagonist with Ki values of 0.1, 10.8, 13.3, and 58.6 nM for δ1, δ2, μ, and κ opioid receptors, respectively. |
|
V77133 | CTAP TFA | CTAP TFA is a specific, BBB (blood-brain barrier) permeable (penetrable) μ opioid receptor antagonist (inhibitor) with IC50 of 3.5 nM. | |
|
V77132 | CTOP TFA | CTOP TFA is a specific μ-opioid receptor antagonist. | |
|
V69895 | Cyprodime | 118111-54-9 | Cyprodime is a selective μ opioid receptor (MOR) antagonist (inhibitor) with Ki of 5.4, 244.6, and 2187 nM for μ, δ, and κ, respectively. |
|
V69901 | Cyprodime hydrochloride | 2387505-50-0 | Cyprodime HCl is a selective μ-opioid receptor antagonist (inhibitor) with Kis of 5.4 nM, 244.6 nM and 2187 nM for μ, δ and κ opioid receptors respectively. |
|
V77107 | DALDA acetate | DALDA acetate is a potent and selective μ-opioid receptor agonist/activator with a Ki of 1.69 nM. | |
|
V79008 | DALDA TFA | DALDA TFA is a potent and selective μ-opioid receptor agonist/activator with a Ki of 1.69 nM. | |
|
V120214 | DOR agonist 3 | 939956-07-7 | DOR agonist 3 (compound 10) is a selective δ-opioid receptor (DOR) positive allosteric modulator. |
|
V69882 | DPDPE | 88373-73-3 | DPDPE is an opioid peptide and a selective opioid receptor (DOR) agonist with anticonvulsant (antiepileptic/antiseizure) properties. |
|
V134789 | Dynorphin B (1-13) TFA | Dysorcinolone B (1-13) TFA can act as an agonist of opioid κ receptors. |